Search Count: 28
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Pi3Ka H1047R Co-Crystal Structure With Inhibitor In Cryptic Pocket Near H1047R (Compound 4).
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.58 Å Release Date: 2024-03-20 Classification: SIGNALING PROTEIN Ligands: YO4, YNZ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-03-20
Ligands: YO4, YNZ
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Pi3Ka H1047R Co-Crystal Structure With Inhibitor In Cryptic Pocket (Compound 5).
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.20 Å Release Date: 2024-03-20 Classification: SIGNALING PROTEIN Ligands: YOR, YNZ, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-03-20
Ligands: YOR, YNZ, CL
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Pi3Ka H1047R Co-Crystal Structure With Inhibitors In Two Cryptic Pockets (Compounds 4 And 5).
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.35 Å Release Date: 2024-03-20 Classification: SIGNALING PROTEIN Ligands: YO4, YOR, YNZ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-03-20
Ligands: YO4, YOR, YNZ
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Pi3Ka H1047R Co-Crystal Structure With Inhibitor In Cryptic Pocket Near H1047R (Compound 12).
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.93 Å Release Date: 2024-03-20 Classification: SIGNALING PROTEIN Ligands: 1LT, YQB |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-03-20
Ligands: 1LT, YQB
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Pi3Ka H1047R Co-Crystal Structure With Inhibitor In Cryptic Pocket Near H1047R (Compound 7).
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.61 Å Release Date: 2024-03-20 Classification: SIGNALING PROTEIN Ligands: YQ2, 1LT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-03-20
Ligands: YQ2, 1LT
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Prmt5/Mep50 Crystal Structure With Sinefungin Bound
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.21 Å Release Date: 2022-03-16 Classification: TRANSFERASE/INHIBITOR Ligands: SFG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-03-16
Ligands: SFG
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Prmt5/Mep50 Crystal Structure With Mta And Phthalazinone Fragment Bound
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.01 Å Release Date: 2022-01-26 Classification: TRANSFERASE Ligands: CL, NA, EDO, 81X, MTA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-01-26
Ligands: CL, NA, EDO, 81X, MTA
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Prmt5/Mep50 Crystal Structure With Mta And A Phthalazinone Inhibitor Bound (Compound 9)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.78 Å Release Date: 2022-01-26 Classification: TRANSFERASE/INHIBITOR Ligands: MTA, 84W |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-01-26
Ligands: MTA, 84W
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Prmt5/Mep50 Crystal Structure With Mta And A Phthalazinone Inhibitor Bound (Compound (M)-31)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2022-01-26 Classification: TRANSFERASE/INHIBITOR Ligands: MTA, 85E |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-01-26
Ligands: MTA, 85E
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Prmt5/Mep50 Crystal Structure With Mta And Mrtx-1719 Bound
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.62 Å Release Date: 2022-01-26 Classification: TRANSFERASE/INHIBITOR Ligands: MTA, 85K |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-01-26
Ligands: MTA, 85K
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Prmt5/Mep50 With Compound 30 Bound
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.14 Å Release Date: 2022-01-26 Classification: TRANSFERASE/INHIBITOR Ligands: 97L, MTA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-01-26
Ligands: 97L, MTA
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Prmt5/Mep50 With Compound 29 Bound
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2022-01-26 Classification: TRANSFERASE/INHIBITOR Ligands: 97X, MTA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-01-26
Ligands: 97X, MTA
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Crystal Structure Of Mnk2-D228G In Complex With Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2018-05-09 Classification: TRANSFERASE/TRANSFERASE Inhibitor Ligands: ZN, F4G |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-05-09
Ligands: ZN, F4G
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Crystal Structure Of Mnk2-D228G In Complex With Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.36 Å Release Date: 2018-05-09 Classification: Transferase/Transferase Inhibitor Ligands: ZN, F4A |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-05-09
Ligands: ZN, F4A
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Co-Crystal Structure Of Mnk2 In Complex With An Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.60 Å Release Date: 2018-05-09 Classification: TRANSFERASE/TRANSFERASE Inhibitor Ligands: ZN, ET8 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-05-09
Ligands: ZN, ET8
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Crystal Structure Of Mnk2-D228G In Complex With Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.38 Å Release Date: 2018-05-09 Classification: TRANSFERASE/TRANSFERASE Inhibitor Ligands: ZN, FYV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-05-09
Ligands: ZN, FYV
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Crystal Structure Of Mnk2-D228G In Complex With Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.05 Å Release Date: 2018-05-09 Classification: TRANSFERASE/TRANSFERASE Inhibitor Ligands: ZN, F4J |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-05-09
Ligands: ZN, F4J
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Co-Crytsal Structure Of Mnk2 In Complex With An Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2018-05-09 Classification: TRANSFERASE/TRANSFERASE Inhibitor Ligands: ZN, F67, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-05-09
Ligands: ZN, F67, CL
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Crystal Structure Of Mnk2-D228G In Complex With Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.32 Å Release Date: 2018-05-09 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ZN, N45 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-05-09
Ligands: ZN, N45
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Co-Crystal Structure Of Mnk2 In Complex With Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.95 Å Release Date: 2018-05-09 Classification: TRANSFERASE/TRANSFERASE Inhibitor Ligands: ZN, FZJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-05-09
Ligands: ZN, FZJ
