Search Count: 119
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Structure Of Crbn:Ikzf2:Compound 15
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2025-09-03 Classification: IMMUNE SYSTEM Ligands: A1CBH, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-09-03
Ligands: A1CBH, ZN
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Structure Of Crbn:Ikzf2:Compound 35
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.34 Å Release Date: 2025-09-03 Classification: IMMUNE SYSTEM Ligands: A1CBG, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-09-03
Ligands: A1CBG, ZN
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Discovery Of Smd-3236, A Potent, Highly Selective And Efficacious Smarca2 Degrader For The Treatment Of Smarc4-Deficient Human Cancers
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.30 Å Release Date: 2025-08-20 Classification: TRANSCRIPTION Ligands: A1A1U |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-08-20
Ligands: A1A1U
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Structure Of Ikzf2:Crbn:Compound 5 Ternary Structure
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.86 Å Release Date: 2025-07-09 Classification: IMMUNE SYSTEM Ligands: A1CAC, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-07-09
Ligands: A1CAC, ZN
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Structure Of Crbn Tbd Bound To Compound C1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.42 Å Release Date: 2025-05-28 Classification: IMMUNE SYSTEM Ligands: A1CAV, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-05-28
Ligands: A1CAV, ZN
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Structure Of Crbn Tbd Bound To Compound C3
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.61 Å Release Date: 2025-05-28 Classification: IMMUNE SYSTEM Ligands: A1CAW, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-05-28
Ligands: A1CAW, ZN
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Pvtx-405: A Potent, Highly Selective, And Orally Efficacious Molecular Glue Degrader Of Ikzf2 For Cancer Immunotherapy
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.69 Å Release Date: 2025-05-14 Classification: TRANSCRIPTION Ligands: A1A8N, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-05-14
Ligands: A1A8N, ZN
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Discovery Of Potent, Highly Selective And Efficacious Smarca2 Degraders - Compound 11
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.26 Å Release Date: 2024-12-18 Classification: TRANSCRIPTION Ligands: A1BF5, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-12-18
Ligands: A1BF5, ZN
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Discovery Of Potent, Highly Selective And Efficacious Smarca2 Degraders - Compound 13
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.71 Å Release Date: 2024-12-18 Classification: TRANSCRIPTION Ligands: A1A1O, ZN, ACT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-12-18
Ligands: A1A1O, ZN, ACT
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Discovery Of Potent, Highly Selective And Efficacious Smarca2 Degraders - Compound 6
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.96 Å Release Date: 2024-12-18 Classification: TRANSCRIPTION Ligands: A1A1P, ZN, ACT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-12-18
Ligands: A1A1P, ZN, ACT
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Voltage-Gated Potassium Channel Kv3.1 With Novel Positive Modulator (9M)-9-{5-Chloro-6-[(3,3-Dimethyl-2,3-Dihydro-1-Benzofuran-4-Yl)Oxy]-4-Methylpyridin-3-Yl}-2-Methyl-7,9-Dihydro-8H-Purin-8-One (Compound 4)
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY Release Date: 2023-10-25 Classification: TRANSPORT PROTEIN Ligands: ZN, X9T, POV, K |
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY
Release Date: 2023-10-25
Ligands: ZN, X9T, POV, K
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Voltage-Gated Potassium Channel Kv3.1 Apo
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY Release Date: 2023-10-25 Classification: TRANSPORT PROTEIN Ligands: ZN, CLR, K |
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY
Release Date: 2023-10-25
Ligands: ZN, CLR, K
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Crystal Structure Of Stub1 With A Macrocyclic Peptide
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:1.79 Å Release Date: 2022-07-27 Classification: TRANSFERASE Ligands: I1J |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2022-07-27
Ligands: I1J
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Discovery Of An Anion-Dependent Farnesyltransferase Inhibitor From A Phenotypic Screen
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION Resolution:2.28 Å Release Date: 2021-09-08 Classification: TRANSFERASE/INHIBITOR Ligands: ACE, 60I, ZN, MG, PPV |
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION
Release Date: 2021-09-08
Ligands: ACE, 60I, ZN, MG, PPV
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Discovery Of An Anion-Dependent Farnesyltransferase Inhibitor From A Phenotypic Screen
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION Resolution:1.98 Å Release Date: 2021-09-08 Classification: TRANSFERASE/INHIBITOR Ligands: ACE, 60I, ZN, MG, DMA |
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION
Release Date: 2021-09-08
Ligands: ACE, 60I, ZN, MG, DMA
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Trimeric Human Arginase 1 In Complex With Mab1 - 2 Harg:3 Mab1 Complex
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY Release Date: 2021-09-01 Classification: HYDROLASE/IMMUNE SYSTEM |
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY
Release Date: 2021-09-01
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Trimeric Human Arginase 1 In Complex With Mab5
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY Release Date: 2021-09-01 Classification: HYDROLASE/IMMUNE SYSTEM Ligands: MN |
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY
Release Date: 2021-09-01
Ligands: MN
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Trimeric Human Arginase 1 In Complex With Mab1 - 2 Harg:2 Mab1 Complex
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY Release Date: 2021-09-01 Classification: HYDROLASE/IMMUNE SYSTEM Ligands: MN |
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY
Release Date: 2021-09-01
Ligands: MN
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Trimeric Human Arginase 1 In Complex With Mab2
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY Release Date: 2021-09-01 Classification: HYDROLASE/IMMUNE SYSTEM |
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY
Release Date: 2021-09-01
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Trimeric Human Arginase 1 In Complex With Mab3
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY Release Date: 2021-09-01 Classification: HYDROLASE/IMMUNE SYSTEM Ligands: MN |
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY
Release Date: 2021-09-01
Ligands: MN
