Search Count: 23
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Potent And Selective Phosphodiesterase 10A Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2012-09-05 Classification: Hydrolase/Hydrolase inhibitor Ligands: ZN, MG, 0T7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-09-05
Ligands: ZN, MG, 0T7
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Potent And Selective Phosphodiesterase 10A Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.02 Å Release Date: 2012-09-05 Classification: Hydrolase/Hydrolase inhibitor Ligands: ZN, MG, 0T6 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-09-05
Ligands: ZN, MG, 0T6
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Highly Potent, Selective, And Orally Active Phosphodiestarase 10A Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.82 Å Release Date: 2011-10-26 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: CL, 540, ZN, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-10-26
Ligands: CL, 540, ZN, MG
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Highly Potent, Selective, And Orally Active Phosphodiestarase 10A Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2011-10-26 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: ZN, MG, CL, 546 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-10-26
Ligands: ZN, MG, CL, 546
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Highly Potent, Selective, And Orally Active Phosphodiestarase 10A Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2011-10-26 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: ZN, MG, 548 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-10-26
Ligands: ZN, MG, 548
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Bace1 In Complex With The Aminohydantoin Compound 102
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2011-08-31 Classification: hydrolase/hydrolase inhibitor Ligands: ZOO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-08-31
Ligands: ZOO
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Pyrazolyl And Thienyl Aminohydantoins As Potent Bace1 Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.16 Å Release Date: 2011-08-31 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 591 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-08-31
Ligands: 591
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Pyrazolyl And Thienyl Aminohydantoins As Potent Bace1 Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2011-08-31 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 532 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-08-31
Ligands: 532
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Bace1 In Complex With The Aminopyridine Compound 44
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2010-04-28 Classification: HYDROLASE Ligands: 879 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-04-28
Ligands: 879
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Bace-1 With The Aminopyridine Compound 32
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.36 Å Release Date: 2010-04-28 Classification: HYDROLASE Ligands: 625 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-04-28
Ligands: 625
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Bace1 In Complex With The Aminohydantoin Compound 4G
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2010-04-21 Classification: HYDROLASE Ligands: Z81 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-04-21
Ligands: Z81
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Bace1 With The Aminohydantoin Compound 29
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.25 Å Release Date: 2010-03-02 Classification: HYDROLASE Ligands: 593 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-03-02
Ligands: 593
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Bace1 With The Aminohydantoin Compound S-34
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2010-03-02 Classification: HYDROLASE Ligands: X17 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-03-02
Ligands: X17
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Bace1 With The Aminohydantoin Compound 37
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2010-03-02 Classification: HYDROLASE Ligands: X45 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-03-02
Ligands: X45
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Bace1 With The Aminohydantoin Compound R-58
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2010-03-02 Classification: HYDROLASE Ligands: 569 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-03-02
Ligands: 569
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Bace1 With Compound 30
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2010-01-19 Classification: HYDROLASE Ligands: 472 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-01-19
Ligands: 472
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Bace1 With Compound 38
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2010-01-19 Classification: HYDROLASE Ligands: BX2 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-01-19
Ligands: BX2
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3,4-Dihydropyrimido(1,2-A)Indol-10(2H)-Ones As Potent Non-Peptidic Inhibitors Of Caspase-3
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2009-11-17 Classification: HYDROLASE Ligands: H0E |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-11-17
Ligands: H0E
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Bace-1 With Compound 3
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.24 Å Release Date: 2009-11-03 Classification: HYDROLASE Ligands: 454 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-11-03
Ligands: 454
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X-Ray Structure Of Bace-1 In Complex With Compound 3.B.10
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2008-12-09 Classification: HYDROLASE Ligands: 310 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-12-09
Ligands: 310
