Search Count: 22
![]() |
Kras-G12V-D92C Covalently Bound To Bi-1830
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2025-12-24 Classification: HYDROLASE Ligands: GDP, EDO, A1IWE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-12-24
Ligands: GDP, EDO, A1IWE
![]() |
Cryo-Em Structure Of Prmt5/Wdr77 In Complex With 6S Complex (Picln Pbm Local Refinement)
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY Release Date: 2025-02-19 Classification: TRANSFERASE |
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY
Release Date: 2025-02-19
![]() |
Cryo-Em Structure Of Prmt5/Wdr77 In Complex With 6S Complex
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY Release Date: 2025-02-19 Classification: TRANSFERASE Ligands: SFG |
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY
Release Date: 2025-02-19
Ligands: SFG
![]() |
Cryo-Em Structure Of Prmt5/Wdr77 In Complex With 6S Complex (Grg Local Refine)
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY Release Date: 2025-02-19 Classification: TRANSFERASE Ligands: SFG |
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY
Release Date: 2025-02-19
Ligands: SFG
![]() |
Cryoem Structure Of Prmt5 Bound To Covalent Pbm-Site Inhibitor Brd-6988
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY Release Date: 2021-03-17 Classification: TRANSFERASE/INHIBITOR Ligands: YJG |
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY
Release Date: 2021-03-17
Ligands: YJG
![]() |
Prmt5 Complex Bound To Covalent Pbm Inhibitor Brd6711
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.88 Å Release Date: 2020-11-25 Classification: SPLICING/TRANSFERASE Ligands: QN4, CL, SFG, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-11-25
Ligands: QN4, CL, SFG, GOL
![]() |
Non-Receptor Protein Tyrosine Phosphatase Shp2 In Complex With Allosteric Inhibitor Tno155
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.17 Å Release Date: 2020-09-23 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: VKS, PO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-09-23
Ligands: VKS, PO4
![]() |
Non-Receptor Protein Tyrosine Phosphatase Shp2 In Complex With Allosteric Inhibitor Compound 24
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.92 Å Release Date: 2020-09-23 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: VKP, PO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-09-23
Ligands: VKP, PO4
![]() |
Prmt5 Bound To Pbm Peptide From Riok1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.11 Å Release Date: 2020-08-26 Classification: TRANSFERASE/SPLICING Ligands: SFG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-08-26
Ligands: SFG
![]() |
Prmt5 Bound To The Pbm Peptide From Picln
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.86 Å Release Date: 2020-08-26 Classification: Transferase/Splicing Ligands: SFG, ACE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-08-26
Ligands: SFG, ACE
![]() |
Braf In Complex With N-(4-Methyl-3-(1-Methyl-2-Oxo-2,3-Dihydro-1H-Benzo[D]Imidazol-5-Yl)Phenyl)-3-(Trifluoromethyl)Benzamide.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.04 Å Release Date: 2019-10-23 Classification: transferase/transferase inhibitor Ligands: K7S |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-10-23
Ligands: K7S
![]() |
Braf In Complex With N-(3-(2-(2-Hydroxyethoxy)-6-Morpholinopyridin-4-Yl)-4-Methylphenyl)-2-(Trifluoromethyl)Isonicotinamide (Lxh254)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.37 Å Release Date: 2019-09-04 Classification: transferase/transferase inhibitor Ligands: K81 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-09-04
Ligands: K81
![]() |
Hdm2 (17-111, Wild Type) Complexed With Nvp-Hdm201 At 1.56A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.56 Å Release Date: 2018-08-22 Classification: LIGASE Ligands: 9QW, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-08-22
Ligands: 9QW, CL
![]() |
Crystal Structure Of A Fab Binding To Extracellular Domain 5 Of Cadherin-6
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.34 Å Release Date: 2017-06-07 Classification: IMMUNE SYSTEM Ligands: A2G |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-06-07
Ligands: A2G
![]() |
Abl1 Kinase (T334I_D382N) In Complex With Asciminib And Nilotinib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.17 Å Release Date: 2017-04-05 Classification: TRANSFERASE Ligands: NIL, AY7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-04-05
Ligands: NIL, AY7
![]() |
Non-Receptor Protein Tyrosine Phosphatase Shp2 In Complex With Allosteric Inhibitor Shp836
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2016-07-06 Classification: Hydrolase/Hydrolase Inhibitor Ligands: 5OA, PO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-07-06
Ligands: 5OA, PO4
![]() |
Non-Receptor Protein Tyrosine Phosphatase Shp2 In Complex With Allosteric Inhibitor Shp099
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2016-06-29 Classification: Hydrolase/Hydrolase Inhibitor Ligands: 5OD, PO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-06-29
Ligands: 5OD, PO4
![]() |
Crystal Structure Of Prmt5:Mep50 In Complex With Mta And H4 Peptide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.34 Å Release Date: 2016-02-24 Classification: TRANSFERASE/PROTEIN BINDING Ligands: MTA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-02-24
Ligands: MTA
![]() |
Her3 Extracellular Domain In Complex With Fab Fragment Of Mor09825
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.40 Å Release Date: 2014-04-16 Classification: Signaling protein, immune system Ligands: NAG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-04-16
Ligands: NAG
![]() |
Structural Basis Of Jak2 Inhibition By The Type Ii Inhibtor Nvp-Bbt594
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.34 Å Release Date: 2012-05-16 Classification: Transferase/transferase inhibitor Ligands: 046, MLI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-05-16
Ligands: 046, MLI
