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Search Count: 18

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9I7Y image
Crystal Structure Of Krasg13C In Complex With Nucleotide-Based Covalent Inhibitor 7B
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.85 Å Release Date: 2025-11-12
Classification: HYDROLASE
Ligands: A1I08, MG

8S13 image
Apo C-Kit-Wt Kinase Domain
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.00 Å Release Date: 2025-09-03
Classification: TRANSFERASE
Ligands: EDO

8S14 image
C-Kit Kinase Domain In Complex With Sunitinib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.50 Å Release Date: 2025-09-03
Classification: TRANSFERASE
Ligands: B49, EDO, CL

8S15 image
C-Kit Kinase Domain In Complex With Nintedanib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.40 Å Release Date: 2025-09-03
Classification: TRANSFERASE
Ligands: XIN

8S16 image
C-Kit Kinase Domain In Complex With Imatinib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.85 Å Release Date: 2025-09-03
Classification: TRANSFERASE
Ligands: STI, CL

8S17 image
C-Kit Kinase Domain In Complex With Ponatinib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.20 Å Release Date: 2025-09-03
Classification: TRANSFERASE
Ligands: 0LI, CL

8S18 image
C-Kit Kinase Domain In Complex With S116836

8S19 image
C-Kit Kinase Domain In Complex With Staurosporine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.30 Å Release Date: 2025-09-03
Classification: TRANSFERASE
Ligands: STU

8S1A image
C-Kit Kinase Domain In Complex With Crenolanib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.85 Å Release Date: 2025-09-03
Classification: TRANSFERASE
Ligands: 6T2

8S1B image
C-Kit Kinase Domain In Complex With Idrx-42 Via Soaking
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.00 Å Release Date: 2025-09-03
Classification: TRANSFERASE
Ligands: K3R, CL

8C6P image
Fragment Screening Hit I Bound To Endothiapepsin

8C6Q image
Fragment Screening Hit Ii Bound To Endothiapepsin

8C6S image
Fragment Screening Hit Iii Bound To Endothiapepsin

8C6T image
Fragment Screening Hit Iv Bound To Endothiapepsin

8C70 image
Pyrrolidine Fragment 1 Bound To Endothiapepsin

8C71 image
Pyrrolidine Fragment 5B Bound To Endothiapepsin

8C72 image
Pyrrolidine Fragment 10B Bound To Endothiapepsin

8C74 image
Pyrrolidine Fragment 10D Bound To Endothiapepsin
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