Search Count: 11
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Crystal Structure Of Human Monoacylglycerol Lipase In Complex With Compound 1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2021-08-11 Classification: HYDROLASE/INHIBITOR Ligands: XPD, ACT, MPD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-08-11
Ligands: XPD, ACT, MPD
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Crystal Structure Of Human Monoacylglycerol Lipase In Complex With Compound 1H
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.25 Å Release Date: 2021-08-11 Classification: HYDROLASE/INHIBITOR Ligands: XP7, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-08-11
Ligands: XP7, CL
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Crystal Structure Of Human Monoacylglycerol Lipase In Complex With Compound 2D
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2021-08-11 Classification: HYDROLASE/INHIBITOR Ligands: XOV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-08-11
Ligands: XOV
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Crystal Structure Of Human Monoacylglycerol Lipase In Complex With Compound 4F
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2021-08-11 Classification: HYDROLASE/INHIBITOR Ligands: ACT, XOM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-08-11
Ligands: ACT, XOM
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Crystal Structure Of Tyk2 With Novel Pyrrolidinone Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2020-02-12 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: N9G |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-02-12
Ligands: N9G
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Structure Of Rorgt In Complex With A Novel Isoquinoline Inverse Agonist.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.18 Å Release Date: 2018-03-21 Classification: transcription/agonist Ligands: MPD, E3S |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-03-21
Ligands: MPD, E3S
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Structure Of Rorgt In Complex With A Novel Inverse Agonist Tak-828.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.00 Å Release Date: 2018-03-21 Classification: transcription/agonist Ligands: MPD, E3V |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-03-21
Ligands: MPD, E3V
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Optimization Of 3,5-Disubstitued Piperidine: Discovery Of Non-Peptide Mimetics As An Orally Active Renin Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2017-10-18 Classification: HYDROLASE/HYDROLASE inhibitor Ligands: NAG, 7EK, PGE, PEG, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-10-18
Ligands: NAG, 7EK, PGE, PEG, DMS
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Optimization Of 3,5-Disubstitued Piperidine: Discovery Of Non-Peptide Mimetics As An Orally Active Renin Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.65 Å Release Date: 2017-10-18 Classification: HYDROLASE/HYDROLASE inhibitor Ligands: NAG, 7EJ, DMS, PEG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-10-18
Ligands: NAG, 7EJ, DMS, PEG
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Discovery Of Tak-272: A Novel, Potent And Orally Active Renin In-Hibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2017-07-05 Classification: HYDROLASE/HYDROLASE inhibitor Ligands: NAG, 6VU, PGE, PEG, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-07-05
Ligands: NAG, 6VU, PGE, PEG, DMS
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Discovery Of Tak-272: A Novel, Potent And Orally Active Renin In-Hibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.41 Å Release Date: 2016-11-16 Classification: HYDROLASE/HYDROLASE inhibitor Ligands: NAG, 6VS, DMS, PEG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-11-16
Ligands: NAG, 6VS, DMS, PEG
