Search Count: 13
![]() |
Crystal Structure Of Rhodesain In Complex With A Macrolactam Inhibitor
Organism: Trypanosoma brucei rhodesiense
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2018-04-11 Classification: HYDROLASE Ligands: C2K, EDO |
Organism: Trypanosoma brucei rhodesiense
Method: X-RAY DIFFRACTION
Release Date: 2018-04-11
Ligands: C2K, EDO
![]() |
Crystal Structure Of Rhodesain In Complex With A Macrolactam Inhibitor
Organism: Trypanosoma brucei rhodesiense
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2018-04-11 Classification: HYDROLASE Ligands: EDO, C3E |
Organism: Trypanosoma brucei rhodesiense
Method: X-RAY DIFFRACTION
Release Date: 2018-04-11
Ligands: EDO, C3E
![]() |
Crystal Structure Of Rhodesain In Complex With A Macrolactam Inhibitor
Organism: Trypanosoma brucei rhodesiense
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2018-04-11 Classification: HYDROLASE Ligands: EDO, C2W |
Organism: Trypanosoma brucei rhodesiense
Method: X-RAY DIFFRACTION
Release Date: 2018-04-11
Ligands: EDO, C2W
![]() |
Cathepsin L In Complex With (3S,14E)-19-Chloro-N-(1-Cyanocyclopropyl)-5-Oxo-12,17-Dioxa-4-Azatricyclo[16.2.2.06,11]Docosa-1(21),6(11),7,9,14,18(22),19-Heptaene-3-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.37 Å Release Date: 2018-04-11 Classification: HYDROLASE Ligands: C3E, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-04-11
Ligands: C3E, GOL
![]() |
Cathepsin L In Complex With (3S,14E)-19-Chloro-N-(1-Cyanocyclopropyl)-5-Oxo-17-Oxa-4-Azatricyclo[16.2.2.06,11]Docosa-1(21),6,8,10,14,18(22),19-Heptaene-3-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.34 Å Release Date: 2018-04-11 Classification: HYDROLASE Ligands: C7Q |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-04-11
Ligands: C7Q
![]() |
Cathepsin L In Complex With (3S,14E)-8-(Azetidin-3-Yl)-19-Chloro-N-(1-Cyanocyclopropyl)-5-Oxo-12,17-Dioxa-4-Azatricyclo[16.2.2.06,11]Docosa-1(21),6,8,10,14,18(22),19-Heptaene-3-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.02 Å Release Date: 2018-04-11 Classification: HYDROLASE Ligands: C7T, ZN, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-04-11
Ligands: C7T, ZN, CL
![]() |
Crystal Structure Of Human Fxr In Complex With 4-({(2S)-2-[2-(4-Chlorophenyl)-5,6-Difluoro-1H-Benzimidazol-1-Yl]-2-Cyclohexylacetyl}Amino)-3-Methylbenzoic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2011-01-19 Classification: HORMONE RECEPTOR Ligands: OLF |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-01-19
Ligands: OLF
![]() |
Crystal Structure Of Human Fxr In Complex With (2S)-2-[2-(4-Chlorophenyl)-5,6-Difluoro-1H-Benzimidazol-1-Yl]-2-Cyclohexyl-N-(2-Methylphenyl)Ethanamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2011-01-19 Classification: HORMONE RECEPTOR Ligands: OMK |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-01-19
Ligands: OMK
![]() |
Crystal Structure Of Human Fxr In Complex With 4-({(2S)-2-[2-(4-Chlorophenyl)-5,6-Difluoro-1H-Benzimidazol-1-Yl]-2-Cyclohexylacetyl}Amino)-3-Fluorobenzoic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2011-01-19 Classification: HORMONE RECEPTOR Ligands: OMM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-01-19
Ligands: OMM
![]() |
Crystal Structure Of Human Fxr In Complex With 4-({(2S)-2-[2-(4-Chlorophenyl)-5,6-Difluoro-1H-Benzimidazol-1-Yl]-2-Cyclohexylacetyl}Amino)Benzoic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.29 Å Release Date: 2011-01-19 Classification: HORMONE RECEPTOR Ligands: OOF |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-01-19
Ligands: OOF
![]() |
Crystal Structure Of Human Fxr In Complex With 4-({(2S)-2-[2-(4-Chlorophenyl)-5,6-Difluoro-1H-Benzimidazol-1-Yl]-2-Cyclohexylacetyl}Amino)-3,5-Difluorobenzoic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.29 Å Release Date: 2011-01-19 Classification: HORMONE RECEPTOR Ligands: OOK |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-01-19
Ligands: OOK
![]() |
Crystal Structure Of Human Fxr In Complex With 2-(4-Chlorophenyl)-1-[(1S)-1-Cyclohexyl-2-(Cyclohexylamino)-2-Oxoethyl]-1H-Benzimidazole-6-Carboxylic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2010-12-29 Classification: HORMONE RECEPTOR Ligands: OKH |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-12-29
Ligands: OKH
![]() |
Crystal Structure Of Human Fxr In Complex With (2S)-2-[2-(4-Chlorophenyl)-1H-Benzimidazol-1-Yl]-N,2-Dicyclohexylethanamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2010-12-29 Classification: HORMONE RECEPTOR Ligands: OKI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-12-29
Ligands: OKI
