Search Count: 13
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Crystal Structure Of Crbn-Ddb1 And Mrt-3486 In Complex With Nek7
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.25 Å Release Date: 2025-07-09 Classification: DNA Binding Protein/Transferase Ligands: A1BX6, ZN, ADP, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-07-09
Ligands: A1BX6, ZN, ADP, MG
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Crystal Structure Of Crbn-Ddb1 And Mrt-23227 In Complex With Vav1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.40 Å Release Date: 2025-07-09 Classification: LIGASE Ligands: ZN, A1BYX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-07-09
Ligands: ZN, A1BYX
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Crystal Structure Of Crbn-Ddb1 And Fpft-2216 In Complex With Mtor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.95 Å Release Date: 2025-07-09 Classification: DNA Binding Protein/Transferase Ligands: ZN, A1BC8 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-07-09
Ligands: ZN, A1BC8
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Discovery Of Lu Af11167, A Phosphodiesterase 10A Inhibitor Clinical Candidate
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2023-04-19 Classification: HYDROLASE Ligands: ZN, MG, EFJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-04-19
Ligands: ZN, MG, EFJ
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Discovery Of Lu Af11167, A Phosphodiesterase 10A Inhibitor Clinical Candidate
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2023-04-19 Classification: HYDROLASE Ligands: EEI, ZN, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-04-19
Ligands: EEI, ZN, MG
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Discovery Of Lu Af11167, A Phosphodiesterase 10A Inhibitor Clinical Candidate
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2023-04-19 Classification: HYDROLASE Ligands: ZN, MG, EIH |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-04-19
Ligands: ZN, MG, EIH
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Discovery Of Lu Af11167, A Phosphodiesterase 10A Inhibitor Clinical Candidate
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2023-04-19 Classification: HYDROLASE Ligands: ZN, MG, EHI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-04-19
Ligands: ZN, MG, EHI
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Discovery Of Lu Af11167, A Phosphodiesterase 10A Inhibitor Clinical Candidate
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.45 Å Release Date: 2023-04-19 Classification: HYDROLASE Ligands: EIK, ZN, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-04-19
Ligands: EIK, ZN, MG
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Fragment-Based Discovery Of Pyrazolopyridones As Jak1 Inhibitors With Excellent Subtype Selectivity
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.99 Å Release Date: 2020-06-10 Classification: TRANSFERASE Ligands: QZ8 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-06-10
Ligands: QZ8
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Fragment-Based Discovery Of Pyrazolopyridones As Jak1 Inhibitors With Excellent Subtype Selectivity
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.87 Å Release Date: 2020-06-10 Classification: TRANSFERASE Ligands: NTW |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-06-10
Ligands: NTW
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Fragment-Based Discovery Of Pyrazolopyridones As Jak1 Inhibitors With Excellent Subtype Selectivity
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.31 Å Release Date: 2020-06-10 Classification: TRANSFERASE Ligands: NTQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-06-10
Ligands: NTQ
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Fragment-Based Discovery Of 6-Arylindazole Jak Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.98 Å Release Date: 2016-04-27 Classification: TRANSFERASE Ligands: 6DP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-04-27
Ligands: 6DP
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Triazoloquinazolines As A Novel Class Of Phosphodiesterase 10A (Pde10A) Inhibitors, Part 2, Lead-Optimisation.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.43 Å Release Date: 2011-06-15 Classification: HYDROLASE Ligands: AXC, ZN, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-06-15
Ligands: AXC, ZN, MG
