Search Count: 88
![]() |
Crystal Structure Of Apoform Human Usp18
Organism: Homo sapiens, Myxococcus xanthus (strain dk1622)
Method: X-RAY DIFFRACTION Resolution:1.92 Å Release Date: 2026-04-29 Classification: HYDROLASE Ligands: ZN |
Organism: Homo sapiens, Myxococcus xanthus (strain dk1622)
Method: X-RAY DIFFRACTION
Release Date: 2026-04-29
Ligands: ZN
![]() |
Crystal Structure Of Apoform Human Eif4A1 C-Terminal Domain
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.73 Å Release Date: 2026-02-18 Classification: TRANSLATION |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-02-18
![]() |
Crystal Structure Of Human Eif4A1 C-Terminal Domain In Complex With Hippuristanol
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2026-02-18 Classification: TRANSLATION Ligands: A1I1L |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-02-18
Ligands: A1I1L
![]() |
Crystal Structure Of Dhps In Complex With An Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.63 Å Release Date: 2024-11-20 Classification: TRANSFERASE Ligands: XTQ, EDO, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-11-20
Ligands: XTQ, EDO, DMS
![]() |
Crystal Structure Of Mnk2-D228G In Complex With Tinodasertib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.59 Å Release Date: 2024-06-12 Classification: TRANSFERASE Ligands: ZN, X8K |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-06-12
Ligands: ZN, X8K
![]() |
Crystal Structure Of Ternary Complex Of Pol Theta Polymerase Domain
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:2.26 Å Release Date: 2022-10-12 Classification: TRANSFERASE Ligands: MG, DG3 |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2022-10-12
Ligands: MG, DG3
![]() |
Crystal Structure Of Pol Theta Polymerase Domain In Complex With Compound 5
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:2.99 Å Release Date: 2022-10-12 Classification: TRANSFERASE Ligands: MG, DG3, K7X |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2022-10-12
Ligands: MG, DG3, K7X
![]() |
Crystal Structure Of Pol Theta Polymerase Domain In Complex With Compound 22
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:2.83 Å Release Date: 2022-10-12 Classification: TRANSFERASE Ligands: MG, DG3, K8I |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2022-10-12
Ligands: MG, DG3, K8I
![]() |
Crystal Structure Of Usp7 In Complex With The Non-Covalent Inhibitor, Ft671
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.35 Å Release Date: 2017-10-18 Classification: HYDROLASE Ligands: 8WK |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-10-18
Ligands: 8WK
![]() |
Crystal Structure Of Usp7 In Complex With The Covalent Inhibitor, Ft827
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.33 Å Release Date: 2017-10-18 Classification: HYDROLASE Ligands: 8WN, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-10-18
Ligands: 8WN, EDO
![]() |
Human Pfkfb3 In Complex With An Indole Inhibitor 1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.01 Å Release Date: 2015-04-22 Classification: TRANSFERASE Ligands: PO4, 8R2, FDP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-04-22
Ligands: PO4, 8R2, FDP
![]() |
Human Pfkfb3 In Complex With An Indole Inhibitor 2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2015-04-22 Classification: TRANSFERASE Ligands: PHS, PO4, F6P, S6L |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-04-22
Ligands: PHS, PO4, F6P, S6L
![]() |
Human Pfkfb3 In Complex With An Indole Inhibitor 3
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.58 Å Release Date: 2015-04-22 Classification: TRANSFERASE Ligands: PHS, PO4, F6P, FD9 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-04-22
Ligands: PHS, PO4, F6P, FD9
![]() |
Human Pfkfb3 In Complex With An Indole Inhibitor 4
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.37 Å Release Date: 2015-04-22 Classification: TRANSFERASE Ligands: PHS, PO4, F6P, 87T |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-04-22
Ligands: PHS, PO4, F6P, 87T
![]() |
Human Pfkfb3 In Complex With An Indole Inhibitor 5
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.35 Å Release Date: 2015-04-22 Classification: TRANSFERASE Ligands: PHS, F6P, PO4, MJP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-04-22
Ligands: PHS, F6P, PO4, MJP
![]() |
Human Pfkfb3 In Complex With An Indole Inhibitor 6
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.03 Å Release Date: 2015-04-22 Classification: TRANSFERASE Ligands: PHS, PO4, F6P, 8V1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-04-22
Ligands: PHS, PO4, F6P, 8V1
![]() |
Crystal Structure Of Human 17Beta-Hydroxysteroid Dehydrogenase Type 5 In Complex With (4-(4-Chlorophenyl)Piperazin-1-Yl)(Morpholino)Methanone (24)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2013-11-13 Classification: Oxidoreductase/Oxidoreductase inhibitor Ligands: NAP, 16J, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-11-13
Ligands: NAP, 16J, EDO
![]() |
Crystal Structure Of Human 17Beta-Hydroxysteroid Dehydrogenase Type 5 In Complex With 1-{4-[(2-Methyl-1-Piperidinyl)Sulfonyl]Phenyl}-2-Pyrrolidinone
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.97 Å Release Date: 2013-03-20 Classification: oxidoreductase/oxidoreductase inhibitor Ligands: NAP, 10H |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-03-20
Ligands: NAP, 10H
![]() |
Crystal Structure Of Human 17Beta-Hydroxysteroid Dehydrogenase Type 5 In Complex With (R)-1-(Naphthalen-2-Ylsulfonyl)Piperidine-3-Carboxylic Acid (86)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2012-10-10 Classification: OXIDOREDUCTASE/OXIDOREDUCTASE inhibitor Ligands: NAP, 0SL, EDO, ACT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-10-10
Ligands: NAP, 0SL, EDO, ACT
![]() |
Crystal Structure Of Human 17Beta-Hydroxysteroid Dehydrogenase Type 5 In Complex With 3-((3,4-Dihydroisoquinolin-2(1H)-Yl)Sulfonyl)-N-Methylbenzamide (80)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2012-10-10 Classification: oxidoreductase/oxidoreductase inhibitor Ligands: NAP, 0T0, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-10-10
Ligands: NAP, 0T0, EDO
