Search Count: 33
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Human Sarm1 Tir Domain Bound To Nb-3-Adpr
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.09 Å Release Date: 2022-09-21 Classification: HYDROLASE/INHIBITOR Ligands: Q1F |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-09-21
Ligands: Q1F
 |
Human Sarm1 Tir Domain Bound To An Nb-7-Adpr Adduct
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.96 Å Release Date: 2022-09-21 Classification: HYDROLASE/INHIBITOR Ligands: Q0L |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-09-21
Ligands: Q0L
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Human Sarm1 Tir Domain Bound To Nb-7
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.88 Å Release Date: 2022-09-21 Classification: HYDROLASE/INHIBITOR Ligands: Q0C |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-09-21
Ligands: Q0C
 |
Human Sarm1 Tir Domain Bound To Nb-2-Adpr
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.74 Å Release Date: 2022-09-21 Classification: HYDROLASE/INHIBITOR Ligands: Q0U |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-09-21
Ligands: Q0U
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Human Sarm1 Tir Domain Bound To Nb-3-Adprp
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.99 Å Release Date: 2022-09-21 Classification: HYDROLASE/INHIBITOR Ligands: Q1X |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-09-21
Ligands: Q1X
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Human Sarm1 Tir Domain Bound To Nb-3-Gdpr
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.37 Å Release Date: 2022-09-21 Classification: HYDROLASE/INHIBITOR Ligands: Q1O |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-09-21
Ligands: Q1O
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Human Sarm1 Bound To An Nb-3 Eadpr Adduct
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2022-09-21 Classification: HYDROLASE/INHIBITOR Ligands: PZ7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-09-21
Ligands: PZ7
 |
Apo Human Sarm1 Tir Domain
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.94 Å Release Date: 2022-09-21 Classification: HYDROLASE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-09-21
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Human Cd38 Ectodomain Bound To A 78C-Adpr Adduct
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.04 Å Release Date: 2022-09-21 Classification: HYDROLASE/INHIBITOR Ligands: Q2C |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-09-21
Ligands: Q2C
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Crystal Structure Of Human Kras G12C Covalently Bound To A Phthalazine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2019-12-25 Classification: SIGNALING PROTEIN/Inhibitor Ligands: MG, GDP, OJ1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-12-25
Ligands: MG, GDP, OJ1
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Crystal Structure Of Human Kras G12C Covalently Bound To A Quinazolinone Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2019-12-25 Classification: SIGNALING PROTEIN/Inhibitor Ligands: GDP, CA, OHY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-12-25
Ligands: GDP, CA, OHY
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Ire1 Kinase/Rnase In Complex With Imidazo[1,2-B]Pyridazin-8-Amine Compound 33
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.73 Å Release Date: 2019-02-27 Classification: SIGNALING PROTEIN Ligands: GUK |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-02-27
Ligands: GUK
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Ire1 Alpha In Complex With Imidazo[1,2-B]Pyridazin-8-Amine Compound 2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.14 Å Release Date: 2019-02-27 Classification: TRANSFERASE Ligands: GXK |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-02-27
Ligands: GXK
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Cct068127 In Complex With Cdk2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.30 Å Release Date: 2017-12-20 Classification: CELL CYCLE/INHIBITOR Ligands: 8QT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-12-20
Ligands: 8QT
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Multi-Parameter Lead Optimization To Give An Oral Chk1 Inhibitor Clinical Candidate: (R)-5-((4-((Morpholin-2-Ylmethyl)Amino)-5-(Trifluoromethyl)Pyridin-2-Yl)Amino)Pyrazine-2-Carbonitrile (Cct245737)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.91 Å Release Date: 2016-05-25 Classification: TRANSFERASE Ligands: 5UY, EDO, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-05-25
Ligands: 5UY, EDO, GOL
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Crystal Structure Of Mgamppcp-Bound Av2-Av1 Complex
Organism: Azotobacter vinelandii
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2015-02-25 Classification: OXIDOREDUCTASE Ligands: HCA, ICS, CLF, FE2, MG, ACP, SF4 |
Organism: Azotobacter vinelandii
Method: X-RAY DIFFRACTION
Release Date: 2015-02-25
Ligands: HCA, ICS, CLF, FE2, MG, ACP, SF4
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Structure Of Pka-Pkb Chimera Complexed With (1S)-2-Amino-1-(4- Chlorophenyl)-1-(4-(1H-Pyrazol-4-Yl)Phenyl)Ethan-1-Ol
Organism: Bos taurus, Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2012-07-25 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: RKD |
Organism: Bos taurus, Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-07-25
Ligands: RKD
 |
Crystal Structure Of Checkpoint Kinase 1 (Chk1) In Complex With Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.01 Å Release Date: 2012-01-11 Classification: TRANSFERASE Ligands: YM3, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-01-11
Ligands: YM3, EDO
 |
Crystal Structure Of Checkpoint Kinase 1 (Chk1) In Complex With Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.35 Å Release Date: 2012-01-11 Classification: TRANSFERASE Ligands: 4YM, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-01-11
Ligands: 4YM, EDO
 |
Crystal Structure Of Checkpoint Kinase 1 (Chk1) In Complex With Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.03 Å Release Date: 2012-01-11 Classification: TRANSFERASE Ligands: YM5, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-01-11
Ligands: YM5, EDO