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6O8I image
Btk In Complex With Inhibitor

5VLR image
Crystal Structure Of Pi3K Delta In Complex With A Trifluoro-Ethyl-Pyrazol-Pyrolotriazine Inhibitor

5T18 image
Crystal Structure Of Bruton Agammabulinemia Tyrosine Kinase Complexed With Bms-986142 Aka (2S)-6-Fluoro-5-[3-(8-Fluoro-1-Methyl-2,4-Dioxo-1,2,3,4-Tetrahydroquinazolin-3-Yl)-2-Methylphenyl]-2-(2-Hydroxypropan-2-Yl)-2,3,4,9-Tetrahydro-1H-Carbazole-8-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.50 Å Release Date: 2017-03-08
Classification: TRANSFERASE
Ligands: 73T

5UBR image
Crystal Structure Of Pi3K Alpha In Complex With A 7-(3-(Piperazin-1-Yl)Phenyl)Pyrrolo[2,1-F][1,2,4] Triazin-4-Amine Deriviatine

5UBT image
Crystal Structure Of Pi3K Delta In Complex With A 7-(3-(Piperazin-1-Yl)Phenyl)Pyrrolo[2,1-F][1,2,4] Triazin-4-Amine Deriviatine

5JRS image
Crystal Structure Of Bruton Agammaglobulinemia Tyrosine Kinase Complexed With 4-[2-Fluoro-3-(4-Oxo -3,4-Dihydroquinazolin-3-Yl)Phenyl]-7-(2-Hydroxypropan-2-Y L)-9H-Carbazole-1-Carboxamide

3M6F image
Cd11A I-Domain Complexed With 6-((5S,9R)-9-(4-Cyanophenyl)-3-(3,5-Dichlorophenyl)-1-Methyl-2,4-Dioxo-1,3,7- Triazaspiro[4.4]Non-7-Yl)Nicotinic Acid

2ICA image
Cd11A (Lfa1) I-Domain Complexed With Bms-587101 Aka 5-[(5S, 9R)-9-(4-Cyanophenyl)-3-(3,5-Dichlorophenyl)-1-Methyl-2,4-Dioxo-1,3,7-Triazaspiro [4.4]Non-7-Yl]Methyl]-3-Thiophenecarboxylicacid
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