Search Count: 9
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Egfr (T790M/V948R) In Complex With Quinazolinone Allosteric Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2022-02-23 Classification: TRANSFERASE/Inhibitor Ligands: ANP, MG, YFA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-02-23
Ligands: ANP, MG, YFA
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Egfr Kinase (T790M/V948R) In Complex With Allosteric Inhibitor Jbj-09-063
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.83 Å Release Date: 2021-09-08 Classification: TRANSFERASE/TRANSFERASE Inhibitor Ligands: MG, ANP, VNS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-09-08
Ligands: MG, ANP, VNS
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Egfr(T790M/V948R) In Complex With Ln3844
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.76 Å Release Date: 2021-05-19 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: UEJ, ANP, MG, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-05-19
Ligands: UEJ, ANP, MG, CL
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Crystal Structure Of Egfr(T790M/V948R) In Complex With Ln3753
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2021-03-31 Classification: TRANSFERASE Ligands: TOV, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-03-31
Ligands: TOV, CL
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A Crystal Structure Of Egfr(T790M/V948R) In Complex With Ln3754
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2021-03-31 Classification: TRANSFERASE Ligands: ANP, MG, TQA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-03-31
Ligands: ANP, MG, TQA
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Crystal Structure Of Egfr With Mutant-Selective Dihydrodibenzodiazepinone Allosteric Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2019-12-18 Classification: Transferase/Transferase Inhibitor Ligands: NQ1, ANP, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-12-18
Ligands: NQ1, ANP, MG
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Crystal Structure Of Egfr In Complex With Eai045
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2019-12-18 Classification: TRANSFERASE/TRANSFERASE Inhibitor Ligands: MG, ANP, 9LL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-12-18
Ligands: MG, ANP, 9LL
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Egfr In Complex With A Dihydrodibenzodiazepinone Allosteric Inhibitor.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2019-12-18 Classification: TRANSFERASE/TRANSFERASE Inhibitor Ligands: ANP, O57, MG, AMP, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-12-18
Ligands: ANP, O57, MG, AMP, EDO
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Egfr With An Allosteric Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2019-06-05 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: MG, ANP, JBJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-06-05
Ligands: MG, ANP, JBJ
