Search Count: 12
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Human B-Raf Kinase Domain Bound To A Type Ii Pyrazolopyridine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.50 Å Release Date: 2012-11-14 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 0WP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-11-14
Ligands: 0WP
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B-Raf V600E Kinase Domain Bound To A Type Ii Dihydroquinazoline Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.20 Å Release Date: 2012-11-14 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: B1E |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-11-14
Ligands: B1E
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Crystal Structure Of B-Raf Kinase Domain In Complex With A Dihydropyrido[2,3-D]Pyrimidinone-Based Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.60 Å Release Date: 2012-05-09 Classification: Transferase/Transferase Inhibitor Ligands: T1Q |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-05-09
Ligands: T1Q
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Human B-Raf Kinase Domain In Complex With An Bromopyridine Benzamide Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.40 Å Release Date: 2011-10-05 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: TV4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-10-05
Ligands: TV4
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Human B-Raf Kinase Domain In Complex With A Methoxypyrazolopyridinyl Benzamide Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.30 Å Release Date: 2011-10-05 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: B0R |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-10-05
Ligands: B0R
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Human B-Raf Kinase In Complex With An Amide Linked Pyrazolopyridine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.20 Å Release Date: 2011-08-17 Classification: Transferase/Transferase Inhibitor Ligands: BR2 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-08-17
Ligands: BR2
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Spirocyclic Sulfonamides As Akt Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2011-04-06 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SM9 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-04-06
Ligands: SM9
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Spirochromane Akt Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2011-03-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SMH |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-03-30
Ligands: SMH
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Spirochromane Akt Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2011-03-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SMR |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-03-30
Ligands: SMR
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Discovery Of Dihydrothieno- And Dihydrofuropyrimidines As Potent Pan Akt Inhibitors
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2010-11-10 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: SMY |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2010-11-10
Ligands: SMY
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Discovery Of Dihydrothieno- And Dihydrofuropyrimidines As Potent Pan Akt Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2010-11-10 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: SMY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-11-10
Ligands: SMY
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Akt1 Kinase Domain With Pyrrolopyrimidine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2010-09-15 Classification: TRANSFERASE Ligands: XM1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-09-15
Ligands: XM1
