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9I7Y image
Crystal Structure Of Krasg13C In Complex With Nucleotide-Based Covalent Inhibitor 7B
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.85 Å Release Date: 2025-11-12
Classification: HYDROLASE
Ligands: A1I08, MG

8S13 image
Apo C-Kit-Wt Kinase Domain
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.00 Å Release Date: 2025-09-03
Classification: TRANSFERASE
Ligands: EDO

8S14 image
C-Kit Kinase Domain In Complex With Sunitinib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.50 Å Release Date: 2025-09-03
Classification: TRANSFERASE
Ligands: B49, EDO, CL

8S15 image
C-Kit Kinase Domain In Complex With Nintedanib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.40 Å Release Date: 2025-09-03
Classification: TRANSFERASE
Ligands: XIN

8S16 image
C-Kit Kinase Domain In Complex With Imatinib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.85 Å Release Date: 2025-09-03
Classification: TRANSFERASE
Ligands: STI, CL

8S17 image
C-Kit Kinase Domain In Complex With Ponatinib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.20 Å Release Date: 2025-09-03
Classification: TRANSFERASE
Ligands: 0LI, CL

8S18 image
C-Kit Kinase Domain In Complex With S116836
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.10 Å Release Date: 2025-09-03
Classification: TRANSFERASE
Ligands: A1H4U, CL

8S19 image
C-Kit Kinase Domain In Complex With Staurosporine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.30 Å Release Date: 2025-09-03
Classification: TRANSFERASE
Ligands: STU

8S1A image
C-Kit Kinase Domain In Complex With Crenolanib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.85 Å Release Date: 2025-09-03
Classification: TRANSFERASE
Ligands: 6T2

8S1B image
C-Kit Kinase Domain In Complex With Idrx-42 Via Soaking
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.00 Å Release Date: 2025-09-03
Classification: TRANSFERASE
Ligands: K3R, CL

8C6P image
Fragment Screening Hit I Bound To Endothiapepsin
Organism: Cryphonectria parasitica
Method: X-RAY DIFFRACTION
Resolution:1.10 Å Release Date: 2023-05-24
Classification: HYDROLASE
Ligands: TT6, GOL

8C6Q image
Fragment Screening Hit Ii Bound To Endothiapepsin
Organism: Cryphonectria parasitica
Method: X-RAY DIFFRACTION
Resolution:1.25 Å Release Date: 2023-05-24
Classification: HYDROLASE
Ligands: GOL, TU5

8C6S image
Fragment Screening Hit Iii Bound To Endothiapepsin
Organism: Cryphonectria parasitica
Method: X-RAY DIFFRACTION
Resolution:1.10 Å Release Date: 2023-05-24
Classification: HYDROLASE
Ligands: GOL, TUU

8C6T image
Fragment Screening Hit Iv Bound To Endothiapepsin
Organism: Cryphonectria parasitica
Method: X-RAY DIFFRACTION
Resolution:1.15 Å Release Date: 2023-05-24
Classification: HYDROLASE
Ligands: GOL, TV6

8C70 image
Pyrrolidine Fragment 1 Bound To Endothiapepsin
Organism: Cryphonectria parasitica
Method: X-RAY DIFFRACTION
Resolution:1.65 Å Release Date: 2023-05-24
Classification: HYDROLASE
Ligands: TVI

8C71 image
Pyrrolidine Fragment 5B Bound To Endothiapepsin
Organism: Cryphonectria parasitica
Method: X-RAY DIFFRACTION
Resolution:1.10 Å Release Date: 2023-05-24
Classification: HYDROLASE
Ligands: GOL, TVO

8C72 image
Pyrrolidine Fragment 10B Bound To Endothiapepsin
Organism: Cryphonectria parasitica
Method: X-RAY DIFFRACTION
Resolution:1.20 Å Release Date: 2023-05-24
Classification: HYDROLASE
Ligands: GOL, TW0

8C74 image
Pyrrolidine Fragment 10D Bound To Endothiapepsin
Organism: Cryphonectria parasitica
Method: X-RAY DIFFRACTION
Resolution:1.15 Å Release Date: 2023-05-24
Classification: HYDROLASE
Ligands: GOL, TWX
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