Search Count: 38
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Macrocyclic Transition-State Mimicking Hiv-1 Protease Inhibitors Encompassing A Tertiary Alcohol
Organism: Human immunodeficiency virus
Method: X-RAY DIFFRACTION Resolution:2.35 Å Release Date: 2014-12-17 Classification: HYDROLASE Ligands: CL, 9MW |
Organism: Human immunodeficiency virus
Method: X-RAY DIFFRACTION
Release Date: 2014-12-17
Ligands: CL, 9MW
 |
Macrocyclic Transition-State Mimicking Hiv-1 Protease Inhibitors Encompassing A Tertiary Alcohol
Organism: Human immunodeficiency virus
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2014-12-17 Classification: HYDROLASE Ligands: CL, 378 |
Organism: Human immunodeficiency virus
Method: X-RAY DIFFRACTION
Release Date: 2014-12-17
Ligands: CL, 378
 |
Macrocyclic Transition-State Mimicking Hiv-1 Protease Inhibitors Encompassing A Tertiary Alcohol
Organism: Human immunodeficiency virus
Method: X-RAY DIFFRACTION Resolution:1.55 Å Release Date: 2014-12-17 Classification: HYDROLASE Ligands: CL, 1T8 |
Organism: Human immunodeficiency virus
Method: X-RAY DIFFRACTION
Release Date: 2014-12-17
Ligands: CL, 1T8
 |
Macrocyclic Transition-State Mimicking Hiv-1 Protease Inhibitors Encompassing A Tertiary Alcohol
Organism: Human immunodeficiency virus
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2014-12-17 Classification: HYDROLASE Ligands: CL, 1T8 |
Organism: Human immunodeficiency virus
Method: X-RAY DIFFRACTION
Release Date: 2014-12-17
Ligands: CL, 1T8
 |
Macrocyclic Transition-State Mimicking Hiv-1 Protease Inhibitors Encompassing A Tertiary Alcohol
Organism: Human immunodeficiency virus
Method: X-RAY DIFFRACTION Resolution:1.82 Å Release Date: 2014-12-17 Classification: HYDROLASE Ligands: CL, V78 |
Organism: Human immunodeficiency virus
Method: X-RAY DIFFRACTION
Release Date: 2014-12-17
Ligands: CL, V78
 |
Macrocyclic Transition-State Mimicking Hiv-1 Protease Inhibitors Encompassing A Tertiary Alcohol
Organism: Human immunodeficiency virus
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2014-12-17 Classification: HYDROLASE Ligands: CL, V78 |
Organism: Human immunodeficiency virus
Method: X-RAY DIFFRACTION
Release Date: 2014-12-17
Ligands: CL, V78
 |
Macrocyclic Transition-State Mimicking Hiv-1 Protease Inhibitors Encompassing A Tertiary Alcohol
Organism: Human immunodeficiency virus
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2014-12-17 Classification: HYDROLASE Ligands: CL, J3W |
Organism: Human immunodeficiency virus
Method: X-RAY DIFFRACTION
Release Date: 2014-12-17
Ligands: CL, J3W
 |
Macrocyclic Transition-State Mimicking Hiv-1 Protease Inhibitors Encompassing A Tertiary Alcohol
Organism: Human immunodeficiency virus
Method: X-RAY DIFFRACTION Resolution:2.45 Å Release Date: 2014-12-10 Classification: HYDROLASE Ligands: CL, M17 |
Organism: Human immunodeficiency virus
Method: X-RAY DIFFRACTION
Release Date: 2014-12-10
Ligands: CL, M17
 |
Macrocyclic Transition-State Mimicking Hiv-1 Protease Inhibitors Encompassing A Tertiary Alcohol
Organism: Human immunodeficiency virus
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2014-12-10 Classification: HYDROLASE Ligands: CL, 9MW |
Organism: Human immunodeficiency virus
Method: X-RAY DIFFRACTION
Release Date: 2014-12-10
Ligands: CL, 9MW
 |
Stereoselective Synthesis, X-Ray Analysis, And Biological Evaluation Of A New Class Of Lactam Based Hiv-1 Protease Inhibitors
Organism: Human immunodeficiency virus
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2012-11-07 Classification: HYDROLASE Ligands: UX9 |
Organism: Human immunodeficiency virus
Method: X-RAY DIFFRACTION
Release Date: 2012-11-07
Ligands: UX9
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Design And Synthesis Of Potent Hydroxyethylamine (Hea) Bace-1 Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2012-10-31 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 996 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-10-31
Ligands: 996
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Design And Synthesis Of Potent Hydroxyethylamine (Hea) Bace-1 Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2012-10-31 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 916 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-10-31
Ligands: 916
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Stereoselective Synthesis, X-Ray Analysis, And Biological Evaluation Of A New Class Of Lactam Based Hiv-1 Protease Inhibitors
Organism: Human immunodeficiency virus
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2012-05-09 Classification: HYDROLASE Ligands: QG8 |
Organism: Human immunodeficiency virus
Method: X-RAY DIFFRACTION
Release Date: 2012-05-09
Ligands: QG8
 |
Stereoselective Synthesis, X-Ray Analysis, And Biological Evaluation Of A New Class Of Lactam Based Hiv-1 Protease Inhibitors
Organism: Human immunodeficiency virus
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2012-05-09 Classification: HYDROLASE Ligands: QG9 |
Organism: Human immunodeficiency virus
Method: X-RAY DIFFRACTION
Release Date: 2012-05-09
Ligands: QG9
 |
Hiv-1 Inhibitors With A Tertiary-Alcohol-Containing Transition-State Mimic And Various P2 And P1 Prime Substituents
Organism: Human immunodeficiency virus 1 (z2/cdc-z34 isolate)
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2011-12-07 Classification: HYDROLASE Ligands: CXG |
Organism: Human immunodeficiency virus 1 (z2/cdc-z34 isolate)
Method: X-RAY DIFFRACTION
Release Date: 2011-12-07
Ligands: CXG
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Hiv-1 Inhibitors With A Tertiary-Alcohol-Containing Transition-State Mimic And Various P2 And P1 Prime Substituents
Organism: Human immunodeficiency virus 1 (z2/cdc-z34 isolate)
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2011-12-07 Classification: HYDROLASE Ligands: G40 |
Organism: Human immunodeficiency virus 1 (z2/cdc-z34 isolate)
Method: X-RAY DIFFRACTION
Release Date: 2011-12-07
Ligands: G40
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Potent Macrocyclic Renin Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2010-12-15 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: ACT, NA, 3OX, 3OW |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-12-15
Ligands: ACT, NA, 3OX, 3OW
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Potent Beta-Secretase 1 Hydroxyethylene Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2010-06-02 Classification: HYDROLASE Ligands: MV7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-06-02
Ligands: MV7
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Hcv Ns3/Ns4A Complexed With Non-Covalent Macrocyclic Compound Tmc435
Organism: Hepatitis c virus
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2010-03-09 Classification: HYDROLASE Ligands: 30B, ZN, GOL |
Organism: Hepatitis c virus
Method: X-RAY DIFFRACTION
Release Date: 2010-03-09
Ligands: 30B, ZN, GOL
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The Hcv Ns3/Ns4A Protease Apo Structure
Organism: Hepatitis c virus
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2010-03-09 Classification: HYDROLASE Ligands: ZN |
Organism: Hepatitis c virus
Method: X-RAY DIFFRACTION
Release Date: 2010-03-09
Ligands: ZN