Search Count: 12
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Crystal Structure Of Ksr1:Mek1 In Complex With Amp-Pnp, And Allosteric Mek Inhibitor Cobimetinib
Organism: Homo sapiens, Oryctolagus cuniculus
Method: X-RAY DIFFRACTION Resolution:3.10 Å Release Date: 2020-10-07 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ANP, MG, EUI |
Organism: Homo sapiens, Oryctolagus cuniculus
Method: X-RAY DIFFRACTION
Release Date: 2020-10-07
Ligands: ANP, MG, EUI
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Crystal Structure Of Ksr2:Mek1 In Complex With Adp
Organism: Homo sapiens, Oryctolagus cuniculus
Method: X-RAY DIFFRACTION Resolution:3.22 Å Release Date: 2020-09-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ADP, MG |
Organism: Homo sapiens, Oryctolagus cuniculus
Method: X-RAY DIFFRACTION
Release Date: 2020-09-30
Ligands: ADP, MG
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Crystal Structure Of Ksr2:Mek1 In Complex With Amp-Pnp, And Allosteric Mek Inhibitor Trametinib
Organism: Homo sapiens, Oryctolagus cuniculus
Method: X-RAY DIFFRACTION Resolution:2.82 Å Release Date: 2020-09-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ANP, MG, QOM |
Organism: Homo sapiens, Oryctolagus cuniculus
Method: X-RAY DIFFRACTION
Release Date: 2020-09-30
Ligands: ANP, MG, QOM
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Crystal Structure Of Ksr2:Mek1 In Complex With Amp-Pnp, And Allosteric Mek Inhibitor Cobimetinib
Organism: Homo sapiens, Oryctolagus cuniculus
Method: X-RAY DIFFRACTION Resolution:2.99 Å Release Date: 2020-09-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ANP, MG, VKD |
Organism: Homo sapiens, Oryctolagus cuniculus
Method: X-RAY DIFFRACTION
Release Date: 2020-09-30
Ligands: ANP, MG, VKD
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Crystal Structure Of Ksr2:Mek1 In Complex With Anp-Pnp, And Allosteric Mek Inhibitor Selumetinib
Organism: Homo sapiens, Oryctolagus cuniculus
Method: X-RAY DIFFRACTION Resolution:3.09 Å Release Date: 2020-09-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ANP, 3EW |
Organism: Homo sapiens, Oryctolagus cuniculus
Method: X-RAY DIFFRACTION
Release Date: 2020-09-30
Ligands: ANP, 3EW
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Crystal Structure Of Ksr2:Mek1 In Complex With Amp-Pnp, And Allosteric Mek Inhibitor Pd0325901
Organism: Homo sapiens, Oryctolagus cuniculus
Method: X-RAY DIFFRACTION Resolution:3.19 Å Release Date: 2020-09-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ANP, MG, 4BM |
Organism: Homo sapiens, Oryctolagus cuniculus
Method: X-RAY DIFFRACTION
Release Date: 2020-09-30
Ligands: ANP, MG, 4BM
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Crystal Structure Of Ksr2:Mek1 In Complex With Amp-Pnp, And Allosteric Mek Inhibitor Aps-9-95-1
Organism: Homo sapiens, Oryctolagus cuniculus
Method: X-RAY DIFFRACTION Resolution:3.36 Å Release Date: 2020-09-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ANP, MG, VKG |
Organism: Homo sapiens, Oryctolagus cuniculus
Method: X-RAY DIFFRACTION
Release Date: 2020-09-30
Ligands: ANP, MG, VKG
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Crystal Structure Of Ksr1:Mek1 In Complex With Amp-Pnp
Organism: Homo sapiens, Oryctolagus cuniculus
Method: X-RAY DIFFRACTION Resolution:2.88 Å Release Date: 2020-09-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ANP, MG |
Organism: Homo sapiens, Oryctolagus cuniculus
Method: X-RAY DIFFRACTION
Release Date: 2020-09-30
Ligands: ANP, MG
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Crystal Structure Of Ksr1:Mek1 In Complex With Amp-Pnp, And Allosteric Mek Inhibitor Trametinib
Organism: Homo sapiens, Oryctolagus cuniculus
Method: X-RAY DIFFRACTION Resolution:3.34 Å Release Date: 2020-09-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ANP, MG, QOM |
Organism: Homo sapiens, Oryctolagus cuniculus
Method: X-RAY DIFFRACTION
Release Date: 2020-09-30
Ligands: ANP, MG, QOM
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Crystal Structure Of Ksr1:Mek1 In Complex With Amp-Pnp, And Allosteric Mek Inhibitor Selumetinib
Organism: Homo sapiens, Oryctolagus cuniculus
Method: X-RAY DIFFRACTION Resolution:3.21 Å Release Date: 2020-09-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ANP, 3EW |
Organism: Homo sapiens, Oryctolagus cuniculus
Method: X-RAY DIFFRACTION
Release Date: 2020-09-30
Ligands: ANP, 3EW
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Crystal Structure Of Ksr1:Mek1 In Complex With Amp-Pnp, And Allosteric Mek Inhibitor Pd0325901
Organism: Homo sapiens, Oryctolagus cuniculus
Method: X-RAY DIFFRACTION Resolution:3.63 Å Release Date: 2020-09-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ANP, MG, 4BM |
Organism: Homo sapiens, Oryctolagus cuniculus
Method: X-RAY DIFFRACTION
Release Date: 2020-09-30
Ligands: ANP, MG, 4BM
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Crystal Structure Of Ksr1:Mek1 In Complex With Amp-Pnp, And Allosteric Mek Inhibitor Aps-9-95-1
Organism: Homo sapiens, Oryctolagus cuniculus
Method: X-RAY DIFFRACTION Resolution:3.62 Å Release Date: 2020-09-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ANP, MG, VKG |
Organism: Homo sapiens, Oryctolagus cuniculus
Method: X-RAY DIFFRACTION
Release Date: 2020-09-30
Ligands: ANP, MG, VKG
