Search Count: 42
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A Novel Bottom-Up Approach To Find Lead-Compounds In Billion-Sized Libraries
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.33 Å Release Date: 2025-08-13 Classification: GENE REGULATION Ligands: A1IXD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-08-13
Ligands: A1IXD
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A Novel Bottom-Up Approach To Find Lead-Compounds In Billion-Sized Libraries
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.94 Å Release Date: 2025-08-13 Classification: GENE REGULATION Ligands: A1IXE, P6G |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-08-13
Ligands: A1IXE, P6G
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A Novel Bottom-Up Approach To Find Lead-Compounds In Billion-Sized Libraries
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.42 Å Release Date: 2025-08-13 Classification: GENE REGULATION Ligands: A1IXF, P4G |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-08-13
Ligands: A1IXF, P4G
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Crystal Structure Of Tnf Alpha In Complex With Compound 1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.36 Å Release Date: 2025-07-23 Classification: CYTOKINE Ligands: A1CB1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-07-23
Ligands: A1CB1
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Crystal Structure Of Tnf Alpha In Complex With Compound 4
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2025-07-23 Classification: CYTOKINE Ligands: A1CB0 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-07-23
Ligands: A1CB0
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Crystal Structure Of Tnf Alpha In Complex With Compound 3.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.16 Å Release Date: 2025-07-23 Classification: CYTOKINE Ligands: A1CBZ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-07-23
Ligands: A1CBZ
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Crystal Structure Of Tnf Alpha In Complex With Compound 19
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.78 Å Release Date: 2025-07-23 Classification: CYTOKINE Ligands: A1CCE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-07-23
Ligands: A1CCE
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Crystal Structure Of Human Hpk1 (Map4K1) Complex With 7-(1-Methyl-1H-Pyrazol-4-Yl)-N-[4-(1-Methylpiperidin-4-Yl)Phenyl]Quinazolin-2-Amine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.94 Å Release Date: 2023-08-16 Classification: TRANSFERASE Ligands: UES |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-08-16
Ligands: UES
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Crystal Structure Of Human Hpk1 (Map4K1) Complex With 2-[8-Amino-7-Fluoro-6-(8-Methyl-2,3-Dihydro-1H-Pyrido[2,3-B][1,4]Oxazin-7-Yl)-Isoquinolin-3-Ylamino]-6-Isopropyl-5,6-Dihydro-4H-1,6,8A-Triaza-Azulen-7-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.82 Å Release Date: 2023-08-16 Classification: TRANSFERASE Ligands: USF |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-08-16
Ligands: USF
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T. Cruzi Topoisomerase Ii Alpha Bound To Dsdna And The Covalent Inhibitor Ct1
Organism: Trypanosoma cruzi strain cl brener, Escherichia coli
Method: ELECTRON MICROSCOPY Release Date: 2023-07-12 Classification: ISOMERASE Ligands: YWX |
Organism: Trypanosoma cruzi strain cl brener, Escherichia coli
Method: ELECTRON MICROSCOPY
Release Date: 2023-07-12
Ligands: YWX
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Btk In Complex With 18A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.94 Å Release Date: 2021-10-06 Classification: TRANSFERASE/INHIBITOR Ligands: 2IE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-10-06
Ligands: 2IE
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Btk In Complex With 25A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.52 Å Release Date: 2021-10-06 Classification: TRANSFERASE/INHIBITOR Ligands: 2IJ, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-10-06
Ligands: 2IJ, DMS
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Btk1 Soaked With Compound 5, Y551 Is Sequestered
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.84 Å Release Date: 2021-05-19 Classification: TRANSFERASE Ligands: X9J, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-05-19
Ligands: X9J, DMS
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Btk1 Soaked With Compound 5, Y551 Is Sequestered
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.33 Å Release Date: 2021-05-19 Classification: TRANSFERASE Ligands: X9M |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-05-19
Ligands: X9M
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Btk1 Soaked With Compound 26
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.34 Å Release Date: 2021-05-19 Classification: TRANSFERASE Ligands: X9P, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-05-19
Ligands: X9P, DMS
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Btk1 Soaked With Compound 24
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.94 Å Release Date: 2021-05-19 Classification: TRANSFERASE Ligands: X9S, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-05-19
Ligands: X9S, DMS
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Btk1 Soaked With Compound 25
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.83 Å Release Date: 2021-05-19 Classification: TRANSFERASE Ligands: X9V, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-05-19
Ligands: X9V, DMS
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Btk1 Soaked With Compound 30
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.38 Å Release Date: 2021-05-19 Classification: TRANSFERASE Ligands: DMS, X9Y |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-05-19
Ligands: DMS, X9Y
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Solution Structure Of The Fus/Tls Rna Recognition Motif In Complex With U1 Snrna Stem Loop Iii
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Organism: Homo sapiens
Method: SOLUTION NMR
Release Date: 2020-10-28
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Structure Of Human Bruton'S Tyrosine Kinase In Complex With Evobrutinib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.41 Å Release Date: 2019-08-14 Classification: Transferase/Transferase Inhibitor Ligands: CL, MZJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-08-14
Ligands: CL, MZJ
