Search Count: 8
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Identification Of Novel, Potent And Selective Gcn2 Inhibitors As First-In-Class Anti-Tumor Agents
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.61 Å Release Date: 2019-10-09 Classification: transferase/transferase inhibitor Ligands: KAV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-10-09
Ligands: KAV
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Identification Of Novel, Potent And Selective Gcn2 Inhibitors As First-In-Class Anti-Tumor Agents
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.01 Å Release Date: 2019-10-09 Classification: transferase/transferase inhibitor Ligands: KA4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-10-09
Ligands: KA4
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Identification Of Novel, Potent And Selective Gcn2 Inhibitors As First-In-Class Anti-Tumor Agents
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2019-10-09 Classification: transferase/transferase inhibitor Ligands: KA7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-10-09
Ligands: KA7
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Structure Of Cdk12/Cyck In Complex With A Small Molecule Inhibitor N-(4-(1-Methyl-1H-Pyrazol-4-Yl)Phenyl)-N-((1R,4R)-4-(Quinazolin-2-Ylamino)Cyclohexyl)Acetamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2018-08-29 Classification: TRANSFERASE/INHIBITOR Ligands: MG, 8M1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-08-29
Ligands: MG, 8M1
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Crystal Structure Of Human K-Ras G12D Mutant In Complex With Gdp And Cyclic Inhibitory Peptide
Organism: Homo sapiens, Enterobacteria phage t7
Method: X-RAY DIFFRACTION Resolution:1.25 Å Release Date: 2017-05-24 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: GDP, EDO |
Organism: Homo sapiens, Enterobacteria phage t7
Method: X-RAY DIFFRACTION
Release Date: 2017-05-24
Ligands: GDP, EDO
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Crystal Structure Of Mcl-1 In Complex With Compound 4
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2013-11-27 Classification: APOPTOSIS Ligands: LC3 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-11-27
Ligands: LC3
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Crystal Structure Of Mcl-1 In Complex With Compound 10
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.15 Å Release Date: 2013-11-27 Classification: APOPTOSIS Ligands: LC6 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-11-27
Ligands: LC6
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Crystal Structure Of Bcl-Xl In Complex With Compound 10
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.45 Å Release Date: 2013-11-27 Classification: APOPTOSIS Ligands: LC6, PO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-11-27
Ligands: LC6, PO4
