Search Count: 34
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Crystal Structure Of Glucokinase In Complex With Compound 6
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2019-07-10 Classification: Transferase/Transferase Inhibitor Ligands: GLC, HKM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-07-10
Ligands: GLC, HKM
 |
Crystal Structure Of Glucokinase In Complex With Compound 72
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2019-07-10 Classification: Transferase/Transferase Inhibitor Ligands: GLC, DMS, HKG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-07-10
Ligands: GLC, DMS, HKG
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Discovery Of 2-Pyridyl Ureas As Glucokinase Activators
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2014-10-08 Classification: TRANSFERASE Ligands: GLC, 3LZ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-10-08
Ligands: GLC, 3LZ
 |
Highly Potent And Selective 3-N-Methylquinazoline-4(3H)-One Based Inhibitors Of B-Rafv600E Kinase
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.40 Å Release Date: 2014-04-09 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 2VX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-04-09
Ligands: 2VX
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Human B-Raf Kinase Domain In Complex With An Imidazopyridine-Based Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.60 Å Release Date: 2013-10-02 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: DFS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-10-02
Ligands: DFS
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Human Glucokinase In Complex With Novel Amino Thiazole Activator
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2013-09-25 Classification: TRANSFERASE/TRANSFERASE ACTIVATOR Ligands: GLC, VO1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-09-25
Ligands: GLC, VO1
 |
Human Glucokinase In Complex With A Novel Amino Thiazole Allosteric Activator
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2013-09-25 Classification: TRANSFERASE/TRANSFERASE ACTIVATOR Ligands: GLC, VO2 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-09-25
Ligands: GLC, VO2
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B-Raf Kinase Domain In Complex With An Aminothienopyrimidine-Based Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.30 Å Release Date: 2013-04-24 Classification: Transferase/Transferase Inhibitor Ligands: RI8 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-04-24
Ligands: RI8
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B-Raf Kinase Domain In Complex With An Aminopyridimine-Based Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.50 Å Release Date: 2013-04-24 Classification: Transferase/Transferase Inhibitor Ligands: RI9 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-04-24
Ligands: RI9
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Human B-Raf Kinase Domain Bound To A Type Ii Pyrazolopyridine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.50 Å Release Date: 2012-11-14 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 0WP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-11-14
Ligands: 0WP
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B-Raf V600E Kinase Domain Bound To A Type Ii Dihydroquinazoline Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.20 Å Release Date: 2012-11-14 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: B1E |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-11-14
Ligands: B1E
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Crystal Structure Of B-Raf Kinase Domain In Complex With A Dihydropyrido[2,3-D]Pyrimidinone-Based Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.60 Å Release Date: 2012-05-09 Classification: Transferase/Transferase Inhibitor Ligands: T1Q |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-05-09
Ligands: T1Q
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Human B-Raf Kinase Domain In Complex With An Bromopyridine Benzamide Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.40 Å Release Date: 2011-10-05 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: TV4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-10-05
Ligands: TV4
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Human B-Raf Kinase Domain In Complex With A Methoxypyrazolopyridinyl Benzamide Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.30 Å Release Date: 2011-10-05 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: B0R |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-10-05
Ligands: B0R
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Human B-Raf Kinase In Complex With An Amide Linked Pyrazolopyridine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.20 Å Release Date: 2011-08-17 Classification: Transferase/Transferase Inhibitor Ligands: BR2 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-08-17
Ligands: BR2
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Human B-Raf Kinase In Complex With A Furopyridine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.70 Å Release Date: 2011-02-02 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: FOI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-02-02
Ligands: FOI
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Human B-Raf Kinase In Complex With A Non-Oxime Furopyridine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.00 Å Release Date: 2011-02-02 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: FNI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-02-02
Ligands: FNI
 |
Crystal Structure Of Human B-Raf Kinase Domain In Complex With A Non-Oxime Furopyridine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2011-02-02 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: FP3 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-02-02
Ligands: FP3
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Crystal Structure Of Human B-Raf Kinase In Complex With A Non-Oxime Furopyridine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.50 Å Release Date: 2011-02-02 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: FP4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-02-02
Ligands: FP4
 |
Crystal Structure Of Human Akt1 With An Allosteric Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2010-10-13 Classification: TRANSFERASE Ligands: IQO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-10-13
Ligands: IQO