Search Count: 38
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Cdk2-Cycline1 In Complex With Allosteric Inhibitor I-198.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.84 Å Release Date: 2024-01-31 Classification: CELL CYCLE/TRANSFERASE/INHIBITOR Ligands: A1AC4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-01-31
Ligands: A1AC4
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Cdk2-Cycline1 In Complex With Allosteric Inhibitor I-125A.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2024-01-31 Classification: CELL CYCLE/TRANSFERASE/INHIBITOR Ligands: A1AC5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-01-31
Ligands: A1AC5
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Structure Of Sars-Cov-2 Mpro Lambda (G15S) In Complex With Nirmatrelvir (Pf-07321332)
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION Resolution:1.68 Å Release Date: 2022-03-09 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 4WI |
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION
Release Date: 2022-03-09
Ligands: 4WI
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Structure Of Sars-Cov-2 Mpro Mutant (K90R) In Complex With Nirmatrelvir (Pf-07321332)
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION Resolution:2.09 Å Release Date: 2022-03-09 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 4WI |
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION
Release Date: 2022-03-09
Ligands: 4WI
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Structure Of Sars-Cov-2 Mpro Omicron P132H In Complex With Nirmatrelvir (Pf-07321332)
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION Resolution:1.63 Å Release Date: 2022-01-26 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 4WI |
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION
Release Date: 2022-01-26
Ligands: 4WI
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Structure Of Sars-Cov-2 Main Protease In Complex With A Covalent Inhibitor
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION Resolution:1.63 Å Release Date: 2021-11-10 Classification: HYDROLASE/INHIBITOR Ligands: 4W8 |
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION
Release Date: 2021-11-10
Ligands: 4W8
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Structure Of Sars-Cov-2 Main Protease In Complex With A Covalent Inhibitor
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION Resolution:1.91 Å Release Date: 2021-11-10 Classification: HYDROLASE/INHIBITOR Ligands: 4WI |
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION
Release Date: 2021-11-10
Ligands: 4WI
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Structure Of Sars-Cov-2 Main Protease In Complex With A Covalent Inhibitor
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2021-11-10 Classification: HYDROLASE/INHIBITOR Ligands: 4YG |
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION
Release Date: 2021-11-10
Ligands: 4YG
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Structure Of Sars-Cov-2 Main Protease In Complex With A Covalent Inhibitor
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION Resolution:1.73 Å Release Date: 2021-11-10 Classification: HYDROLASE/INHIBITOR Ligands: 4WI |
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION
Release Date: 2021-11-10
Ligands: 4WI
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Crystal Structure Of Human Naa50 In Complex With A Cofactor Derived Inhibitor (Compound 1)
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:2.29 Å Release Date: 2020-07-01 Classification: TRANSFERASE/INHIBITOR Ligands: COA |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2020-07-01
Ligands: COA
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Crystal Structure Of Human Naa50 In Complex With A Truncated Cofactor Derived Inhibitor (Compound 2)
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:2.04 Å Release Date: 2020-07-01 Classification: TRANSFERASE/INHIBITOR Ligands: U44 |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2020-07-01
Ligands: U44
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Crystal Structure Of Human Naa50 In Complex With An Inhibitor (Compound 3) Identified Using Dna Encoded Library Technology
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.16 Å Release Date: 2020-07-01 Classification: TRANSFERASE/INHIBITOR Ligands: COA, U3V |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-07-01
Ligands: COA, U3V
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Crystal Structure Of Human Naa50 In Complex With Coa And An Inhibitor (Compound 4A) Identified Using Dna Encoded Library Technology
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.87 Å Release Date: 2020-07-01 Classification: TRANSFERASE Ligands: COA, U2J |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-07-01
Ligands: COA, U2J
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Crystal Structure Of Human Naa50 In Complex With Accoa And An Inhibitor (Compound 4A) Identified Using Dna Encoded Library Technology
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.07 Å Release Date: 2020-07-01 Classification: TRANSFERASE/INHIBITOR Ligands: ACO, U2J |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-07-01
Ligands: ACO, U2J
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Crystal Structure Of Human Naa50 In Complex With Accoa And An Inhibitor (Compound 4B) Identified Using Dna Encoded Library Technology
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2020-07-01 Classification: TRANSFERASE/INHIBITOR Ligands: ACO, U3Y |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-07-01
Ligands: ACO, U3Y
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Structure Of Hs/Acprc2 In Complex With 5,8-Dichloro-2-[(4-Methoxy-6-Methyl-2-Oxo-1,2-Dihydropyridin-3-Yl)Methyl]-7-[(R)-Methoxy(Oxetan-3-Yl)Methyl]-3,4-Dihydroisoquinolin-1(2H)-One
Organism: Anolis carolinensis, Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.81 Å Release Date: 2017-12-27 Classification: Transferase/Transferase Inhibitor Ligands: ZN, CJD |
Organism: Anolis carolinensis, Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-12-27
Ligands: ZN, CJD
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Discovery Of A Novel And Selective Ido-1 Inhibitor Pf-06840003 And Its Characterization As A Potential Clinical Candidate.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.28 Å Release Date: 2017-12-27 Classification: OXIDOREDUCTASE/Inhibitor Ligands: HEM, AOJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-12-27
Ligands: HEM, AOJ
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Structure Of Hs/Acprc2 In Complex With 5,8-Dichloro-7-(3,5-Dimethyl-1,2-Oxazol-4-Yl)-2-[(4,6-Dimethyl-2-Oxo-1,2-Dihydropyridin-3-Yl)Methyl]-3,4-Dihydroisoquinolin-1(2H)-One
Organism: Anolis carolinensis, Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.05 Å Release Date: 2017-12-27 Classification: METAL BINDING PROTEIN Ligands: ZN, CJG |
Organism: Anolis carolinensis, Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-12-27
Ligands: ZN, CJG
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Crystal Structure Of Mat2A Bound To The Allosteric Inhibitor Pf-02929366
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.06 Å Release Date: 2017-05-17 Classification: TRANSFERASE Ligands: 8AJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-05-17
Ligands: 8AJ
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Structure Of Human Anaplastic Lymphoma Kinase In Complex With 2-[(1R)-1-{[2-Amino-5-(1,3-Dimethyl-1H-Pyrazol-4-Yl)Pyridin-3-Yl]Oxy}Ethyl]-4-Fluoro-N,N-Dimethylbenzamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2016-08-17 Classification: Transferase/Transferase Inhibitor Ligands: 6YL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-08-17
Ligands: 6YL
