Search Count: 82
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Human Cdk8/Cyclin-C Complex With Inhibitor 2-9
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.57 Å Release Date: 2025-01-22 Classification: TRANSCRIPTION Ligands: EDO, GOL, A1IS8, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-01-22
Ligands: EDO, GOL, A1IS8, DMS
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Human Cdk8/Cyclin-C Complex With Inhibitor 3-7
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.16 Å Release Date: 2025-01-22 Classification: TRANSCRIPTION Ligands: CL, EDO, GOL, A1ITF, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-01-22
Ligands: CL, EDO, GOL, A1ITF, DMS
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Human Pi4Kiiib In Complex With Covalently Bound Inhibitor (Compound 4)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.51 Å Release Date: 2023-12-13 Classification: TRANSFERASE Ligands: KHR, MG, EDO, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-12-13
Ligands: KHR, MG, EDO, GOL
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Human Pi4Kiiib In Complex With Covalently Bound Inhibitor (Compound 8)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.54 Å Release Date: 2023-12-13 Classification: TRANSFERASE Ligands: KIH, MG, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-12-13
Ligands: KIH, MG, EDO
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Human Pi4Kiiib In Complex With Covalently Bound Inhibitor (Compound 11)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.94 Å Release Date: 2023-12-13 Classification: TRANSFERASE Ligands: MG, KI7, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-12-13
Ligands: MG, KI7, EDO
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Crystal Structure Of Prostaglandin D2 Synthase In Complex With Fragment 1A At 1.84A Resolution.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.84 Å Release Date: 2021-07-28 Classification: ISOMERASE Ligands: GSH, MG, QPN, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-07-28
Ligands: GSH, MG, QPN, GOL
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H-Pdgs Complexed With A 2-Phenylimidazo[1,2-A]Pyridine-6-Carboxamide Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.88 Å Release Date: 2021-05-26 Classification: Isomerase, Transferase/Inhibitor Ligands: GSH, VH4, MG, NA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-05-26
Ligands: GSH, VH4, MG, NA
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H-Pdgs Complexed With A 2-Phenylimidazo[1,2-A]Pyridine-6-Carboxamide Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.13 Å Release Date: 2021-05-26 Classification: Isomerase, Transferase/Inhibitor Ligands: CL, EDO, GSH, VH7, MG, NA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-05-26
Ligands: CL, EDO, GSH, VH7, MG, NA
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Hpgds Complexed With A Quinoline-3-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.65 Å Release Date: 2019-03-27 Classification: HYDROLASE Ligands: GSH, KCD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-03-27
Ligands: GSH, KCD
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Rat Hpgds Complexed With A Quinoline
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2019-03-27 Classification: HYDROLASE Ligands: GSH, KDV |
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION
Release Date: 2019-03-27
Ligands: GSH, KDV
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Crystal Structure Of Spleen Tyrosine Kinase (Syk) In Complex With A 2-(Pyridinyloxymethyl)Pyridine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2018-10-10 Classification: TRANSFERASE Ligands: GDK, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-10-10
Ligands: GDK, GOL
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Crystal Structure Of Spleen Tyrosine Kinase (Syk) In Complex With A 2-(Phenoxymethyl)Pyridine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.64 Å Release Date: 2018-10-10 Classification: TRANSFERASE Ligands: GDH, BR, GOL, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-10-10
Ligands: GDH, BR, GOL, DMS
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Crystal Structure Of Human Lipoprotein-Associated Phospholipase A2 In Complex With A [1.1.1]Bicyclopentane-Containing Inhibitor At 1.91A Resolution.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.91 Å Release Date: 2017-02-01 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: CL, 71H |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-02-01
Ligands: CL, 71H
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Fragment-Based Inhibitors Of Lipoprotein Associated Phospholipase A2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.17 Å Release Date: 2016-12-21 Classification: HYDROLASE Ligands: 7BJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-12-21
Ligands: 7BJ
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Fragment-Based Inhibitors Of Lipoprotein Associated Phospholipase A2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2016-12-21 Classification: HYDROLASE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-12-21
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Fragment-Based Inhibitors Of Lipoprotein Associated Phospholipase A2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.07 Å Release Date: 2016-12-21 Classification: HYDROLASE Ligands: CL, 7BW |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-12-21
Ligands: CL, 7BW
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Fragment-Based Inhibitors Of Lipoprotein Associated Phospholipase A2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2016-12-21 Classification: HYDROLASE Ligands: CL, 7K4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-12-21
Ligands: CL, 7K4
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Fragment-Based Inhibitors Of Lipoprotein Associated Phospholipase A2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2016-12-21 Classification: HYDROLASE Ligands: CL, 7BK |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-12-21
Ligands: CL, 7BK
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Fragment-Based Inhibitors Of Lipoprotein Associated Phospholipase A2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.11 Å Release Date: 2016-12-21 Classification: HYDROLASE Ligands: CL, 7BP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-12-21
Ligands: CL, 7BP
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Fragment-Based Inhibitors Of Lipoprotein Associated Phospholipase A2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.06 Å Release Date: 2016-12-21 Classification: HYDROLASE Ligands: CL, NA, 7BR |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-12-21
Ligands: CL, NA, 7BR
