Search Count: 19
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Crystal Structure Of The Acvr1 (Alk2) Kinase Domain In Complex With Inhibitor Cdd-2789
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.72 Å Release Date: 2024-11-27 Classification: TRANSFERASE Ligands: GOL, A1A29, PO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-11-27
Ligands: GOL, A1A29, PO4
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Crystal Structure Of The Acvr1 (Alk2) Kinase Domain In Complex With Inhibitor Cdd-2281
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.86 Å Release Date: 2024-11-27 Classification: TRANSFERASE Ligands: PO4, GOL, A1A3C |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-11-27
Ligands: PO4, GOL, A1A3C
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Crystal Structure Of The Acvr1 (Alk2) Kinase Domain In Complex With Inhibitor Cdd-2282
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2024-11-27 Classification: TRANSFERASE Ligands: A1A3D, PO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-11-27
Ligands: A1A3D, PO4
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Crystal Structure Of Serine/Threonine-Protein Kinase 33 (Stk33) Kinase Domain In Complex With Inhibitor Cdd-2211
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2024-06-05 Classification: CYTOSOLIC PROTEIN Ligands: A1AAY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-06-05
Ligands: A1AAY
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Crystal Structure Of Coq8A-Ca157 Inhibitor Complex In Space Group C2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.01 Å Release Date: 2023-01-18 Classification: TRANSFERASE Ligands: MVS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-01-18
Ligands: MVS
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Crystal Structure Of Coq8A-Ca157 Inhibitor Complex In Space Group P1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2023-01-18 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: MVS, NA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-01-18
Ligands: MVS, NA
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X-Ray Structure Of Danio Rerio Histone Deacetylase 6 (Hdac6) Cd2 In Complex With An Inhibitor Sw101
Organism: Danio rerio
Method: X-RAY DIFFRACTION Resolution:1.13 Å Release Date: 2021-08-04 Classification: HYDROLASE Ligands: ZN, QRB, GOL, K, SCN |
Organism: Danio rerio
Method: X-RAY DIFFRACTION
Release Date: 2021-08-04
Ligands: ZN, QRB, GOL, K, SCN
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Egfr(T790M/V948R) In Complex With Ln3844
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.76 Å Release Date: 2021-05-19 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: UEJ, ANP, MG, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-05-19
Ligands: UEJ, ANP, MG, CL
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Crystal Structure Of Egfr(T790M/V948R) In Complex With Ln3753
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2021-03-31 Classification: TRANSFERASE Ligands: TOV, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-03-31
Ligands: TOV, CL
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A Crystal Structure Of Egfr(T790M/V948R) In Complex With Ln3754
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2021-03-31 Classification: TRANSFERASE Ligands: ANP, MG, TQA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-03-31
Ligands: ANP, MG, TQA
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X-Ray Structure Of Danio Rerio Histone Deacetylase 6 (Hdac6) Cd2 In Complex With A Inhibitor Ss208
Organism: Danio rerio
Method: X-RAY DIFFRACTION Resolution:1.15 Å Release Date: 2019-10-09 Classification: HYDROLASE Ligands: ZN, K, JNN, SCN |
Organism: Danio rerio
Method: X-RAY DIFFRACTION
Release Date: 2019-10-09
Ligands: ZN, K, JNN, SCN
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Glycogen Synthase Kinase 3 Beta Complexed With Brd0209
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2018-03-14 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 6VK |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-03-14
Ligands: 6VK
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Glycogen Synthase Kinase 3 Beta Complexed With Brd0705
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2018-03-14 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 6VL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-03-14
Ligands: 6VL
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Glycogen Synthase Kinase 3 Beta Complexed With Brd3731
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.69 Å Release Date: 2018-03-14 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 6VM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-03-14
Ligands: 6VM
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Exploiting An Asp-Glu Switch In Glycogen Synthase Kinase 3 To Design Paralog Selective Inhibitors For Use In Acute Myeloid Leukemia
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.85 Å Release Date: 2018-02-21 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: 6VL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-02-21
Ligands: 6VL
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Crystal Structure Of Jak3 In Complex With Compound 4 (Fm381)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.55 Å Release Date: 2016-10-26 Classification: TRANSFERASE Ligands: 79T, PHU, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-10-26
Ligands: 79T, PHU, EDO
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Crystal Structure Of Jak3 In Complex With Compound 5 (Fm409)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2016-10-26 Classification: TRANSFERASE Ligands: PHU, EDO, 79R, 79S |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-10-26
Ligands: PHU, EDO, 79R, 79S
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Bivalent Binding To Bet Bromodomains
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.01 Å Release Date: 2016-09-28 Classification: TRANSCRIPTION Ligands: ETU |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-09-28
Ligands: ETU
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Bivalent Binding To Bet Bromodomains
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.49 Å Release Date: 2016-09-28 Classification: TRANSCRIPTION Ligands: K6K |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-09-28
Ligands: K6K