Search Count: 42
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Crystal Structure Of Humanised Cereblon From Magnetospirillum Gryphiswaldense Bound By Dihydrouracil-Indole Compound [1-(1H-Indol-6-Yl)Dihydro-2,4(1H,3H)-Pyrimidinedione].
Organism: Magnetospirillum gryphiswaldense
Method: X-RAY DIFFRACTION Resolution:1.39 Å Release Date: 2025-09-03 Classification: LIGASE Ligands: A1IMN, ZN |
Organism: Magnetospirillum gryphiswaldense
Method: X-RAY DIFFRACTION
Release Date: 2025-09-03
Ligands: A1IMN, ZN
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Crystal Structure Of The Smarca2 Bromodomain Bound To A Fragment Screening Hit
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.07 Å Release Date: 2025-06-18 Classification: GENE REGULATION Ligands: A1I5P, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-06-18
Ligands: A1I5P, ZN
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Crystal Structure Of The Smarca2 Bromodomain Bound To A Tricyclic Pyrimidoindolone Inhibitor (Compound 17)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.08 Å Release Date: 2025-05-14 Classification: GENE REGULATION Ligands: A1I45, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-05-14
Ligands: A1I45, ZN
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Discovery Of A Series Of Covalent, Cell Active Bfl-1 Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.56 Å Release Date: 2024-10-02 Classification: APOPTOSIS Ligands: A1IDP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-10-02
Ligands: A1IDP
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Discovery Of A Series Of Covalent, Cell Active Bfl-1 Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.68 Å Release Date: 2024-10-02 Classification: APOPTOSIS Ligands: A1IDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-10-02
Ligands: A1IDO
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Discovery Of A Series Of Covalent, Cell Active Bfl-1 Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.94 Å Release Date: 2024-10-02 Classification: APOPTOSIS Ligands: A1IDG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-10-02
Ligands: A1IDG
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Crystal Structure Of Mus81-Eme1, Apo Form.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.15 Å Release Date: 2024-07-03 Classification: HYDROLASE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-07-03
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Crystal Structure Of Mus81-Eme1 Bound By Compound 15.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.73 Å Release Date: 2024-07-03 Classification: HYDROLASE Ligands: MG, A1IA7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-07-03
Ligands: MG, A1IA7
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Crystal Structure Of Mus81-Eme1 Bound By Compound 16.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.02 Å Release Date: 2024-07-03 Classification: HYDROLASE Ligands: MG, EOH, A1IA8 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-07-03
Ligands: MG, EOH, A1IA8
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Crystal Structure Of Mus81-Eme1 Bound By Compound 10.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2024-06-19 Classification: HYDROLASE Ligands: A1IA5, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-06-19
Ligands: A1IA5, MG
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Crystal Structure Of Mus81-Eme1 Bound By Compound 12.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.91 Å Release Date: 2024-06-19 Classification: HYDROLASE Ligands: A1IA6, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-06-19
Ligands: A1IA6, MG
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Crystal Structure Of Mus81-Eme1 Bound By Compound 21.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.47 Å Release Date: 2024-06-19 Classification: HYDROLASE Ligands: MG, A1IA4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-06-19
Ligands: MG, A1IA4
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Structure Of The Human Ddb1-Dda1-Dcaf15 E3 Ubiquitin Ligase Bound To Compound Furan 12
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY Release Date: 2024-04-03 Classification: LIGASE Ligands: A1H17 |
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY
Release Date: 2024-04-03
Ligands: A1H17
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Structure Of The Human Ddb1-Dda1-Dcaf15 E3 Ubiquitin Ligase Bound To Compound Furan 24
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY Release Date: 2024-04-03 Classification: LIGASE Ligands: A1H18 |
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY
Release Date: 2024-04-03
Ligands: A1H18
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Crystal Structure Of D1228V C-Met Bound By Compound 29
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.77 Å Release Date: 2023-07-05 Classification: TRANSFERASE Ligands: GOL, EDO, FMT, W49 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-07-05
Ligands: GOL, EDO, FMT, W49
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Crystal Structure Of D1228V C-Met Bound By Compound 15
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.78 Å Release Date: 2023-07-05 Classification: TRANSFERASE Ligands: W3R, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-07-05
Ligands: W3R, CL
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Crystal Structure Of D1228V C-Met Bound By Compound 10
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2023-07-05 Classification: TRANSFERASE Ligands: W3W |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-07-05
Ligands: W3W
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Crystal Structure Of D1228V C-Met Bound By Compound 16
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.21 Å Release Date: 2023-07-05 Classification: TRANSFERASE Ligands: IOD, W3N |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-07-05
Ligands: IOD, W3N
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Crystal Structure Of Wild-Type C-Met Bound By Compound 2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.27 Å Release Date: 2023-07-05 Classification: TRANSFERASE Ligands: W40 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-07-05
Ligands: W40
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Crystal Structure Of D1228V C-Met Bound By Compound 2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.63 Å Release Date: 2023-07-05 Classification: TRANSFERASE Ligands: W40 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-07-05
Ligands: W40
