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Search Count: 10

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9TF3 image
Erap1 In Complex With (3S,4S)-1-(3-Cyano-6-Methylpyridin-2-Yl)-4-(Propan-2-Yl)Pyrrolidine-3-Carboxylic Acid

9TF4 image
Erap1 In Complex With (3R,4R)-1-(3-Cyano-6-Methylpyridin-2-Yl)-4-(Propan-2-Yl)Pyrrolidine-3-Carboxylic Acid

9TF6 image
Erap1 In Complex With (3R,4R)-1-[3-Cyano-6-(Cyclopropylamino)Pyridin-2-Yl]-4-(Propan-2-Yl)Pyrrolidine-3-Carboxylic Acid

9TFN image
Erap1 In Complex With (3R,4R)-1-{3-Cyano-4-Methyl-6-[(4-Methyloxan-4-Yl)Amino]Pyridin-2-Yl}-4-(Propan-2-Yl)Pyrrolidine-3-Carboxylic Acid

9GJN image
Erap1 In Complex With 1-[2-(3-Oxo-3,4-Dihydro-2H-1,4-Benzothiazin-4-Yl)Acetamido]Cyclohexane-1-Carboxylic Acid

9GJS image
Erap1 In Complex With 1-[2-(6-Bromo-3-Oxo-3,4-Dihydro-2H-1,4-Benzoxazin-4-Yl)Acetamido]-4,4-Difluorocyclohexane-1-Carboxylic Acid

9GK6 image
Erap1 In Complex With 1-[2-(6-Chloro-3-Oxo-3,4-Dihydro-2H-1,4-Benzothiazin-4-Yl)Acetamido]Cyclohexane-1-Carboxylic Acid

9GKE image
Erap1 In Complex With 1-[2-(2-Oxo-5-Phenyl-2,3-Dihydro-1,3-Benzothiazol-3-Yl)Acetamido]Cyclohexane-1-Carboxylic Acid

7Z28 image
High-Resolution Crystal Structure Of Erap1 With Bound Bestatin Analogue Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.55 Å Release Date: 2022-07-27
Classification: HYDROLASE
Ligands: NAG, ZN, I88, EDO, MLT, PGE

7ZYF image
Insulin Regulated Aminopeptidase (Irap) In Complex With A Nanomolar Alpha Hydroxy Beta Amino Acid Based Inhibitor.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.81 Å Release Date: 2022-07-20
Classification: HYDROLASE
Ligands: ZN, NAG, KFR, EDO, PEG, TRS
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