Search Count: 51
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Crystal Structure Of Brd4(1) In Complex With The Inhibitor Mpm2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.77 Å Release Date: 2023-02-08 Classification: PROTEIN BINDING Ligands: I5K, BU3, DMS, P6G |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-02-08
Ligands: I5K, BU3, DMS, P6G
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Crystal Structure Of Danio Rerio Histone Deacetylase 10 In Complex With Piperidine-4-Hydroxamic Acid Inhibitor
Organism: Danio rerio
Method: X-RAY DIFFRACTION Resolution:2.18 Å Release Date: 2023-01-11 Classification: HYDROLASE Ligands: EDO, LDI, ZN, K, PO4, NA |
Organism: Danio rerio
Method: X-RAY DIFFRACTION
Release Date: 2023-01-11
Ligands: EDO, LDI, ZN, K, PO4, NA
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Crystal Structure Of Brd4(1) In Complex With The Inhibitor Mpm6
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.92 Å Release Date: 2022-06-08 Classification: PROTEIN BINDING Ligands: SOK, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-06-08
Ligands: SOK, DMS
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Crystal Structure Of Trypanosoma Cruzi Histone Deacetylase Dac2 Complexed With Quisinostat
Organism: Trypanosoma cruzi
Method: X-RAY DIFFRACTION Resolution:1.75 Å Release Date: 2021-12-15 Classification: HYDROLASE Ligands: ZN, K, GOK, GOL |
Organism: Trypanosoma cruzi
Method: X-RAY DIFFRACTION
Release Date: 2021-12-15
Ligands: ZN, K, GOK, GOL
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Crystal Structure Of Trypanosoma Cruzi Histone Deacetylase Dac2 Complexed With A Hydroxamate Inhibitor
Organism: Trypanosoma cruzi
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2021-12-15 Classification: HYDROLASE Ligands: ZN, K, T56 |
Organism: Trypanosoma cruzi
Method: X-RAY DIFFRACTION
Release Date: 2021-12-15
Ligands: ZN, K, T56
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Crystal Structure Of Schistosoma Mansoni Hdac8 Complexed With A Benzohydroxamate Inhibitor 12
Organism: Schistosoma mansoni
Method: X-RAY DIFFRACTION Resolution:1.55 Å Release Date: 2021-09-15 Classification: HYDROLASE Ligands: ZN, K, GOL, 5IB |
Organism: Schistosoma mansoni
Method: X-RAY DIFFRACTION
Release Date: 2021-09-15
Ligands: ZN, K, GOL, 5IB
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Crystal Structure Of Brd4(1) Bound To Inhibitor Bux6 (12)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2020-12-16 Classification: TRANSCRIPTION Ligands: BU3, L2Z |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-12-16
Ligands: BU3, L2Z
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Crystal Structure Of Brd4(1) Bound To Inhibitor Bug0 (6)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.40 Å Release Date: 2020-12-09 Classification: TRANSCRIPTION Ligands: KLK |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-12-09
Ligands: KLK
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Crystal Structure Of Brd4(1) Bound To Inhibitor Bux1 (8)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2020-12-09 Classification: TRANSCRIPTION Ligands: BU3, KUH, CA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-12-09
Ligands: BU3, KUH, CA
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Crystal Structure Of Brd4(1) Bound To Inhibitor Bux2 (9)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.40 Å Release Date: 2020-12-09 Classification: TRANSCRIPTION Ligands: KXK, BU3 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-12-09
Ligands: KXK, BU3
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Crystal Structure Of Brd4(1) Bound To Inhibitor Bux3 (10)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2020-12-09 Classification: TRANSCRIPTION Ligands: BU3, L25 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-12-09
Ligands: BU3, L25
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Crystal Structure Of Brd4(1) Bound To Inhibitor Bux4 (13)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2020-12-09 Classification: TRANSCRIPTION Ligands: L2N |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-12-09
Ligands: L2N
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Crystal Structure Of Brd4(1) Bound To Inhibitor Bux5 (11)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2020-12-09 Classification: TRANSCRIPTION Ligands: L2W |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-12-09
Ligands: L2W
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Crystal Structure Of Brd4(1) Bound To Inhibitor Bux14 (7)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2020-12-09 Classification: TRANSCRIPTION Ligands: L45, BU3 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-12-09
Ligands: L45, BU3
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Crystal Structure Of Schistosoma Mansoni Hdac8 Complexed With A N-Alkyl Hydroxamate
Organism: Schistosoma mansoni
Method: X-RAY DIFFRACTION Resolution:1.55 Å Release Date: 2019-03-13 Classification: HYDROLASE Ligands: ZN, K, E7Q, GOL |
Organism: Schistosoma mansoni
Method: X-RAY DIFFRACTION
Release Date: 2019-03-13
Ligands: ZN, K, E7Q, GOL
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Crystal Structure Of Schistosoma Mansoni Hdac8 Complexed With Pci-34051
Organism: Schistosoma mansoni
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2018-10-31 Classification: HYDROLASE Ligands: ZN, K, GKW, GOL |
Organism: Schistosoma mansoni
Method: X-RAY DIFFRACTION
Release Date: 2018-10-31
Ligands: ZN, K, GKW, GOL
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Crystal Structure Of Schistosoma Mansoni Hdac8 Complexed With Ncc-149
Organism: Schistosoma mansoni
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2018-10-31 Classification: HYDROLASE Ligands: ZN, K, GM5, DMF, GOL |
Organism: Schistosoma mansoni
Method: X-RAY DIFFRACTION
Release Date: 2018-10-31
Ligands: ZN, K, GM5, DMF, GOL
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Crystal Structure Of Schistosoma Mansoni Hdac8 Mutant H292M Complexed With Pci-34051
Organism: Schistosoma mansoni
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2018-10-31 Classification: HYDROLASE Ligands: ZN, K, GKW, DMF, GOL |
Organism: Schistosoma mansoni
Method: X-RAY DIFFRACTION
Release Date: 2018-10-31
Ligands: ZN, K, GKW, DMF, GOL
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Crystal Structure Of Schistosoma Mansoni Hdac8 H292M Mutant Complexed With Ncc-149
Organism: Schistosoma mansoni
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2018-10-31 Classification: HYDROLASE Ligands: ZN, K, GM5, DMF, GOL |
Organism: Schistosoma mansoni
Method: X-RAY DIFFRACTION
Release Date: 2018-10-31
Ligands: ZN, K, GM5, DMF, GOL
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Crystal Structure Of Schistosoma Mansoni Hdac8 Complexed With Quisinostat
Organism: Schistosoma mansoni
Method: X-RAY DIFFRACTION Resolution:1.55 Å Release Date: 2018-10-31 Classification: HYDROLASE Ligands: ZN, K, GOK, DMF, GOL |
Organism: Schistosoma mansoni
Method: X-RAY DIFFRACTION
Release Date: 2018-10-31
Ligands: ZN, K, GOK, DMF, GOL
