Search Count: 9
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Crystal Structure Of Human 11-Beta-Hydroxysteroid Dehydrogenase 1 (11B-Hsd1) In Complex With 4,4-Disubstituted Cyclohexylbenzamide Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2011-10-05 Classification: OXIDOREDUCTASE/OXIDOREDUCTASE INHIBITOR Ligands: 3PJ, NAP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-10-05
Ligands: 3PJ, NAP
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Crystal Structure Of 11Beta-Hydroxysteroid Dehydrogenase-1 (11B-Hsd1) In Complex With Diarylsulfone Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2011-07-20 Classification: OXIDOREDUCTASE/OXIDOREDUCTASE INHIBITOR Ligands: NAP, 3OQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-07-20
Ligands: NAP, 3OQ
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Crystal Structure Of 11Beta-Hydroxysteroid Dehydrogenase 1 (11B-Hsd1) In Complex With Benzamide Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.65 Å Release Date: 2009-12-01 Classification: OXIDOREDUCTASE Ligands: NAP, IIG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-12-01
Ligands: NAP, IIG
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Crystal Structure Of 11B-Hydroxysteroid Dehydrogenase-1 (11B-Hsd1) In Complex With Piperidyl Benzamide Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2009-06-16 Classification: OXIDOREDUCTASE Ligands: NAP, A49 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-06-16
Ligands: NAP, A49
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Further Studies With The 2-Amino-1,3-Thiazol-4(5H)-One Class Of 11-Hydroxysteroid Dehydrogenase Type 1 (11-Hsd1) Inhibitors: Reducing Pregnane X Receptor (Pxr) Activity And Exploring Activity In A Monkey Pharmacodynamic Model
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.00 Å Release Date: 2008-11-11 Classification: OXIDOREDUCTASE Ligands: NDP, 352 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-11-11
Ligands: NDP, 352
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Crystal Structure Of 11B-Hsd1 In Complex With Triazole Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.55 Å Release Date: 2008-10-07 Classification: OXIDOREDUCTASE Ligands: NAP, T30 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-10-07
Ligands: NAP, T30
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Crystal Structure Of Human 11-Beta-Hydroxysteroid Dehydrogenase (Hsd1) In Complex With Sulfonamide Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2008-07-22 Classification: OXIDOREDUCTASE Ligands: NAP, D4N |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-07-22
Ligands: NAP, D4N
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Crystal Structure Of Human 11-Beta-Hydroxysteroid Dehydrogenase (Hsd1) In Complex With Benzamide Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2008-07-01 Classification: OXIDOREDUCTASE Ligands: NAP, D3E |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-07-01
Ligands: NAP, D3E
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Crystal Structure Of Human 11-Beta-Hydroxysteroid Dehydrogenase (Hsd1) In Complex With Arylsulfonylpiperazine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.35 Å Release Date: 2008-06-17 Classification: OXIDOREDUCTASE Ligands: NAP, 3CZ, CPS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-06-17
Ligands: NAP, 3CZ, CPS