Search Count: 6
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Crystal Structure Of Flt3 With A Small Molecule Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.10 Å Release Date: 2015-04-22 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: P30 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-04-22
Ligands: P30
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Crystal Structure Of The First Bromodomain Of Human Brd4 In Complex With The Inhibitor Bi-2536
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.73 Å Release Date: 2014-02-26 Classification: TRANSCRIPTION/INHIBITOR Ligands: EDO, R78 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-02-26
Ligands: EDO, R78
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Crystal Structure Of The First Bromodomain Of Human Brd4 In Complex With The Inhibitor Tg-101348
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.65 Å Release Date: 2014-02-26 Classification: TRANSCRIPTION/INHIBITOR Ligands: EDO, 2TA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-02-26
Ligands: EDO, 2TA
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Equally Potent Inhibition Of C-Src And Abl By Compounds That Recognize Inactive Kinase Conformations
Organism: Gallus gallus
Method: X-RAY DIFFRACTION Resolution:2.31 Å Release Date: 2009-03-24 Classification: TRANSFERASE Ligands: G6G, GOL |
Organism: Gallus gallus
Method: X-RAY DIFFRACTION
Release Date: 2009-03-24
Ligands: G6G, GOL
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Src Thr338Ile Inhibited In The Dfg-Asp-Out Conformation
Organism: Gallus gallus
Method: X-RAY DIFFRACTION Resolution:2.35 Å Release Date: 2009-03-24 Classification: TRANSFERASE Ligands: G6H |
Organism: Gallus gallus
Method: X-RAY DIFFRACTION
Release Date: 2009-03-24
Ligands: G6H
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Structure Of The Kinase Domain Of An Imatinib-Resistant Abl Mutant In Complex With The Aurora Kinase Inhibitor Vx-680
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.91 Å Release Date: 2006-01-24 Classification: TRANSFERASE Ligands: VX6 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2006-01-24
Ligands: VX6
