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8GC7 image
Bruton'S Tyrosine Kinase In Complex With 5-(Piperidin-1-Yl)-3-{[4-(Piperidin-4-Yl)Phenyl]Amino}Pyrazine-2-Carboxamide

8GC8 image
Bruton'S Tyrosine Kinase L528W Mutant In Complex With 5-(Piperidin-1-Yl)-3-{[4-(Piperidin-4-Yl)Phenyl]Amino}Pyrazine-2-Carboxamide

8EJB image
Bruton'S Tyrosine Kinase In Complex With 3-{[4-(1-Acetylpiperidin-4-Yl)Phenyl]Amino}-5-[(3R)-3-(3-Methyl-2-Oxoimidazolidin-1-Yl)Piperidin-1-Yl]Pyrazine-2-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.58 Å Release Date: 2023-02-15
Classification: TRANSFERASE
Ligands: WKC, EDO, PD, CL


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