Search Count: 16
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Crystal Structure Of Brd9 Bromodomain In Complex With Compound Ea-89
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.76 Å Release Date: 2022-08-10 Classification: TRANSCRIPTION Ligands: L8L |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-08-10
Ligands: L8L
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Crystal Structure Of Egfr 696-1022 T790M In Complex With Ibrutinib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2017-12-27 Classification: ONCOPROTEIN Ligands: 1E8, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-12-27
Ligands: 1E8, CL
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Structure Of Dub Complex
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.27 Å Release Date: 2017-12-20 Classification: Hydrolase/Inhibitor Ligands: 9QD, ACT, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-12-20
Ligands: 9QD, ACT, GOL
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Structure Of Dub Complex
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2017-12-20 Classification: Hydrolase/Inhibitor Ligands: 9QA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-12-20
Ligands: 9QA
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Structure Of Dub Complex
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.33 Å Release Date: 2017-12-20 Classification: hydrolase/hydrolase inhibitor Ligands: 9HS, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-12-20
Ligands: 9HS, ZN
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Crystal Structure Of Sm1-71 Bound To Tak1-Tab1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.37 Å Release Date: 2017-02-15 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: 6H3 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-02-15
Ligands: 6H3
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Crystal Structure Of Tl11-113 Bound To Tak1-Tab1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2017-02-15 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: 6H4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-02-15
Ligands: 6H4
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Crystal Structure Of Cpt1691 Bound To Tak1-Tab1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.75 Å Release Date: 2017-02-15 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: 6HF |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-02-15
Ligands: 6HF
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Crystal Structure Of Tl10-92 Bound To Tak1-Tab1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.37 Å Release Date: 2017-02-15 Classification: Transferase/Transferase Inhibitor Ligands: T92 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-02-15
Ligands: T92
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Crystal Structure Of Tl11-128 Bound To Tak1-Tab1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.37 Å Release Date: 2017-02-15 Classification: Transferase/Transferase Inhibitor Ligands: 6L4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-02-15
Ligands: 6L4
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Crystal Structure Of Tl10-81 Bound To Tak1-Tab1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.11 Å Release Date: 2016-09-21 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: 5KW |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-09-21
Ligands: 5KW
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Crystal Structure Of Egfr 696-1022 T790M/V948R, Crystal Form Ii
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.97 Å Release Date: 2016-06-15 Classification: TRANSFERASE Ligands: ANP, MG, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-06-15
Ligands: ANP, MG, EDO
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Crystal Structure Of Egfr 696-1022 T790M In Complex With Ql-X138
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.30 Å Release Date: 2016-05-04 Classification: TRANSFERASE/INHIBITOR Ligands: 3LH, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-05-04
Ligands: 3LH, CL
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Crystal Structure Of The Human Ddr1 Kinase Domain In Complex With Ddr1-In-1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2014-01-15 Classification: TRANSFERASE Ligands: DI1, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-01-15
Ligands: DI1, EDO
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Discovery Of A Small Molecule Type Ii Inhibitor Of Wild-Type And Gatekeeper Mutants Of Bcr-Abl, Pdgfralpha, Kit, And Src Kinases
Organism: Gallus gallus
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2012-02-15 Classification: TRANSFERASE Ligands: NG7, MES, GOL |
Organism: Gallus gallus
Method: X-RAY DIFFRACTION
Release Date: 2012-02-15
Ligands: NG7, MES, GOL
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Human Abl Kinase In Complex With Nilotinib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.21 Å Release Date: 2008-04-22 Classification: TRANSFERASE Ligands: NIL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-04-22
Ligands: NIL
