Search Count: 68
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Crystal Structure Of Pde3B In Complex With Gsk4394835A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2024-02-07 Classification: HYDROLASE Ligands: MG, X5W |
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Human P300 Complexed With A Proline-Based Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.15 Å Release Date: 2022-11-09 Classification: TRANSFERASE/INHIBITOR Ligands: ZN, EDO, C0C |
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Human P300 Complexed With A Glycine-Based Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.36 Å Release Date: 2022-11-09 Classification: TRANSFERASE/INHIBITOR Ligands: ZN, EDO, C3I, ACT |
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Human P300 Complexed With An Azaindazole Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2022-11-09 Classification: TRANSFERASE/INHIBITOR Ligands: ETL |
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Tnni3K Complexed With N-Methyl-4-(4-(3-(3-(Trifluoromethyl) Phenyl) Ureido) Phenoxy)Picolinamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.95 Å Release Date: 2021-11-10 Classification: TRANSFERASE/INHIBITOR Ligands: ZFS |
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Tnni3K Complexed With 1-(3,5-Dichloro-4-((6-(Methylamino)Pyrimidin-4-Yl)Oxy)Phenyl)-3-(3-(Trifluoromethyl)Phenyl)Urea
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.10 Å Release Date: 2021-11-10 Classification: TRANSFERASE/INHIBITOR Ligands: ZGD |
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Hpgds Complexed With An Aza-Quinoline
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2020-11-04 Classification: HYDROLASE Ligands: GSH, SWS |
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H-Pgds Complexed With Inhibitor 1Y
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.97 Å Release Date: 2020-11-04 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: GSH, EDO, TJG |
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Rip2 Kinase Catalytic Domain Complex With 5Amino1Tertbutyl3(3Methoxyphenyl)1H Pyrazole4Carboxamide.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.53 Å Release Date: 2019-12-04 Classification: TRANSFERASE Ligands: M5W, CA |
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Rip2 Kinase Catalytic Domain Complex With (5S,6S,8R)-2-(Benzo[D]Thiazol-5-Yl)-6-Hydroxy-4,5,6,7,8,9-Hexahydro-5,8-Methanopyrazolo[1,5-A][1,3]Diazocine-3-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.68 Å Release Date: 2019-12-04 Classification: TRANSFERASE Ligands: Q9J, CA |
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Rip2 Kinase Catalytic Domain Complex With 5-Amino-1-Phenylpyrazole-4-Carboxamide.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.94 Å Release Date: 2019-10-23 Classification: TRANSFERASE Ligands: M2B, CA |
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Hpgds Complexed With A Quinoline-3-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.65 Å Release Date: 2019-03-27 Classification: HYDROLASE Ligands: GSH, KCD |
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Rat Hpgds Complexed With A Quinoline
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2019-03-27 Classification: HYDROLASE Ligands: GSH, KDV |
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Tnni3K Complexed With A 4,6-Diaminopyrimidine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.97 Å Release Date: 2018-04-04 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: CV4 |
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Tankyrase 2 Complexed With A Selective Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.23 Å Release Date: 2016-09-07 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ZN, PO4, 59B |
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Braf Complexed With An Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.05 Å Release Date: 2016-03-16 Classification: Transferase/Transferase Inhibitor Ligands: GOL, 4EF |
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Tnni3K Complexed With Inhibitor 2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.07 Å Release Date: 2015-09-23 Classification: Transferase/Transferase Inhibitor Ligands: 4CV |
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Tnni3K Complexed With Inhibitor 1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2015-09-23 Classification: Transferase/Transferase Inhibitor Ligands: 4CW |
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Human Cd38 Complexed With Inhibitor 1 [6-Fluoro-2-Methyl-4-[(2,3,6-Trichlorobenzyl)Amino]Quinoline-8-Carboxamide]
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2015-08-26 Classification: Hydrolase, Transferase Ligands: 733, HSX |
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Human Cd38 Complexed With Inhibitor 2 [4-[(2,6-Dimethylbenzyl)Amino]-2-Methylquinoline-8-Carboxamide]
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2015-08-26 Classification: Hydrolase, Transferase Ligands: 41Z, NA7 |




















