Search Count: 18
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Crystal Structure Of Krasg13C In Complex With Nucleotide-Based Covalent Inhibitor 7B
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2025-11-12 Classification: HYDROLASE Ligands: A1I08, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-11-12
Ligands: A1I08, MG
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Apo C-Kit-Wt Kinase Domain
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2025-09-03 Classification: TRANSFERASE Ligands: EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-09-03
Ligands: EDO
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C-Kit Kinase Domain In Complex With Sunitinib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2025-09-03 Classification: TRANSFERASE Ligands: B49, EDO, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-09-03
Ligands: B49, EDO, CL
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C-Kit Kinase Domain In Complex With Nintedanib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2025-09-03 Classification: TRANSFERASE Ligands: XIN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-09-03
Ligands: XIN
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C-Kit Kinase Domain In Complex With Imatinib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2025-09-03 Classification: TRANSFERASE Ligands: STI, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-09-03
Ligands: STI, CL
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C-Kit Kinase Domain In Complex With Ponatinib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2025-09-03 Classification: TRANSFERASE Ligands: 0LI, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-09-03
Ligands: 0LI, CL
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C-Kit Kinase Domain In Complex With S116836
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2025-09-03 Classification: TRANSFERASE Ligands: A1H4U, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-09-03
Ligands: A1H4U, CL
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C-Kit Kinase Domain In Complex With Staurosporine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2025-09-03 Classification: TRANSFERASE Ligands: STU |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-09-03
Ligands: STU
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C-Kit Kinase Domain In Complex With Crenolanib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2025-09-03 Classification: TRANSFERASE Ligands: 6T2 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-09-03
Ligands: 6T2
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C-Kit Kinase Domain In Complex With Idrx-42 Via Soaking
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2025-09-03 Classification: TRANSFERASE Ligands: K3R, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-09-03
Ligands: K3R, CL
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Fragment Screening Hit I Bound To Endothiapepsin
Organism: Cryphonectria parasitica
Method: X-RAY DIFFRACTION Resolution:1.10 Å Release Date: 2023-05-24 Classification: HYDROLASE Ligands: TT6, GOL |
Organism: Cryphonectria parasitica
Method: X-RAY DIFFRACTION
Release Date: 2023-05-24
Ligands: TT6, GOL
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Fragment Screening Hit Ii Bound To Endothiapepsin
Organism: Cryphonectria parasitica
Method: X-RAY DIFFRACTION Resolution:1.25 Å Release Date: 2023-05-24 Classification: HYDROLASE Ligands: GOL, TU5 |
Organism: Cryphonectria parasitica
Method: X-RAY DIFFRACTION
Release Date: 2023-05-24
Ligands: GOL, TU5
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Fragment Screening Hit Iii Bound To Endothiapepsin
Organism: Cryphonectria parasitica
Method: X-RAY DIFFRACTION Resolution:1.10 Å Release Date: 2023-05-24 Classification: HYDROLASE Ligands: GOL, TUU |
Organism: Cryphonectria parasitica
Method: X-RAY DIFFRACTION
Release Date: 2023-05-24
Ligands: GOL, TUU
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Fragment Screening Hit Iv Bound To Endothiapepsin
Organism: Cryphonectria parasitica
Method: X-RAY DIFFRACTION Resolution:1.15 Å Release Date: 2023-05-24 Classification: HYDROLASE Ligands: GOL, TV6 |
Organism: Cryphonectria parasitica
Method: X-RAY DIFFRACTION
Release Date: 2023-05-24
Ligands: GOL, TV6
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Pyrrolidine Fragment 1 Bound To Endothiapepsin
Organism: Cryphonectria parasitica
Method: X-RAY DIFFRACTION Resolution:1.65 Å Release Date: 2023-05-24 Classification: HYDROLASE Ligands: TVI |
Organism: Cryphonectria parasitica
Method: X-RAY DIFFRACTION
Release Date: 2023-05-24
Ligands: TVI
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Pyrrolidine Fragment 5B Bound To Endothiapepsin
Organism: Cryphonectria parasitica
Method: X-RAY DIFFRACTION Resolution:1.10 Å Release Date: 2023-05-24 Classification: HYDROLASE Ligands: GOL, TVO |
Organism: Cryphonectria parasitica
Method: X-RAY DIFFRACTION
Release Date: 2023-05-24
Ligands: GOL, TVO
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Pyrrolidine Fragment 10B Bound To Endothiapepsin
Organism: Cryphonectria parasitica
Method: X-RAY DIFFRACTION Resolution:1.20 Å Release Date: 2023-05-24 Classification: HYDROLASE Ligands: GOL, TW0 |
Organism: Cryphonectria parasitica
Method: X-RAY DIFFRACTION
Release Date: 2023-05-24
Ligands: GOL, TW0
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Pyrrolidine Fragment 10D Bound To Endothiapepsin
Organism: Cryphonectria parasitica
Method: X-RAY DIFFRACTION Resolution:1.15 Å Release Date: 2023-05-24 Classification: HYDROLASE Ligands: GOL, TWX |
Organism: Cryphonectria parasitica
Method: X-RAY DIFFRACTION
Release Date: 2023-05-24
Ligands: GOL, TWX
