Search Count: 7
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Crystal Structure Of Wild-Type Egfr In Complex With The Reversible Inhibitor Sevabertinib (Bay 2927088)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.14 Å Release Date: 2025-10-15 Classification: TRANSFERASE Ligands: SIN, CL, DMS, EDO, A1JBI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-10-15
Ligands: SIN, CL, DMS, EDO, A1JBI
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Kat6A In Complex With Small Molecule Inhibitor Bay-184
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.69 Å Release Date: 2024-11-06 Classification: TRANSFERASE Ligands: ZN, A1IDR, EPE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-11-06
Ligands: ZN, A1IDR, EPE
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Crystal Structure Of Human Mbp-Myeloid Cell Leukemia 1 (Mcl-1) In Complex With Brd810 Inhibitor
Organism: Escherichia coli k-12, Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.56 Å Release Date: 2024-06-19 Classification: APOPTOSIS Ligands: MG, YI7, DMS, PGE |
Organism: Escherichia coli k-12, Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-06-19
Ligands: MG, YI7, DMS, PGE
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X-Ray Structure Of Human K-Ras G12C In Complex With Covalent Isoquinolinone Inhibitor (Compound 3)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.64 Å Release Date: 2020-04-08 Classification: HYDROLASE Ligands: GDP, MG, MZQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-08
Ligands: GDP, MG, MZQ
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X-Ray Structure Of Human K-Ras G12C In Complex With Covalent Isoquinolinone Inhibitor (Compound 17)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.16 Å Release Date: 2020-04-08 Classification: HYDROLASE Ligands: GDP, MG, MZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-08
Ligands: GDP, MG, MZN
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Crystal Structure Of Compound 1 With Erk5
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.47 Å Release Date: 2019-02-27 Classification: TRANSFERASE Ligands: G92 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-02-27
Ligands: G92
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Crystal Structure Of Compound 35 With Erk5
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.33 Å Release Date: 2019-02-27 Classification: TRANSFERASE Ligands: G9E |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-02-27
Ligands: G9E
