Search Count: 142
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X-Ray Structure Of Furin (Pcsk3) In Complex With The Biphenyl-Derived Compound 26 (Mi2456)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2025-12-24 Classification: HYDROLASE Ligands: A1JA6, CA, NA, CL, DMS, NAG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-12-24
Ligands: A1JA6, CA, NA, CL, DMS, NAG
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X-Ray Structure Of Furin (Pcsk3) In Complex With The Biphenyl-Derived Compound 42 (Mi2464)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2025-12-24 Classification: HYDROLASE Ligands: CA, NA, CL, DMS, NAG, A1JA1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-12-24
Ligands: CA, NA, CL, DMS, NAG, A1JA1
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X-Ray Structure Of Furin (Pcsk3) In Complex With The Biphenyl-Derived Compound 34 (Mi2470)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2025-12-24 Classification: HYDROLASE Ligands: CA, NA, CL, DMS, NAG, A1JA2 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-12-24
Ligands: CA, NA, CL, DMS, NAG, A1JA2
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X-Ray Structure Of Furin (Pcsk3) In Complex With The Biphenyl-Derived Compound 27 (Mi2471)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2025-12-24 Classification: HYDROLASE Ligands: A1JA3, CA, NA, CL, DMS, NAG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-12-24
Ligands: A1JA3, CA, NA, CL, DMS, NAG
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X-Ray Structure Of Furin (Pcsk3) In Complex With The Biphenyl-Derived Compound 13 (Mi3102)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.65 Å Release Date: 2025-12-24 Classification: HYDROLASE Ligands: CA, NA, CL, DMS, NAG, A1JA5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-12-24
Ligands: CA, NA, CL, DMS, NAG, A1JA5
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X-Ray Structure Of Furin (Pcsk3) In Complex With The Biphenyl-Derived Compound 24 (Mi3140)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2025-12-24 Classification: HYDROLASE Ligands: A1JA4, CA, NA, CL, DMS, NAG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-12-24
Ligands: A1JA4, CA, NA, CL, DMS, NAG
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Macrocyclic Inhibitors Targeting The Prime Site Of The Fibrinolytic Serine Protease Plasmin
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2024-10-30 Classification: HYDROLASE/INHIBITOR Ligands: A1AHR |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-10-30
Ligands: A1AHR
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X-Ray Structure Of Furin (Pcsk3) In Complex With Guanidinomethyl-Phac-Can-Tle-Can-6-(Aminomethyl)-3-Amino-Isoindol
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2024-03-13 Classification: HYDROLASE Ligands: CA, NA, CL, DMS |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2024-03-13
Ligands: CA, NA, CL, DMS
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X-Ray Structure Of Furin (Pcsk3) In Complex With Benzamidine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2023-10-04 Classification: HYDROLASE Ligands: BEN, CA, NA, CL, DMS, NAG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-10-04
Ligands: BEN, CA, NA, CL, DMS, NAG
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X-Ray Structure Of Furin (Pcsk3) In Complex With 1H-Isoindol-3-Amine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2023-10-04 Classification: HYDROLASE Ligands: F05, CA, NA, CL, DMS, NAG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-10-04
Ligands: F05, CA, NA, CL, DMS, NAG
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X-Ray Structure Of Furin (Pcsk3) In Complex With Guanidinomethyl-Phac-R-Tle-K-6-(Aminomethyl)-3-Amino-Isoindol
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2023-10-04 Classification: HYDROLASE Ligands: CA, NA, CL, DMS |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2023-10-04
Ligands: CA, NA, CL, DMS
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Crystal Structure Of Unlinked Ns2B-Ns3 Protease From Zika Virus In Complex With Inhibitor Mi-2230
Organism: Zika virus
Method: X-RAY DIFFRACTION Resolution:1.23 Å Release Date: 2023-06-14 Classification: VIRAL PROTEIN Ligands: KPO |
Organism: Zika virus
Method: X-RAY DIFFRACTION
Release Date: 2023-06-14
Ligands: KPO
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Crystal Structure Of Unlinked Ns2B-Ns3 Protease From Zika Virus In Complex With Inhibitor Mi-2259
Organism: Zika virus
Method: X-RAY DIFFRACTION Resolution:1.38 Å Release Date: 2023-05-31 Classification: VIRAL PROTEIN Ligands: JG0 |
Organism: Zika virus
Method: X-RAY DIFFRACTION
Release Date: 2023-05-31
Ligands: JG0
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Crystal Structure Of Unlinked Ns2B-Ns3 Protease From Zika Virus In Complex With Inhibitor Mi-2196
Organism: Zika virus
Method: X-RAY DIFFRACTION Resolution:1.75 Å Release Date: 2023-05-24 Classification: VIRAL PROTEIN Ligands: V7T, ZAL, V8N, 4CF, 3CF |
Organism: Zika virus
Method: X-RAY DIFFRACTION
Release Date: 2023-05-24
Ligands: V7T, ZAL, V8N, 4CF, 3CF
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Crystal Structure Of Unlinked Ns2B-Ns3 Protease From Zika Virus In Complex With Inhibitor Mi-2293
Organism: Zika virus
Method: X-RAY DIFFRACTION Resolution:1.40 Å Release Date: 2023-03-22 Classification: VIRAL PROTEIN Ligands: JVC |
Organism: Zika virus
Method: X-RAY DIFFRACTION
Release Date: 2023-03-22
Ligands: JVC
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Crystal Structure Of Unlinked Ns2B-Ns3 Protease From Zika Virus In Complex With Inhibitor Mi-2205
Organism: Zika virus
Method: X-RAY DIFFRACTION Resolution:1.52 Å Release Date: 2023-03-22 Classification: VIRAL PROTEIN Ligands: JVL |
Organism: Zika virus
Method: X-RAY DIFFRACTION
Release Date: 2023-03-22
Ligands: JVL
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Crystal Structure Of Unlinked Ns2B-Ns3 Protease From Zika Virus In Complex With Inhibitor Mi-2206
Organism: Zika virus
Method: X-RAY DIFFRACTION Resolution:1.68 Å Release Date: 2023-03-22 Classification: VIRAL PROTEIN Ligands: GOL, JW6 |
Organism: Zika virus
Method: X-RAY DIFFRACTION
Release Date: 2023-03-22
Ligands: GOL, JW6
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Crystal Structure Of Unlinked Ns2B-Ns3 Protease From Zika Virus In Complex With Inhibitor Mi-2128
Organism: Zika virus
Method: X-RAY DIFFRACTION Resolution:1.45 Å Release Date: 2023-03-22 Classification: VIRAL PROTEIN Ligands: JVU |
Organism: Zika virus
Method: X-RAY DIFFRACTION
Release Date: 2023-03-22
Ligands: JVU
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Crystal Structure Of Unlinked Ns2B-Ns3 Protease From Zika Virus In Complex With Inhibitor Mi-2130
Organism: Zika virus
Method: X-RAY DIFFRACTION Resolution:1.75 Å Release Date: 2023-03-22 Classification: VIRAL PROTEIN Ligands: JN9 |
Organism: Zika virus
Method: X-RAY DIFFRACTION
Release Date: 2023-03-22
Ligands: JN9
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Crystal Structure Of Unlinked Ns2B-Ns3 Protease From Zika Virus In Complex With Inhibitor Mi-2195
Organism: Zika virus
Method: X-RAY DIFFRACTION Resolution:1.69 Å Release Date: 2023-03-22 Classification: VIRAL PROTEIN Ligands: IBW |
Organism: Zika virus
Method: X-RAY DIFFRACTION
Release Date: 2023-03-22
Ligands: IBW
