Search Count: 15
![]() |
Kras G12D (Gppcp) With Mrtx-1133
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.27 Å Release Date: 2022-03-16 Classification: HYDROLASE/INHIBITOR Ligands: 6IC, GCP, GDP, GOL, ACT, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-03-16
Ligands: 6IC, GCP, GDP, GOL, ACT, MG
![]() |
Identification Of The Clinical Development Candidate Mrtx849, A Covalent Krasg12C Inhibitor For The Treatment Of Cancer
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.27 Å Release Date: 2020-04-22 Classification: HYDROLASE/INHIBITOR Ligands: GDP, MG, M1R |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-22
Ligands: GDP, MG, M1R
![]() |
Identification Of The Clinical Development Candidate Mrtx849, A Covalent Krasg12C Inhibitor For The Treatment Of Cancer
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.03 Å Release Date: 2020-04-22 Classification: HYDROLASE/INHIBITOR Ligands: GDP, MG, QH4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-22
Ligands: GDP, MG, QH4
![]() |
Identification Of The Clinical Development Candidate Mrtx849, A Covalent Krasg12C Inhibitor For The Treatment Of Cancer
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.94 Å Release Date: 2020-04-22 Classification: HYDROLASE/INHIBITOR Ligands: GDP, MG, M1X |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-22
Ligands: GDP, MG, M1X
![]() |
Crystal Structure Of Glucokinase In Complex With Compound 6
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2019-07-10 Classification: Transferase/Transferase Inhibitor Ligands: GLC, HKM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-07-10
Ligands: GLC, HKM
![]() |
Crystal Structure Of Glucokinase In Complex With Compound 72
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2019-07-10 Classification: Transferase/Transferase Inhibitor Ligands: GLC, DMS, HKG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-07-10
Ligands: GLC, DMS, HKG
![]() |
Crystal Structure Of Erk2 In Complex With Compound 22
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.76 Å Release Date: 2016-07-06 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 6QB, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-07-06
Ligands: 6QB, EDO
![]() |
Crystal Structure Of Cdk2 In Complex With Compound 22
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2016-07-06 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 6QB |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-07-06
Ligands: 6QB
![]() |
Crystal Structure Of The Complex Of The Wild-Type Von Willebrand Factor A1 Domain And Glycoprotein Ib Alpha At 2.6 Angstrom Resolution
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2004-04-13 Classification: BLOOD CLOTTING |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2004-04-13
![]() |
Structure Of Bacillus Subtilis Nicotinic Acid Mononucleotide Adenylyl Transferase
Organism: Bacillus subtilis
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2002-07-12 Classification: TRANSFERASE |
Organism: Bacillus subtilis
Method: X-RAY DIFFRACTION
Release Date: 2002-07-12
![]() |
Structure Of Bacillus Subtilis Nicotinic Acid Mononucleotide Adenylyl Transferase
Organism: Bacillus subtilis
Method: X-RAY DIFFRACTION Resolution:3.20 Å Release Date: 2002-07-12 Classification: TRANSFERASE Ligands: DND |
Organism: Bacillus subtilis
Method: X-RAY DIFFRACTION
Release Date: 2002-07-12
Ligands: DND
![]() |
E.Coli Gdp-Mannose 4,6-Dehydratase
Organism: Escherichia coli
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 1999-11-24 Classification: LYASE |
Organism: Escherichia coli
Method: X-RAY DIFFRACTION
Release Date: 1999-11-24
![]() |
Gdp-Fucose Synthetase From Escherichia Coli Complex With Nadph
Organism: Escherichia coli
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 1999-08-26 Classification: OXIDOREDUCTASE Ligands: NDP |
Organism: Escherichia coli
Method: X-RAY DIFFRACTION
Release Date: 1999-08-26
Ligands: NDP
![]() |
Gdp-Fucose Synthetase From Escherichia Coli Complex With Nadp
Organism: Escherichia coli
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 1999-08-26 Classification: OXIDOREDUCTASE Ligands: NAP |
Organism: Escherichia coli
Method: X-RAY DIFFRACTION
Release Date: 1999-08-26
Ligands: NAP
![]() |
Gdp-Fucose Synthetase From E. Coli
Organism: Escherichia coli
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 1999-08-17 Classification: OXIDOREDUCTASE |
Organism: Escherichia coli
Method: X-RAY DIFFRACTION
Release Date: 1999-08-17
