Search Count: 23
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Crystal Structure Of Human Kdm4A In Complex With Compound 18A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.25 Å Release Date: 2019-06-12 Classification: OXIDOREDUCTASE Ligands: ZN, FQH, GOL, CL, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-06-12
Ligands: ZN, FQH, GOL, CL, DMS
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Crystal Structure Of Human Kdm4A In Complex With Compound 16A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.19 Å Release Date: 2019-06-12 Classification: OXIDOREDUCTASE Ligands: ZN, FQ5, DMS, CL, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-06-12
Ligands: ZN, FQ5, DMS, CL, GOL
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Crystal Structure Of Human Kdm4A In Complex With Compound 34A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.31 Å Release Date: 2019-06-12 Classification: OXIDOREDUCTASE Ligands: ZN, FO2, GOL, DMS, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-06-12
Ligands: ZN, FO2, GOL, DMS, CL
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Crystal Structure Of Human Kdm4A In Complex With Compound 17F
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.14 Å Release Date: 2019-06-12 Classification: OXIDOREDUCTASE Ligands: ZN, FQB, DMS, GOL, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-06-12
Ligands: ZN, FQB, DMS, GOL, CL
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Crystal Structure Of Human Kdm4A In Complex With Compound 16M
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.45 Å Release Date: 2019-06-12 Classification: OXIDOREDUCTASE Ligands: ZN, FQE, DMS, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-06-12
Ligands: ZN, FQE, DMS, CL
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Crystal Structure Of Human Kdm4A In Complex With Compound 19A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.38 Å Release Date: 2019-06-12 Classification: OXIDOREDUCTASE Ligands: ZN, FOW, CL, GOL, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-06-12
Ligands: ZN, FOW, CL, GOL, DMS
 |
Crystal Structure Of Human Kdm4A In Complex With Compound 34B
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.21 Å Release Date: 2019-06-12 Classification: OXIDOREDUCTASE Ligands: ZN, FO2, DMS, GOL, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-06-12
Ligands: ZN, FO2, DMS, GOL, CL
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Crystal Structure Of Human Kdm4A In Complex With Compound 34G
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.15 Å Release Date: 2019-06-12 Classification: OXIDOREDUCTASE Ligands: ZN, FQN, CL, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-06-12
Ligands: ZN, FQN, CL, DMS
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Crystal Structure Of Human Kdm4A In Complex With Compound 19D
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.81 Å Release Date: 2019-06-12 Classification: OXIDOREDUCTASE Ligands: ZN, FQQ, DMS, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-06-12
Ligands: ZN, FQQ, DMS, CL
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Crystal Structure Of Human Kdm4A In Complex With Compound 17B
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.34 Å Release Date: 2019-06-12 Classification: OXIDOREDUCTASE Ligands: ZN, FNQ, DMS, GOL, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-06-12
Ligands: ZN, FNQ, DMS, GOL, CL
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Crystal Structure Of Human Kdm4A In Complex With Compound 17E
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.38 Å Release Date: 2019-06-12 Classification: OXIDOREDUCTASE Ligands: ZN, FO8, CL, DMS, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-06-12
Ligands: ZN, FO8, CL, DMS, GOL
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Crystal Structure Of Human Kdm5B In Complex With Compound 16A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2019-06-12 Classification: OXIDOREDUCTASE Ligands: ZN, MN, FQ5, DMS, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-06-12
Ligands: ZN, MN, FQ5, DMS, EDO
 |
Crystal Structure Of Human Kdm5B In Complex With Compound 34A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.19 Å Release Date: 2019-06-12 Classification: OXIDOREDUCTASE Ligands: ZN, MN, EDO, PO4, FO2, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-06-12
Ligands: ZN, MN, EDO, PO4, FO2, DMS
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Crystal Structure Of Human Kdm5B In Complex With Compound 34F
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.21 Å Release Date: 2019-06-12 Classification: OXIDOREDUCTASE Ligands: ZN, MN, DMS, EDO, PO4, FQK |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-06-12
Ligands: ZN, MN, DMS, EDO, PO4, FQK
 |
Crystal Structure Of Human Kdm5B In Complex With Compound 34G
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.14 Å Release Date: 2019-06-12 Classification: OXIDOREDUCTASE Ligands: ZN, MN, DMS, PO4, FQN, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-06-12
Ligands: ZN, MN, DMS, PO4, FQN, EDO
 |
Ire1 Kinase/Rnase In Complex With Imidazo[1,2-B]Pyridazin-8-Amine Compound 33
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.73 Å Release Date: 2019-02-27 Classification: SIGNALING PROTEIN Ligands: GUK |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-02-27
Ligands: GUK
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Ire1 Alpha In Complex With Imidazo[1,2-B]Pyridazin-8-Amine Compound 2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.14 Å Release Date: 2019-02-27 Classification: TRANSFERASE Ligands: GXK |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-02-27
Ligands: GXK
 |
Introduction Of A Methyl Group Curbs Metabolism Of Pyrido[3,4-D]Pyrimidine Mps1 Inhibitors And Enables The Discovery Of The Phase 1 Clinical Candidate Bos172722.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.48 Å Release Date: 2018-09-19 Classification: TRANSFERASE Ligands: FMW, 7PE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-09-19
Ligands: FMW, 7PE
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Rapid Discovery Of Pyrido[3,4-D]Pyrimidine Inhibitors Of Monopolar Spindle Kinase 1 (Mps1) Using A Structure-Based Hydridization Approach
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.18 Å Release Date: 2016-04-20 Classification: TRANSFERASE Ligands: 5NW, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-04-20
Ligands: 5NW, DMS
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Rapid Discovery Of Pyrido[3,4-D]Pyrimidine Inhibitors Of Monopolar Spindle Kinase 1 (Mps1) Using A Structure-Based Hydridization Approach
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.26 Å Release Date: 2016-04-20 Classification: TRANSFERASE Ligands: 7PE, 5O4, EDO, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-04-20
Ligands: 7PE, 5O4, EDO, DMS