Search Count: 23
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Structure Enabled Discovery Of A Stapled Peptide Inhibitor To Target The Oncogenic Transcriptional Repressor Tle1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.04 Å Release Date: 2017-04-05 Classification: TRANSCRIPTION Ligands: DMS, EBU |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-04-05
Ligands: DMS, EBU
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Rapid Discovery Of Pyrido[3,4-D]Pyrimidine Inhibitors Of Monopolar Spindle Kinase 1 (Mps1) Using A Structure-Based Hydridization Approach
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.66 Å Release Date: 2016-11-09 Classification: TRANSFERASE Ligands: 0SQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-11-09
Ligands: 0SQ
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Rapid Discovery Of Pyrido[3,4-D]Pyrimidine Inhibitors Of Monopolar Spindle Kinase 1 (Mps1) Using A Structure-Based Hydridization Approach
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.18 Å Release Date: 2016-11-09 Classification: TRANSFERASE Ligands: 5O1, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-11-09
Ligands: 5O1, DMS
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Rapid Discovery Of Pyrido[3,4-D]Pyrimidine Inhibitors Of Monopolar Spindle Kinase 1 (Mps1) Using A Structure-Based Hydridization Approach
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.18 Å Release Date: 2016-04-20 Classification: TRANSFERASE Ligands: 5NW, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-04-20
Ligands: 5NW, DMS
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Rapid Discovery Of Pyrido[3,4-D]Pyrimidine Inhibitors Of Monopolar Spindle Kinase 1 (Mps1) Using A Structure-Based Hydridization Approach
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.26 Å Release Date: 2016-04-20 Classification: TRANSFERASE Ligands: 7PE, 5O4, EDO, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-04-20
Ligands: 7PE, 5O4, EDO, DMS
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Rapid Discovery Of Pyrido[3,4-D]Pyrimidine Inhibitors Of Monopolar Spindle Kinase 1 (Mps1) Using A Structure-Based Hydridization Approach
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.67 Å Release Date: 2016-04-20 Classification: TRANSFERASE Ligands: 5O7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-04-20
Ligands: 5O7
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Rapid Discovery Of Pyrido[3,4-D]Pyrimidine Inhibitors Of Monopolar Spindle Kinase 1 (Mps1) Using A Structure-Based Hydridization Approach
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.01 Å Release Date: 2016-04-20 Classification: TRANSFERASE Ligands: 5OQ, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-04-20
Ligands: 5OQ, DMS
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Rapid Discovery Of Pyrido[3,4-D]Pyrimidine Inhibitors Of Monopolar Spindle Kinase 1 (Mps1) Using A Structure-Based Hydridization Approach
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.17 Å Release Date: 2016-04-20 Classification: TRANSFERASE Ligands: 5OE, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-04-20
Ligands: 5OE, DMS
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Nek2-Ede Bound To Cct248662
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2012-04-25 Classification: TRANSFERASE Ligands: JUP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-04-25
Ligands: JUP
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Nek2 Bound To Hybrid Compound 21
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2012-04-25 Classification: TRANSFERASE Ligands: GGY, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-04-25
Ligands: GGY, EDO
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Structure Of Nek2 Bound To Cct
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2011-03-30 Classification: TRANSFERASE Ligands: WGZ, EDO, CL, TRS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-03-30
Ligands: WGZ, EDO, CL, TRS
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Structure Of Nek2 Bound To Cct242430
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2011-03-30 Classification: TRANSFERASE Ligands: 430, CL, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-03-30
Ligands: 430, CL, EDO
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Structure Of Nek2 Bound To Cct243779
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.98 Å Release Date: 2011-03-30 Classification: TRANSFERASE Ligands: ED8, CL, EDO, GOL, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-03-30
Ligands: ED8, CL, EDO, GOL, DMS
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Structure Of Nek2 Bound To Cct244858
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.98 Å Release Date: 2011-03-30 Classification: TRANSFERASE Ligands: WCX, CL, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-03-30
Ligands: WCX, CL, EDO
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Structure Of Nek2 Bound To Aminipyrazine Compound 5
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2010-11-03 Classification: TRANSFERASE Ligands: WI2, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-11-03
Ligands: WI2, CL
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Structure Of Nek2 Bound To Aminopyrazine Compound 35
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2010-10-27 Classification: TRANSFERASE Ligands: XK3, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-10-27
Ligands: XK3, CL
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Structure Of Nek2 Bound To Aminopyrazine Compound 17
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2010-10-27 Classification: TRANSFERASE Ligands: OL2, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-10-27
Ligands: OL2, CL
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Structure Of Nek2 Bound To Aminopyrazine Compound 36
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2010-10-27 Classification: TRANSFERASE Ligands: EQH, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-10-27
Ligands: EQH, CL
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Structure Of Nek2 Bound To Aminopyrazine Compound 23
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.99 Å Release Date: 2010-10-27 Classification: TRANSFERASE Ligands: 30E, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-10-27
Ligands: 30E, CL
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Structure Of Nek2 Bound To Aminopyrazine Compound 15
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2010-10-27 Classification: TRANSFERASE Ligands: 5R1, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-10-27
Ligands: 5R1, CL
