Search Count: 10
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Crystal Structure Of Human Cdk13/Cyclin K In Complex With The Inhibitor Thz531
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.36 Å Release Date: 2021-05-12 Classification: TRANSCRIPTION Ligands: 5I1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-05-12
Ligands: 5I1
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Crystal Structure Of Human Cdk12/Cyclin K In Complex With The Inhibitor Bsj-01-175
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.00 Å Release Date: 2021-05-12 Classification: TRANSCRIPTION Ligands: UUB |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-05-12
Ligands: UUB
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Structure Of The (Sr) Ca2+-Atpase Bound To The Inhibitor Compound Cad204520 And Tnp-Atp
Organism: Oryctolagus cuniculus
Method: X-RAY DIFFRACTION Resolution:3.40 Å Release Date: 2020-05-20 Classification: HYDROLASE Ligands: 128, OHW, K |
Organism: Oryctolagus cuniculus
Method: X-RAY DIFFRACTION
Release Date: 2020-05-20
Ligands: 128, OHW, K
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Glycogen Synthase Kinase 3 Beta Complexed With Brd0209
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2018-03-14 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 6VK |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-03-14
Ligands: 6VK
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Glycogen Synthase Kinase 3 Beta Complexed With Brd0705
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2018-03-14 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 6VL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-03-14
Ligands: 6VL
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Glycogen Synthase Kinase 3 Beta Complexed With Brd3731
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.69 Å Release Date: 2018-03-14 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 6VM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-03-14
Ligands: 6VM
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Exploiting An Asp-Glu Switch In Glycogen Synthase Kinase 3 To Design Paralog Selective Inhibitors For Use In Acute Myeloid Leukemia
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.85 Å Release Date: 2018-02-21 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: 6VL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-02-21
Ligands: 6VL
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Non-Receptor Protein Tyrosine Phosphatase Shp2 F285S In Complex With Allosteric Inhibitor Jlr-2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.22 Å Release Date: 2017-12-13 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: DZJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-12-13
Ligands: DZJ
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X-Ray Crystal Structure Of Gsk3B In Complex With Chir99021
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.10 Å Release Date: 2016-05-25 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 65C, MG, MES |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-05-25
Ligands: 65C, MG, MES
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X-Ray Crystal Structure Of Gsk3B In Complex With Brd3937
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.45 Å Release Date: 2016-05-25 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 65A |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-05-25
Ligands: 65A
