Search Count: 19
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C-Terminal Bromodomain Of Human Brd2 With 5-(1-Benzyl-4-Chloro-1H-Imidazol-2-Yl)-1,3-Dimethylpyridin-2(1H)-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2024-06-26 Classification: TRANSCRIPTION Ligands: EDO, PE4, A1IBV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-06-26
Ligands: EDO, PE4, A1IBV
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N-Terminal Bromodomain Of Human Brd4 With (5-(4-Chloro-1-((Tetrahydro-2H-Pyran-4-Yl)Methyl)-1H-Imidazol-2-Yl)-1,3-Dimethylpyridin-2(1H)-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2024-06-26 Classification: TRANSCRIPTION Ligands: EDO, A1IB5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-06-26
Ligands: EDO, A1IB5
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N-Terminal Bromodomain Of Human Brd4 With I-Bet567
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.67 Å Release Date: 2022-12-14 Classification: TRANSCRIPTION Ligands: AKQ, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-12-14
Ligands: AKQ, EDO
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C-Terminal Bromodomain Of Human Brd2 With 7,8-Dimethoxy-3-Methyl-1,3-Dihydro-2H-Benzo[D]Azepin-2-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.62 Å Release Date: 2022-11-30 Classification: TRANSCRIPTION Ligands: EDO, P4M, MES |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-11-30
Ligands: EDO, P4M, MES
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C-Terminal Bromodomain Of Human Brd2 With (R)-7-((R)-1,2-Dihydroxyethyl)-1,3-Dimethyl-5-(1-Methyl-1H-Pyrazol-4-Yl)-1,3-Dihydro-2H-Benzo[D]Azepin-2-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2022-11-30 Classification: TRANSCRIPTION Ligands: EDO, 7PE, P4X |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-11-30
Ligands: EDO, 7PE, P4X
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C-Terminal Bromodomain Of Human Brd2 With 7,8-Dimethoxy-1,3-Dimethyl-1,3-Dihydro-2H-Benzo[D]Azepin-2-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2022-11-30 Classification: TRANSCRIPTION Ligands: EDO, PE4, P0U |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-11-30
Ligands: EDO, PE4, P0U
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C-Terminal Bromodomain Of Human Brd2 With 7,8-Dimethoxy-1,3-Dimethyl-1,3-Dihydro-2H-Benzo[D]Azepin-2-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2022-11-30 Classification: TRANSCRIPTION Ligands: EDO, PE4, P3R |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-11-30
Ligands: EDO, PE4, P3R
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Bromodomain Of Human Taf1 (2) With Naphthyridinone Compound
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.17 Å Release Date: 2021-10-13 Classification: TRANSCRIPTION Ligands: 5LV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-10-13
Ligands: 5LV
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Brd9 With 4-Chloro-2-Methyl-Methylamino-Pyridazinone
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2021-04-14 Classification: TRANSCRIPTION Ligands: 82I |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-04-14
Ligands: 82I
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Brd9 With Biphenyl-Methylamino-Dimethylpyridazinone
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.68 Å Release Date: 2021-03-24 Classification: TRANSCRIPTION Ligands: P8W |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-03-24
Ligands: P8W
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Brd9 With Methylpiperazinyl-Benzyl-Amino-Dimethylpyridazinone
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.68 Å Release Date: 2021-03-24 Classification: TRANSCRIPTION Ligands: P8Z |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-03-24
Ligands: P8Z
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N-Terminal Domain Of Brd4 With Biphenyl-Methyamino-Dimethylpyridazinone
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.39 Å Release Date: 2021-03-24 Classification: TRANSCRIPTION Ligands: P8W, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-03-24
Ligands: P8W, EDO
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Bromodomain Of Human Brd9 With 7-(3,4-Dimethoxyphenyl)-2-(4- Methanesulfonylpiperazine-1-Carbonyl)-5-Methyl-4H,5H-Thieno-3,2-C- Pyridin-4-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.30 Å Release Date: 2015-04-22 Classification: TRANSCRIPTION Ligands: N1D |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-04-22
Ligands: N1D
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Bromodomain Of Human Brd9 With 7-(3,4-Dimethoxyphenyl)-N-(1,1-Dioxo-1- Thian-4-Yl)-5-Methyl-4-Oxo-4H,5H-Thieno-3,2-C-Pyridine-2-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.64 Å Release Date: 2015-04-22 Classification: TRANSCRIPTION Ligands: TVU |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-04-22
Ligands: TVU
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Bromodomain Of Human Brd9 With N-(1,1-Dioxo-1-Thian-4-Yl)-5-Methyl-4- Oxo-7-3-(Trifluoromethyl)Phenyl-4H,5H-Thieno-3,2-C-Pyridine-2- Carboximidamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.72 Å Release Date: 2015-04-22 Classification: TRANSCRIPTION Ligands: EDO, XZB |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-04-22
Ligands: EDO, XZB
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Bromodomain Of Human Brd9 With N-(1,1-Dioxo-1-Thian-4-Yl)-5-Ethyl-4- Oxo-7-3-(Trifluoromethyl)Phenyl-4H,5H-Thieno-3,2-C-Pyridine-2- Carboximidamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.73 Å Release Date: 2015-04-22 Classification: TRANSCRIPTION Ligands: EDO, H1B |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-04-22
Ligands: EDO, H1B
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N-Terminal Bromodomain Of Human Brd4 With 7-(3,4-Dimethoxyphenyl)-N-(1,1-Dioxo-1-Thian-4-Yl)-5-Methyl-4-Oxo-4H,5H-Thieno-3,2-C-Pyridine-2- Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.58 Å Release Date: 2015-04-22 Classification: TRANSCRIPTION Ligands: CA, EDO, TVU |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-04-22
Ligands: CA, EDO, TVU
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N-Terminal Bromodomain Of Human Brd4 With N-(1,1-Dioxo-1-Thian-4-Yl)- 5-Methyl-4-Oxo-7-3-(Trifluoromethyl)Phenyl-4H,5H-Thieno-3,2-C- Pyridine-2-Carboximidamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.30 Å Release Date: 2015-04-22 Classification: TRANSCRIPTION Ligands: EDO, 5V2 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-04-22
Ligands: EDO, 5V2
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N-Terminal Bromodomain Of Human Brd4 With 7-(3,4-Dimethoxyphenyl)-2-(4-Methanesulfonylpiperazine-1-Carbonyl)-5-Methyl-4H,5H-Thieno-3,2-C- Pyridin-4-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.19 Å Release Date: 2015-04-22 Classification: TRANSCRIPTION Ligands: EDO, N1D |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-04-22
Ligands: EDO, N1D
