Search Count: 9
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Selectivity Switch Between Fak And Pyk2: Macrocyclization Of Fak Inhibitors Improves Pyk2 Potency
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.12 Å Release Date: 2017-11-29 Classification: Transferase/Transferase Inhibitor Ligands: YAM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-11-29
Ligands: YAM
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Selectivity Switch Between Fak And Pyk2: Macrocyclization Of Fak Inhibitors Improves Pyk2 Potency
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.98 Å Release Date: 2016-12-21 Classification: Transferase/Transferase Inhibitor Ligands: 7FM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-12-21
Ligands: 7FM
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Human Beta-Tryptase Ii With Inhibitor Cra-29382
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2006-03-21 Classification: HYDROLASE Ligands: C3A |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2006-03-21
Ligands: C3A
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Human Tryptase With 2-Amino Benzimidazole
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2006-03-07 Classification: HYDROLASE Ligands: AX7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2006-03-07
Ligands: AX7
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Human Beta Tryptase Ii With Inhibitor Cra-28427
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2006-03-07 Classification: HYDROLASE Ligands: C4A |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2006-03-07
Ligands: C4A
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Human Beta-Tryptase Ii Complexed With 4-Piperidinebutyrate To Make Acylenzyme
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.25 Å Release Date: 2006-02-14 Classification: HYDROLASE Ligands: C1R |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2006-02-14
Ligands: C1R
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Bovine Trypsin Bound By 4-Piperidinebutyrate To Make Acylenzyme Complex
Organism: Bos taurus
Method: X-RAY DIFFRACTION Resolution:1.65 Å Release Date: 2006-02-14 Classification: HYDROLASE Ligands: CA, C1R |
Organism: Bos taurus
Method: X-RAY DIFFRACTION
Release Date: 2006-02-14
Ligands: CA, C1R
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Bovine Trypsin Complexed With 2-Aminobenzamidazole
Organism: Bos taurus
Method: X-RAY DIFFRACTION Resolution:1.57 Å Release Date: 2006-02-14 Classification: HYDROLASE Ligands: CA, AX7 |
Organism: Bos taurus
Method: X-RAY DIFFRACTION
Release Date: 2006-02-14
Ligands: CA, AX7
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Human Beta Tryptase Ii Complexed With Activated Ketone Inhibitor Cra-29382
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2006-02-09 Classification: HYDROLASE Ligands: C3A |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2006-02-09
Ligands: C3A
