Search Count: 16
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Crystal Structure Of The High Affinity Heterodimer Of Hif2 Alpha And Arnt C-Terminal Pas Domains In Complex With A Tetrazole-Containing Antagonist
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2015-12-09 Classification: TRANSCRIPTION Ligands: 43L |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-12-09
Ligands: 43L
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Crystal Structure Of Pyruvate Dehydrogenase Kinase Isoform 2 In Complex With Inhibitor Pa1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.75 Å Release Date: 2014-01-01 Classification: Transferase/Transferase Inhibitor Ligands: PV1, TLA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-01-01
Ligands: PV1, TLA
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Crystal Structure Of Pyruvate Dehydrogenase Kinase Isoform 2 In Complex With Inhibitor Pa7
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2014-01-01 Classification: Transferase/Transferase Inhibitor Ligands: PFT, TLA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-01-01
Ligands: PFT, TLA
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Crystal Structure Of Pyruvate Dehydrogenase Kinase Isoform 2 In Complex With Inhibitor Ps2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2014-01-01 Classification: Transferase/Transferase Inhibitor Ligands: TLA, PV2 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-01-01
Ligands: TLA, PV2
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Crystal Structure Of Pyruvate Dehydrogenase Kinase Isoform 2 In Complex With Inhibitor Ps8
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2014-01-01 Classification: Transferase/Transferase Inhibitor Ligands: PV8, TLA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-01-01
Ligands: PV8, TLA
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Crystal Structure Of Pyruvate Dehydrogenase Kinase Isoform 2 In Complex With Inhibitor Ps10
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.75 Å Release Date: 2014-01-01 Classification: TRANSFERASE Ligands: PV0, TLA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-01-01
Ligands: PV0, TLA
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Crystal Structure Of Branched-Chain Alpha-Ketoacid Dehydrogenase Kinase In Complex With Alpha-Ketoisocaproic Acid And Adp
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2013-06-05 Classification: transferase/transferase inhibitor Ligands: ADP, COI, MG, K |
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION
Release Date: 2013-06-05
Ligands: ADP, COI, MG, K
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Crystal Structure Of Branched-Chain Alpha-Ketoacid Dehydrogenase Kinase/(R)-2-Chloro-3-Phenylpropanoic Acid Complex With Adp
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2013-06-05 Classification: transferase/transferase inhibitor Ligands: ADP, MG, K, WJ2 |
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION
Release Date: 2013-06-05
Ligands: ADP, MG, K, WJ2
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Crystal Structure Of Branched-Chain Alpha-Ketoacid Dehydrogenase Kinase/(R)-Alpha-Chloroisocaproate Complex With Adp
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2013-06-05 Classification: transferase/transferase inhibitor Ligands: ADP, MG, K, HRI |
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION
Release Date: 2013-06-05
Ligands: ADP, MG, K, HRI
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Crystal Structure Of The High Affinity Heterodimer Of Hif2 Alpha And Arnt C-Terminal Pas Domains In Complex With An Inactive Benzoxadiazole Antagonist
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.72 Å Release Date: 2013-04-03 Classification: TRANSCRIPTION Ligands: 0XB, PE8 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-04-03
Ligands: 0XB, PE8
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Crystal Structure Of Branched-Chain Alpha-Ketoacid Dehydrogenase Kinase/(S)-2-Chloro-3-Phenylpropanoic Acid Complex With Adp
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2013-03-27 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ADP, MG, K, WJ1 |
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION
Release Date: 2013-03-27
Ligands: ADP, MG, K, WJ1
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Crystal Structure Of The High Affinity Heterodimer Of Hif2 Alpha And Arnt C-Terminal Pas Domains In Complex With A Benzoxadiazole Antagonist
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2013-02-27 Classification: TRANSCRIPTION Ligands: 0X3 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-02-27
Ligands: 0X3
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Crystal Structure Of Branched-Chain Alpha-Ketoacid Dehydrogenase Kinase/S-Alpha-Chloroisocaproate Complex
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2012-10-03 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 03H |
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION
Release Date: 2012-10-03
Ligands: 03H
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Crystal Structure Of Branched-Chain Alpha-Ketoacid Dehydrogenase Kinase/Phenylbutyrate Complex
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION Resolution:2.85 Å Release Date: 2012-10-03 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: CLT |
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION
Release Date: 2012-10-03
Ligands: CLT
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Crystal Structure Of Branched-Chain Alpha-Ketoacid Dehydrogenase Kinase/S-Alpha-Chloroisocaproate Complex With Adp
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION Resolution:2.25 Å Release Date: 2012-10-03 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ADP, 03H, MG, K |
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION
Release Date: 2012-10-03
Ligands: ADP, 03H, MG, K
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Crystal Structure Of Branched-Chain Alpha-Ketoacid Dehydrogenase Kinase/Phenylbutyrate Complex With Adp
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2012-10-03 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ADP, MG, K, CLT |
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION
Release Date: 2012-10-03
Ligands: ADP, MG, K, CLT
