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7X7O image
Sars-Cov-2 Spike Rbd In Complex With Neutralizing Antibody Ut28K

5VP0 image
Discovery Of Clinical Candidate N-{(1S)-1-[3-Fluoro-4-(Trifluoromethoxy)Phenyl]-2-Methoxyethyl}-7-Methoxy-2-Oxo-2,3-Dihydropyrido[2,3-B]Pyrazine-4(1H)-Carboxamide (Tak-915), A Highly Potent, Selective, And Brain-Penetrating Phosphodiesterase 2A Inhibitor For The Treatment Of Cognitive Disorders

5XKM image
Crystal Structure Of Human Phosphodiesterase 2A In Complex With 6-Methyl-N-(1-(4-(Trifluoromethoxy)Phenyl)Propyl)Pyrazolo[1,5-A]Pyrimidine-3-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.16 Å Release Date: 2017-08-16
Classification: HYDROLASE
Ligands: MG, ZN, 87R

5XCO image
Crystal Structure Of Human K-Ras G12D Mutant In Complex With Gdp And Cyclic Inhibitory Peptide

5F1Z image
Structure Of Tyk2 With Inhibitor 16: 3-Azanyl-5-[(2~{S})-3-Methylbutan-2-Yl]-7-[1-Methyl-5-(2-Oxidanylpropan-2-Yl)Pyrazol-3-Yl]-1~{H}-Pyrazolo[4,3-C]Pyridin-4-One

5F20 image
Structure Of Tyk2 With Inhibitor 4: 3-Azanyl-5-(2-Methylphenyl)-7-(1-Methylpyrazol-3-Yl)-1~{H}-Pyrazolo[4,3-C]Pyridin-4-One

3WE4 image
Crystal Structure Of S6K1 Kinase Domain In Complex With A Pyrimidine Derivative Pf-4708671 2-{[4-(5-Ethylpyrimidin-4-Yl)Piperazin-1-Yl]Methyl}-5-(Trifluoromethyl)-1H-Benzimidazole

3WF5 image
Crystal Structure Of S6K1 Kinase Domain In Complex With A Pyrazolopyrimidine Derivative 4-[4-(1H-Benzimidazol-2-Yl)Piperidin-1-Yl]-1H-Pyrazolo[3,4-D]Pyrimidine

3WF6 image
Crystal Structure Of S6K1 Kinase Domain In Complex With A Pyrazolopyrimidine Derivative 4-[4-(1H-Indol-3-Yl)-3,6-Dihydropyridin-1(2H)-Yl]-1H-Pyrazolo[3,4-D]Pyrimidine

3WF7 image
Crystal Structure Of S6K1 Kinase Domain In Complex With A Purine Derivative 1-(9H-Purin-6-Yl)-N-[3-(Trifluoromethyl)Phenyl]Piperidine-4-Carboxamide

3WF8 image
Crystal Structure Of S6K1 Kinase Domain In Complex With A Quinoline Derivative 2-Oxo-2-[(4-Sulfamoylphenyl)Amino]Ethyl 7,8,9,10-Tetrahydro-6H-Cyclohepta[B]Quinoline-11-Carboxylate

3WF9 image
Crystal Structure Of S6K1 Kinase Domain In Complex With A Quinoline Derivative 1-Oxo-1-[(4-Sulfamoylphenyl)Amino]Propan-2-Yl-2-Methyl-1,2,3,4-Tetrahydroacridine-9-Carboxylate

3WD9 image
Crystal Structure Of Phosphodiesterase 4B In Complex With Compound 10F

3W5E image
Crystal Structure Of Phosphodiesterase 4B In Complex With Compound 31E

3A35 image
Crystal Structure Of Lump Complexed With Riboflavin

3A3B image
Crystal Structure Of Lump Complexed With Flavin Mononucleotide

3A3G image
Crystal Structure Of Lump Complexed With 6,7-Dimethyl-8-(1'-D-Ribityl) Lumazine

2D57 image
Double Layered 2D Crystal Structure Of Aquaporin-4 (Aqp4M23) At 3.2 A Resolution By Electron Crystallography
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