Search Count: 15
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N-Terminal Bromodomain Of Human Brd4 With I-Bet567
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.67 Å Release Date: 2022-12-14 Classification: TRANSCRIPTION Ligands: AKQ, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-12-14
Ligands: AKQ, EDO
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N-Terminal Bromodomain Of Human Brd4 With I-Bet282
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2021-10-13 Classification: TRANSCRIPTION Ligands: EDO, UYK |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-10-13
Ligands: EDO, UYK
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N-Terminal Bromodomain Of Human Brd4 With 1-(2R,4S)-2-Methyl-4-(Phenylamino)-6-4-(Piperidin-1-Ylmethyl)Phenyl-1,2,3,4- Tetrahydroquinolin-1-Yl-Ethan-1-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.01 Å Release Date: 2015-10-07 Classification: TRANSCRIPTION Ligands: EDO, 9S3 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-10-07
Ligands: EDO, 9S3
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The Kinase Domain Of Human Spleen Tyrosine (Syk) In Complex With Gtc000222
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2015-09-30 Classification: TRANSFERASE Ligands: 4DF, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-09-30
Ligands: 4DF, GOL
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The Kinase Domain Of Human Spleen Tyrosine (Syk) In Complex With Gtc000223
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.83 Å Release Date: 2015-09-30 Classification: TRANSFERASE Ligands: 4DL, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-09-30
Ligands: 4DL, DMS
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Syk Kinase Domain In Complex With Inhibitor Gtc000224
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.34 Å Release Date: 2015-09-30 Classification: TRANSFERASE Ligands: 4DK |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-09-30
Ligands: 4DK
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Syk Kinase Domain In Complex With Inhibitor Gtc000225
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.32 Å Release Date: 2015-09-30 Classification: TRANSFERASE Ligands: 4DJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-09-30
Ligands: 4DJ
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The Kinase Domain Of Human Spleen Tyrosine (Syk) In Complex With Gtc000226
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.22 Å Release Date: 2015-09-30 Classification: TRANSFERASE Ligands: 4DN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-09-30
Ligands: 4DN
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The Kinase Domain Of Human Spleen Tyrosine (Syk) In Complex With Gtc000233
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.52 Å Release Date: 2015-09-30 Classification: TRANSFERASE Ligands: GOL, 4DQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-09-30
Ligands: GOL, 4DQ
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The Kinase Domain Of Human Spleen Tyrosine (Syk) In Complex With Gtc000249
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.67 Å Release Date: 2015-09-30 Classification: TRANSFERASE Ligands: 4DO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-09-30
Ligands: 4DO
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N-Terminal Bromodomain Of Human Brd4 With I-Bet295
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.40 Å Release Date: 2014-12-24 Classification: TRANSCRIPTION Ligands: EDO, IES |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-12-24
Ligands: EDO, IES
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N-Terminal Bromodomain Of Human Brd4 With Ibet-295
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2014-12-24 Classification: TRANSCRIPTION Ligands: EDO, 83T |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-12-24
Ligands: EDO, 83T
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Discovery Of Epigenetic Regulator I-Bet762: Lead Optimization To Afford A Clinical Candidate Inhibitor Of The Bet Bromodomains
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.87 Å Release Date: 2013-10-02 Classification: CELL CYCLE Ligands: H4C |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-10-02
Ligands: H4C
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Discovery Of Epigenetic Regulator I-Bet762: Lead Optimization To Afford A Clinical Candidate Inhibitor Of The Bet Bromodomains
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.55 Å Release Date: 2013-10-02 Classification: CELL CYCLE Ligands: L5S, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-10-02
Ligands: L5S, EDO
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Crystal Structure Of Spleen Tyrosine Kinase (Syk) In Complex With A Diaminopyrimidine Carboxamide Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2011-09-21 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: S19, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-09-21
Ligands: S19, GOL