Search Count: 12
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Crystal Structure Of Bcl-Xl In Complex With A Small Molecule Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.96 Å Release Date: 2024-10-16 Classification: APOPTOSIS Ligands: A1AFG, CD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-10-16
Ligands: A1AFG, CD
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Crystal Structure Of Bcl-Xl In Complex With A Benzothiazole-Based Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.41 Å Release Date: 2021-06-23 Classification: APOPTOSIS Ligands: XZM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-06-23
Ligands: XZM
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Crystal Structure Of Bcl-2 In Complex With Prodrug Abbv-167
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:2.07 Å Release Date: 2021-04-14 Classification: APOPTOSIS Ligands: XZD |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2021-04-14
Ligands: XZD
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Crystal Structure Of Bcl-Xl In Complex With Tetrahydroisoquinoline-Pyridine Based Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2020-10-21 Classification: APOPTOSIS/APOPTOSIS INHIBITOR Ligands: RQ7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-10-21
Ligands: RQ7
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Crystal Structure Of Mcl-1 In Complex With A Bim Competitive Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.25 Å Release Date: 2017-10-04 Classification: signaling protein/inhibitor Ligands: CJY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-10-04
Ligands: CJY
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Crystal Structure Of Mcl-1 In Complex With A Bim Competitive Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2017-10-04 Classification: signaling protein/inhibitor Ligands: CN7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-10-04
Ligands: CN7
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Crystal Structure Of Mcl-1 In Complex With A Bim Competitive Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.31 Å Release Date: 2017-05-03 Classification: signaling protein/inhibitor Ligands: 9EA, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-05-03
Ligands: 9EA, ZN
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Discovery Of A Potent And Selective Bcl-Xl Inhibitor That Demonstrates Thrombocytopenia And Inhibits Tumor Growth In Vivo
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2015-07-22 Classification: APOPTOSIS/INHIBITOR Ligands: 3CQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-07-22
Ligands: 3CQ
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Bcl-Xl In Complex With Inhibitor (Compound 10)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2014-10-15 Classification: APOPTOSIS Ligands: 38H, EDO, ACT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-10-15
Ligands: 38H, EDO, ACT
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Discovery Of 3H-Benzo[4,5]Thieno[3,2-D]Pyrimidin-4-Ones As Potent, Highly Selective And Orally Bioavailable Pim Kinases Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2009-11-10 Classification: TRANSFERASE Ligands: LXG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-11-10
Ligands: LXG
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Discovery Of 3H-Benzo[4,5]Thieno[3,2-D]Pyrimidin-4-Ones As Potent, Highly Selective And Orally Bioavailable Pim Kinases Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2009-11-10 Classification: TRANSFERASE Ligands: LYG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-11-10
Ligands: LYG
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Discovery Of 3H-Benzo[4,5]Thieno[3,2-D]Pyrimidin-4-Ones As Potent, Highly Selective And Orally Bioavailable Pim Kinases Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2009-11-10 Classification: TRANSFERASE Ligands: LWG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-11-10
Ligands: LWG
