Search Count: 41
![]() |
Crystal Structure Of Pde3B In Complex With Gsk4394835A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2024-02-07 Classification: HYDROLASE Ligands: MG, X5W |
![]() |
Hpgds Complexed With An Aza-Quinoline
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2020-11-04 Classification: HYDROLASE Ligands: GSH, SWS |
![]() |
H-Pgds Complexed With Inhibitor 1Y
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.97 Å Release Date: 2020-11-04 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: GSH, EDO, TJG |
![]() |
Hpgds Complexed With A Quinoline-3-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.65 Å Release Date: 2019-03-27 Classification: HYDROLASE Ligands: GSH, KCD |
![]() |
Rat Hpgds Complexed With A Quinoline
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2019-03-27 Classification: HYDROLASE Ligands: GSH, KDV |
![]() |
Tankyrase 2 Complexed With A Selective Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.23 Å Release Date: 2016-09-07 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ZN, PO4, 59B |
![]() |
Human Cd38 Complexed With Inhibitor 1 [6-Fluoro-2-Methyl-4-[(2,3,6-Trichlorobenzyl)Amino]Quinoline-8-Carboxamide]
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2015-08-26 Classification: Hydrolase, Transferase Ligands: 733, HSX |
![]() |
Human Cd38 Complexed With Inhibitor 2 [4-[(2,6-Dimethylbenzyl)Amino]-2-Methylquinoline-8-Carboxamide]
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2015-08-26 Classification: Hydrolase, Transferase Ligands: 41Z, NA7 |
![]() |
Structure Of A Human Cd38 Mutant Complexed With Nmn
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2014-10-08 Classification: HYDROLASE Ligands: NMN |
![]() |
Soluble Epoxide Hydrolase Complexed With A Carboxamide Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.96 Å Release Date: 2013-06-05 Classification: Hydrolase/hydrolase inhibitor Ligands: 1LF |
![]() |
Structure Of Dpp2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2012-09-19 Classification: HYDROLASE Ligands: NAG, ZN |
![]() |
Crystal Structure Of Gsk6414 Bound To Perk (R587-R1092, Delete A660-T867) At 2.28 A Resolution
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.28 Å Release Date: 2012-08-08 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: GOL, 0WH |
![]() |
Crystal Structure Of Gsk6924 Bound To Perk (R587-R1092, Delete A660-T867) At 2.70 A Resolution
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2012-08-08 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 924 |
![]() |
Insulin Receptor Kinase Complexed With An Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2008-12-30 Classification: TRANSFERASE Ligands: GS3 |
![]() |
Jnk1 Complexed With A Bis-Anilino-Pyrrolopyrimidine Inhibitor.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2008-12-30 Classification: TRANSFERASE Ligands: GS7 |
![]() |
Cdk2/Cyclina Complexed With A Imidazo Triazin-2-Amine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.20 Å Release Date: 2008-11-04 Classification: TRANSFERASE/CELL CYCLE Ligands: T2A |
![]() |
Cdk2/Cyclina Complexed With A Pyrazolopyridazine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.15 Å Release Date: 2008-10-21 Classification: Transferase/Cell Cycle Ligands: PO5 |
![]() |
Cdk2/Cyclina Complexed With A Pyrazolopyridazine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.22 Å Release Date: 2008-10-21 Classification: Transferase/Cell cycle Ligands: 5BP |
![]() |
Ligand Binding Domain Of The Glucocorticoid Receptor Complexed With Fluticazone Furoate
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.84 Å Release Date: 2008-06-24 Classification: TRANSCRIPTION Ligands: GW6 |
![]() |
Erbb4 Kinase Domain Complexed With A Thienopyrimidine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2008-03-18 Classification: TRANSFERASE Ligands: GW7 |




















