Search Count: 19
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Crystal Structure Of Ternary Complex Of Pol Theta Polymerase Domain
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:2.26 Å Release Date: 2022-10-12 Classification: TRANSFERASE Ligands: MG, DG3 |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2022-10-12
Ligands: MG, DG3
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Crystal Structure Of Pol Theta Polymerase Domain In Complex With Compound 5
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:2.99 Å Release Date: 2022-10-12 Classification: TRANSFERASE Ligands: MG, DG3, K7X |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2022-10-12
Ligands: MG, DG3, K7X
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Crystal Structure Of Pol Theta Polymerase Domain In Complex With Compound 22
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:2.83 Å Release Date: 2022-10-12 Classification: TRANSFERASE Ligands: MG, DG3, K8I |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2022-10-12
Ligands: MG, DG3, K8I
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Erk5 In Complex With A Pyrrole Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.38 Å Release Date: 2018-06-20 Classification: TRANSFERASE Ligands: 9N8, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-06-20
Ligands: 9N8, DMS
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Brd4 In Complex With Erk5 Inhibitor Xmd8-92
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2017-08-30 Classification: TRANSCRIPTION Ligands: 4WG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-08-30
Ligands: 4WG
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Human Pfkfb3 In Complex With An Indole Inhibitor 1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.01 Å Release Date: 2015-04-22 Classification: TRANSFERASE Ligands: PO4, 8R2, FDP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-04-22
Ligands: PO4, 8R2, FDP
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Human Pfkfb3 In Complex With An Indole Inhibitor 2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2015-04-22 Classification: TRANSFERASE Ligands: PHS, PO4, F6P, S6L |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-04-22
Ligands: PHS, PO4, F6P, S6L
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Human Pfkfb3 In Complex With An Indole Inhibitor 3
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.58 Å Release Date: 2015-04-22 Classification: TRANSFERASE Ligands: PHS, PO4, F6P, FD9 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-04-22
Ligands: PHS, PO4, F6P, FD9
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Human Pfkfb3 In Complex With An Indole Inhibitor 4
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.37 Å Release Date: 2015-04-22 Classification: TRANSFERASE Ligands: PHS, PO4, F6P, 87T |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-04-22
Ligands: PHS, PO4, F6P, 87T
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Human Pfkfb3 In Complex With An Indole Inhibitor 5
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.35 Å Release Date: 2015-04-22 Classification: TRANSFERASE Ligands: PHS, F6P, PO4, MJP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-04-22
Ligands: PHS, F6P, PO4, MJP
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Human Pfkfb3 In Complex With An Indole Inhibitor 6
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.03 Å Release Date: 2015-04-22 Classification: TRANSFERASE Ligands: PHS, PO4, F6P, 8V1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-04-22
Ligands: PHS, PO4, F6P, 8V1
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Crystal Structure Of Human 17Beta-Hydroxysteroid Dehydrogenase Type 5 In Complex With (4-(4-Chlorophenyl)Piperazin-1-Yl)(Morpholino)Methanone (24)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2013-11-13 Classification: Oxidoreductase/Oxidoreductase inhibitor Ligands: NAP, 16J, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-11-13
Ligands: NAP, 16J, EDO
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Crystal Structure Of Human 17Beta-Hydroxysteroid Dehydrogenase Type 5 In Complex With 1-{4-[(2-Methyl-1-Piperidinyl)Sulfonyl]Phenyl}-2-Pyrrolidinone
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.97 Å Release Date: 2013-03-20 Classification: oxidoreductase/oxidoreductase inhibitor Ligands: NAP, 10H |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-03-20
Ligands: NAP, 10H
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Crystal Structure Of Human 17Beta-Hydroxysteroid Dehydrogenase Type 5 In Complex With (R)-1-(Naphthalen-2-Ylsulfonyl)Piperidine-3-Carboxylic Acid (86)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2012-10-10 Classification: OXIDOREDUCTASE/OXIDOREDUCTASE inhibitor Ligands: NAP, 0SL, EDO, ACT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-10-10
Ligands: NAP, 0SL, EDO, ACT
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Crystal Structure Of Human 17Beta-Hydroxysteroid Dehydrogenase Type 5 In Complex With 3-((3,4-Dihydroisoquinolin-2(1H)-Yl)Sulfonyl)-N-Methylbenzamide (80)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2012-10-10 Classification: oxidoreductase/oxidoreductase inhibitor Ligands: NAP, 0T0, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-10-10
Ligands: NAP, 0T0, EDO
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Crystal Structure Of Human 17Beta-Hydroxysteroid Dehydrogenase Type 5 In Complex With 3-((3,4-Dihydroisoquinolin-2(1H)-Yl)Sulfonyl)Benzoic Acid (17)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2012-10-10 Classification: oxidoreductase/oxidoreductase inhibitor Ligands: NAP, 0SZ, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-10-10
Ligands: NAP, 0SZ, EDO
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Crystal Structure Of Chk2 In Complex With An Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2011-01-12 Classification: TRANSFERASE Ligands: XBJ, MG, NO3 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-01-12
Ligands: XBJ, MG, NO3
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Co-Crystal Structure Of A Small Molecule Inhibitor Bound To The Kinase Domain Of Chk2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.40 Å Release Date: 2011-01-12 Classification: TRANSFERASE Ligands: B4W |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-01-12
Ligands: B4W
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Structure Of A Small Molecule Inhibitor With The Kinase Domain Of Chk2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2011-01-12 Classification: TRANSFERASE Ligands: LWH, NO3 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-01-12
Ligands: LWH, NO3
