Search Count: 25
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The Crystal Structure Of Apo-Ldhc
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.38 Å Release Date: 2025-09-03 Classification: STRUCTURAL PROTEIN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-09-03
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Crystal Structure Of Human Sirt5 In Complex With An Internally Quenched Fluorescent Substrate Gluiqf
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:1.39 Å Release Date: 2020-12-23 Classification: TRANSFERASE Ligands: ZN, NA, GUA |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2020-12-23
Ligands: ZN, NA, GUA
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Crystal Structure Of Human Sirt5 In Complex With The Fluorogenic Tetrapeptide Substrate P13
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:1.78 Å Release Date: 2020-10-28 Classification: TRANSFERASE Ligands: ZN, MCM |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2020-10-28
Ligands: ZN, MCM
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Crystal Structure Of Human Sirt5 In Complex With The Fluorogenic Tetrapeptide Substrate P15
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2020-10-28 Classification: HYDROLASE Ligands: ZN, MCM |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2020-10-28
Ligands: ZN, MCM
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Crystal Structure Of Human Kras G12C Covalently Bound To A Phthalazine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2019-12-25 Classification: SIGNALING PROTEIN/Inhibitor Ligands: MG, GDP, OJ1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-12-25
Ligands: MG, GDP, OJ1
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Crystal Structure Of Human Kras G12C Covalently Bound To A Quinazolinone Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2019-12-25 Classification: SIGNALING PROTEIN/Inhibitor Ligands: GDP, CA, OHY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-12-25
Ligands: GDP, CA, OHY
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Crystal Structure Of Zebra Fish Y-Box Protein1 (Yb-1) Cold-Shock Domain In Complex With 6Mer M5C Rna
Organism: Danio rerio, Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.26 Å Release Date: 2019-06-19 Classification: RNA BINDING PROTEIN/RNA Ligands: ZN |
Organism: Danio rerio, Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-06-19
Ligands: ZN
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Crystal Structure Of Human Pim-1 Kinase In Complex With A Quinazolinone-Pyrrolodihydropyrrolone Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2019-01-16 Classification: TRANSFERASE Ligands: JYG, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-01-16
Ligands: JYG, GOL
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Crystal Structure Of Sirt2 In Complex With Selective Inhibitor A2I
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2018-10-17 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: A2I, ZN, BME |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-10-17
Ligands: A2I, ZN, BME
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Crystal Structure Of Sirt2 In Complex With Selective Inhibitor A29
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.74 Å Release Date: 2018-10-17 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: ZN, A2X, BME |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-10-17
Ligands: ZN, A2X, BME
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Crystal Structure Of Sirt2 In Complex With Selective Inhibitor L55
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2018-10-17 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: ZN, L55, PEG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-10-17
Ligands: ZN, L55, PEG
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Crystal Structure Of Sirt2 In Complex With Selective Inhibitor L5C
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.48 Å Release Date: 2018-10-17 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: ZN, L5C |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-10-17
Ligands: ZN, L5C
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Crystal Structure Of Sirt5 Complexed With A Fluorogenic Small-Molecule Substrate Subka
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.19 Å Release Date: 2018-05-02 Classification: HYDROLASE Ligands: PHQ, SLL, MCM, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-05-02
Ligands: PHQ, SLL, MCM, ZN
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Crystal Structure Of Human Pim-1 Kinase In Complex With An Imidazopyridazine Inhibitor.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2016-11-09 Classification: transferase/transferase inhibitor Ligands: 6YN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-11-09
Ligands: 6YN
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Crystal Structure Of Human Pim-1 Kinase In Complex With A Quinazolinone-Pyrrolopyrrolone Inhibitor.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2016-06-22 Classification: transferase/transferase inhibitor Ligands: 6CD, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-06-22
Ligands: 6CD, GOL
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Crystal Structure Of Human Pim-1 Kinase In Complex With A Macrocyclic Quinoxaline-Pyrrolodihydropiperidinone Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2016-05-04 Classification: transferase/transferase inhibitor Ligands: 5QO, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-05-04
Ligands: 5QO, GOL
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Crystal Structure Of Human Pim-1 Kinase In Complex With A Thiazolamine-Indazole Inhibitor.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2015-02-11 Classification: transferase/transferase inhibitor Ligands: 3U5, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-02-11
Ligands: 3U5, GOL
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Crystal Structure Of Human Pim-1 Kinase In Complex With A Thiadiazolamine-Indole Inhibitor.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2015-02-11 Classification: transferase/transferase inhibitor Ligands: 3U6, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-02-11
Ligands: 3U6, GOL
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Co-Crystal Structure Of Pim1 With Compound 3
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.05 Å Release Date: 2015-02-04 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 3UR |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-02-04
Ligands: 3UR
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Crystal Structure Of Human Pim-1 Kinase In Complex With An Aminooxadiazole-Indole Inhibitor.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2015-02-04 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 38W, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-02-04
Ligands: 38W, GOL
