Search Count: 11
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Crystal Structure Of Egfr(L858R/T790M/C797S) In Complex With Aur-3418
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.32 Å Release Date: 2025-03-05 Classification: TRANSFERASE/INHIBITOR Ligands: A1A5V, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-03-05
Ligands: A1A5V, CL
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Crystal Structure Of Egfr(L858R/T790M/C797S) In Complex With Aur-8250
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.53 Å Release Date: 2025-03-05 Classification: TRANSFERASE/INHIBITOR Ligands: A1A5L, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-03-05
Ligands: A1A5L, CL
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Discovery Of Potent And Selective Covalent Protein Arginine Methyltransferase (Prmt5) Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2019-06-19 Classification: TRANSFERASE Ligands: CUX, DMS, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-06-19
Ligands: CUX, DMS, EDO
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P38 Inhibitor-Bound
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.09 Å Release Date: 2011-11-02 Classification: TRANSFERASE/transferase inhibitor Ligands: BOG, P5K |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2011-11-02
Ligands: BOG, P5K
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P38 Inhibitor-Bound
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2011-10-12 Classification: transferase/transferase inhibitor Ligands: BOG, P78 |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2011-10-12
Ligands: BOG, P78
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P38 Inhibitor-Bound
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2011-10-12 Classification: transferase/transferase inhibitor Ligands: BOG, P79 |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2011-10-12
Ligands: BOG, P79
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P38 Inhibitor-Bound
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.31 Å Release Date: 2011-10-12 Classification: transferase/transferase inhibitor Ligands: BOG, P7A |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2011-10-12
Ligands: BOG, P7A
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P38 Inhibitor-Bound
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2011-10-12 Classification: transferase/transferase inhibitor Ligands: P7B, BOG |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2011-10-12
Ligands: P7B, BOG
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P38 Inhibitor-Bound
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2011-10-12 Classification: transferase/transferase inhibitor Ligands: BOG, P7C |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2011-10-12
Ligands: BOG, P7C
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Human P38 Map Kinase In Complex With Inhibitor 1A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2005-11-08 Classification: TRANSFERASE Ligands: BOG, BI5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2005-11-08
Ligands: BOG, BI5
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Two Classes Of P38Alpha Map Kinase Inhibitors Having A Common Diphenylether Core But Exhibiting Divergent Binding Modes
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2005-10-18 Classification: TRANSFERASE Ligands: BOG, B11 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2005-10-18
Ligands: BOG, B11
