Search Count: 27
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Crystal Structure Of Human Dcaf1 Wd40 Repeats (Q1250L) In Complex With Compound 1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2023-06-14 Classification: TRANSFERASE Ligands: EDO, ACT, LQH |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-06-14
Ligands: EDO, ACT, LQH
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Crystal Structure Of Human Dcaf1 Wd40 Repeats (Q1250L) In Complex With Compound 1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.25 Å Release Date: 2023-06-14 Classification: TRANSFERASE Ligands: LQH, ACT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-06-14
Ligands: LQH, ACT
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Crystal Structure Of Human Dcaf1 Wd40 Repeats (Q1250L) In Complex With Compound 2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.64 Å Release Date: 2023-06-14 Classification: TRANSFERASE Ligands: ACT, EDO, VMR |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-06-14
Ligands: ACT, EDO, VMR
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Crystal Structure Of Human Dcaf1 Wd40 Repeats (Q1250L) In Complex With Compound 3
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.11 Å Release Date: 2023-06-14 Classification: TRANSFERASE Ligands: VM8, ACT, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-06-14
Ligands: VM8, ACT, EDO
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Crystal Structure Of Human Dcaf1 Wd40 Repeats (Q1250L) In Complex With Compound 4
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.95 Å Release Date: 2023-06-14 Classification: TRANSFERASE Ligands: VM3 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-06-14
Ligands: VM3
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Crystal Structure Of Human Dcaf1 Wd40 Repeats (Q1250L) In Complex With Compound 6
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2023-06-14 Classification: TRANSFERASE Ligands: EDO, DMS, VLW |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-06-14
Ligands: EDO, DMS, VLW
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Crystal Structure Of Human Dcaf1 Wd40 Repeats (Q1250L) In Complex With Compound 8
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.27 Å Release Date: 2023-06-14 Classification: TRANSFERASE Ligands: EDO, VN5, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-06-14
Ligands: EDO, VN5, DMS
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Crystal Structure Of Human Dcaf1 Wd40 Repeats (Q1250L) In Complex With Compound 11
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.09 Å Release Date: 2023-06-14 Classification: TRANSFERASE Ligands: DMS, MG, ACT, EDO, VMZ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-06-14
Ligands: DMS, MG, ACT, EDO, VMZ
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Human Malt1(329-729) In Complex With A Chromane Urea Containing Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.32 Å Release Date: 2020-12-09 Classification: HYDROLASE Ligands: RJK |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-12-09
Ligands: RJK
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Human Malt1(329-729) In Complex With A Chromane Urea Containing Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.51 Å Release Date: 2020-12-09 Classification: HYDROLASE Ligands: RJH, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-12-09
Ligands: RJH, MG
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Crystal Structure Of Jak2-V617F Pseudokinase Domain In Complex With Compound 2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2019-03-27 Classification: TRANSFERASE Ligands: EKT, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-03-27
Ligands: EKT, EDO
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Jak2 Pseudokinase V617F In Complex With At9283
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.19 Å Release Date: 2019-03-20 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 35R |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-03-20
Ligands: 35R
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Jak2 Pseudokinase In Complex With Nu6140
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.04 Å Release Date: 2018-08-01 Classification: TRANSFERASE Ligands: AQG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-08-01
Ligands: AQG
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Jak2 Pseudokinase In Complex With Bi-D1870
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2018-08-01 Classification: TRANSFERASE Ligands: 584 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-08-01
Ligands: 584
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Jak2 Pseudokinase In Complex With Azd7762
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2018-08-01 Classification: TRANSFERASE Ligands: YDJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-08-01
Ligands: YDJ
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Jak2 Pseudokinase In Complex With At9283
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.55 Å Release Date: 2018-08-01 Classification: TRANSFERASE Ligands: 35R |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-08-01
Ligands: 35R
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Jak2 Pseudokinase In Complex With Jnj7706621
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.38 Å Release Date: 2018-08-01 Classification: TRANSFERASE Ligands: SKE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-08-01
Ligands: SKE
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Structural Basis Of Jak2 Inhibition By The Type Ii Inhibtor Nvp-Bbt594
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.34 Å Release Date: 2012-05-16 Classification: Transferase/transferase inhibitor Ligands: 046, MLI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-05-16
Ligands: 046, MLI
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Crystal Structure Of Jak2 Complexed With A Potent Quinoxaline Atp Site Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2010-07-21 Classification: TRANSFERASE Ligands: DQX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-07-21
Ligands: DQX
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Crystal Structure Of Jak2 Complexed With A Potent 2,8-Diaryl-Quinoxaline Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2010-04-28 Classification: TRANSFERASE Ligands: NVB |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-04-28
Ligands: NVB
