Search Count: 72
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Co-Crystal Structure Of The Ternary Complex Of Human Fkbp12, Qdpr And Compound 4
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.39 Å Release Date: 2025-10-08 Classification: LIGASE Ligands: GOL, CL, A1BB9 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-10-08
Ligands: GOL, CL, A1BB9
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Co-Crystal Structure Of The Ternary Complex Of Human Fkbp12, Brd9 Bromo Domain And Compound 1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.01 Å Release Date: 2025-10-08 Classification: LIGASE Ligands: A1BB8, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-10-08
Ligands: A1BB8, GOL
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Crystal Structure Of The Catalytic Domain Of Human Pkc Alpha (D463N, V568I, S657E) In Complex With Nvp-Cjl037 At 2.48-A Resolution
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.48 Å Release Date: 2024-01-24 Classification: TRANSFERASE/INHIBITOR Ligands: V5U, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-01-24
Ligands: V5U, MG
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Crystal Structure Of The Catalytic Domain Of Human Pkc Alpha (D463N, V568I, S657E) In Complex With Darovasertib (Nvp-Lxs196) At 2.82-A Resolution
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.82 Å Release Date: 2024-01-24 Classification: TRANSFERASE/INHIBITOR Ligands: W39 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-01-24
Ligands: W39
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Structure Of Complement C5 In Complex With Small Molecule Inhibitor And Cvf
Organism: Homo sapiens, Naja kaouthia
Method: ELECTRON MICROSCOPY Release Date: 2022-12-21 Classification: IMMUNE SYSTEM Ligands: H1H, MG |
Organism: Homo sapiens, Naja kaouthia
Method: ELECTRON MICROSCOPY
Release Date: 2022-12-21
Ligands: H1H, MG
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Bruton'S Tyrosine Kinase In Complex With Compound 45
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2022-05-18 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 0B9 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-05-18
Ligands: 0B9
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Bruton'S Tyrosine Kinase In Complex With Compound 21
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.62 Å Release Date: 2022-05-18 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 0BG, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-05-18
Ligands: 0BG, DMS
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Bruton'S Tyrosine Kinase In Complex With Compound 65
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2022-05-18 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 0B0 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-05-18
Ligands: 0B0
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Brutons Tyrosine Kinase In Complex With Compound 50.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.72 Å Release Date: 2019-06-12 Classification: transferase/transferase inhibitor Ligands: L9S, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-06-12
Ligands: L9S, EDO
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Apo Structure Of Wt Lipoprotein Lipase In Complex With Gpihbp1 Mutant N78D N82D Produced In Gnti-Deficient Hek293-F Cells
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.48 Å Release Date: 2019-05-08 Classification: HYDROLASE/PROTEIN BINDING Ligands: NAG, MLI, CA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-05-08
Ligands: NAG, MLI, CA
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Apo Structure Of Wt Lipoprotein Lipase In Complex With Gpihbp1 Mutant N78D N82D Produced In Hek293-F Cells
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.04 Å Release Date: 2019-05-08 Classification: HYDROLASE/PROTEIN BINDING Ligands: NAG, EDO, CA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-05-08
Ligands: NAG, EDO, CA
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Compound 2 Bound Structure Of Wt Lipoprotein Lipase In Complex With Gpihbp1 Mutant N78D N82D Produced In Hek293-F Cells
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.81 Å Release Date: 2019-05-08 Classification: HYDROLASE/PROTEIN BINDING Ligands: NAG, M3D, EDO, CA, TRS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-05-08
Ligands: NAG, M3D, EDO, CA, TRS
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Crystal Structure Of An Extender (Spd28345)-Modified Human Pdk1 Complex 2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.50 Å Release Date: 2011-04-20 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SYP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-04-20
Ligands: SYP
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Pdk1 In Complex With Dfg-Out Inhibitor Xxx
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2011-04-20 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: MP7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-04-20
Ligands: MP7
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Crystal Structure Of Human Caspase-1 With A Naturally-Occurring Arg240->Gln Substitution In Complex With 3-[2-(2-Benzyloxycarbonylamino-3-Methyl-Butyrylamino)-Propionylamino]-4-Oxo-Pentanoic Acid (Z-Vad-Fmk)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2010-03-02 Classification: HYDROLASE/HYDROLASE INHIBITOR |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-03-02
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Crystal Structure Of Human Caspase-1 With A Naturally-Occurring Asn263->Ser Substitution In Complex With 3-[2-(2-Benzyloxycarbonylamino-3-Methyl-Butyrylamino)-Propionylamino]-4-Oxo-Pentanoic Acid (Z-Vad-Fmk)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2010-03-02 Classification: HYDROLASE/HYDROLASE INHIBITOR |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-03-02
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Crystal Structure Of Human Caspase-1 With A Naturally-Occurring Lys319->Arg Substitution In Complex With 3-[2-(2-Benzyloxycarbonylamino-3-Methyl-Butyrylamino)-Propionylamino]-4-Oxo-Pentanoic Acid (Z-Vad-Fmk)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2010-03-02 Classification: HYDROLASE/HYDROLASE INHIBITOR |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-03-02
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The 1.6 A Crystal Structure Of Human Bruton'S Tyrosine Kinase Bound To A Pyrrolopyrimidine-Containing Compound
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2010-01-19 Classification: TRANSFERASE Ligands: B43 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-01-19
Ligands: B43
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Structures Of Human Bruton'S Tyrosine Kinase In Active And Inactive Conformations Suggests A Mechanism Of Activation For Tec Family Kinases.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.94 Å Release Date: 2010-01-19 Classification: TRANSFERASE Ligands: 1N1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-01-19
Ligands: 1N1
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Crystal Structure Of Mouse Aurora A (Asn186->Gly, Lys240->Arg, Met302->Leu) In Complex With 1-(3-Chloro-Phenyl)-3-{5-[2-(Thieno[3,2-D]Pyrimidin-4-Ylamino)- Ethyl]-Thiazol-2-Yl}-Urea [Sns-314]
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2009-05-12 Classification: TRANSFERASE Ligands: AK2 |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2009-05-12
Ligands: AK2