Search Count: 26
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Crystal Structure Of Selective Ire1A Inhibitor 29 At The Enzyme Active Site
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.43 Å Release Date: 2024-05-29 Classification: TRANSFERASE/INHIBITOR Ligands: EDO, XOE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-05-29
Ligands: EDO, XOE
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Crystal Structure Of Ire1A In Complex With G-6904
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.45 Å Release Date: 2021-04-21 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: N8S, EPE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-04-21
Ligands: N8S, EPE
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Crystal Structure Of Ire1 In Complex With G-3053
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2021-04-21 Classification: TRANSFERASE/INHIBITOR Ligands: N97 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-04-21
Ligands: N97
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Crystal Structure Of Ire1A In Complex With G-4100
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.54 Å Release Date: 2021-04-21 Classification: TRANSFERASE/TRANSFERASE INHIBITOR |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-04-21
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Usp7 In Complex With Ligand Compound 18
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.93 Å Release Date: 2020-04-29 Classification: HYDROLASE Ligands: R44, ACT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-29
Ligands: R44, ACT
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Usp7 In Complex With Ligand Compound 23
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.73 Å Release Date: 2020-04-29 Classification: HYDROLASE Ligands: R3Y |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-29
Ligands: R3Y
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Usp7 In Complex With Ligand Compound 1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.69 Å Release Date: 2020-04-29 Classification: HYDROLASE Ligands: R4D |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-29
Ligands: R4D
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Usp7 In Complex With Ligand Compound 7
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2020-04-29 Classification: HYDROLASE Ligands: R41 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-29
Ligands: R41
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Usp7 In Complex With Ligand Compound 14
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.99 Å Release Date: 2020-04-29 Classification: HYDROLASE Ligands: R4J, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-29
Ligands: R4J, ZN
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E. Coli Lepb In Complex With Gne0775 ((4S,7S,10S)-10-((S)-4-Amino-2-(2-(4-(Tert-Butyl)Phenyl)-4-Methylpyrimidine-5-Carboxamido)-N-Methylbutanamido)-16,26-Bis(2-Aminoethoxy)-N-(2-Iminoethyl)-7-Methyl-6,9-Dioxo-5,8-Diaza-1,2(1,3)-Dibenzenacyclodecaphane-4-Carboxamide)
Organism: Escherichia coli (strain k12)
Method: X-RAY DIFFRACTION Resolution:2.41 Å Release Date: 2018-10-10 Classification: HYDROLASE/HYDROLASE inhibitor Ligands: CZD, 1PE |
Organism: Escherichia coli (strain k12)
Method: X-RAY DIFFRACTION
Release Date: 2018-10-10
Ligands: CZD, 1PE
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Structure Of The Human Glun1/Glun2A Lbd In Complex With Compound 2 (Gne9178)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2016-11-30 Classification: TRANSPORT PROTEIN Ligands: ACT, GLU, 7H0, CA, GLY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-11-30
Ligands: ACT, GLU, 7H0, CA, GLY
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Structure Of The Human Glun1/Glun2A Lbd In Complex With Compound 9 (Gne3500)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.48 Å Release Date: 2016-11-30 Classification: TRANSPORT PROTEIN Ligands: GLU, 7H2, GLY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-11-30
Ligands: GLU, 7H2, GLY
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Structure Of The Human Glun1/Glun2A Lbd In Complex With Gne6901
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.09 Å Release Date: 2016-07-13 Classification: TRANSPORT PROTEIN Ligands: ACT, GLU, GLY, 6RM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-07-13
Ligands: ACT, GLU, GLY, 6RM
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Structure Of The Human Glun1/Glun2A Lbd In Complex With Gne0723
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.44 Å Release Date: 2016-07-13 Classification: TRANSPORT PROTEIN Ligands: ACT, GLU, 6RV, GLY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-07-13
Ligands: ACT, GLU, 6RV, GLY
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Crystal Structure Of Erk2 In Complex With Compound 22
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.76 Å Release Date: 2016-07-06 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 6QB, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-07-06
Ligands: 6QB, EDO
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Crystal Structure Of Cdk2 In Complex With Compound 22
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2016-07-06 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 6QB |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-07-06
Ligands: 6QB
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Structure Of The Human Glun1/Glun2A Lbd In Complex With 7-{[Ethyl(4-Fluorophenyl)Amino]Methyl}-N,2-Dimethyl-5-Oxo-5H-[1,3]Thiazolo[3,2-A]Pyrimidine-3-Carboxamide (Compound 19)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.86 Å Release Date: 2016-03-16 Classification: TRANSPORT PROTEIN Ligands: GLU, GLY, 67H |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-03-16
Ligands: GLU, GLY, 67H
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Structure Of The Human Glun1/Glun2A Lbd In Complex With N-Ethyl-7-{[2-Fluoro-3-(Trifluoromethyl)Phenyl]Methyl}-2-Methyl-5-Oxo-5H-[1,3]Thiazolo[3,2-A]Pyrimidine-3-Carboxamide (Compound 29)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.12 Å Release Date: 2016-03-16 Classification: TRANSPORT PROTEIN Ligands: CA, GLU, 67J, EPE, GLY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-03-16
Ligands: CA, GLU, 67J, EPE, GLY
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Structure Of The Apo Human Glun1/Glun2A Lbd
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.81 Å Release Date: 2016-02-24 Classification: TRANSPORT PROTEIN Ligands: GOL, GLU, GLY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-02-24
Ligands: GOL, GLU, GLY
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Structure Of The Human Glun1/Glun2A Lbd In Complex With Gne3419
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.23 Å Release Date: 2016-02-24 Classification: TRANSPORT PROTEIN Ligands: ACT, GLU, CA, GLY, 5YC |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-02-24
Ligands: ACT, GLU, CA, GLY, 5YC