Search Count: 13
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Crystal Structure Of Ternary Complex Helios-Zf2:Crbn:Ddb1 In Complex With Bms-986449, A Molecular Glue Degrader
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.53 Å Release Date: 2026-09-02 Classification: LIGASE Ligands: ZN, A1CSO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-09-02
Ligands: ZN, A1CSO
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Crystal Structure Of Casein Kinase 2 (Ck2) Alpha In Complex With Bms-595
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.96 Å Release Date: 2026-06-10 Classification: TRANSFERASE Ligands: A1DAS, MN, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-06-10
Ligands: A1DAS, MN, CL
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Crystal Structure Of Rar-Related Orphan Receptor C (Nhis-Rorgt(244-487)-L6-Src1(678-692)) In Complex With {3,5-Dichloro-4-[4-Methoxy-3-(Propan-2-Yl)Phenoxy]Phenyl}Methanol
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.62 Å Release Date: 2021-01-20 Classification: TRANSFERASE/Agonist Ligands: Z7G |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-01-20
Ligands: Z7G
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Crystal Structure Of Rar-Related Orphan Receptor C (Nhis-Rorgt(244-487)-L6-Src1(678-692)) In Complex With {3,5-Dichloro-4-[4-Methoxy-3-(Propan-2-Yl)Phenoxy]Phenyl}Methanol
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.42 Å Release Date: 2021-01-20 Classification: TRANSFERASE/Agonist Ligands: Z7H |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-01-20
Ligands: Z7H
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Crystal Structure Of Rar-Related Orphan Receptor C (Nhis-Rorgt(244-487)-L6-Src1(678-692)) In Complex With {3,5-Dichloro-4-[4-Methoxy-3-(Propan-2-Yl)Phenoxy]Phenyl}Methanol
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.14 Å Release Date: 2021-01-20 Classification: TRANSFERASE/Agonist Ligands: Z7I |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-01-20
Ligands: Z7I
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Crystal Structure Of Janus Kinase 2 In Complex With N,N-Dicyclopropyl-10-Ethyl-7-[(3-Methoxypropyl)Amino] -3-Methyl-3,5,8,10-Tetraazatricyclo[7.3.0.0,6] Dodeca-1(9),2(6),4,7,11-Pentaene-11-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.38 Å Release Date: 2015-08-26 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 50Y |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-08-26
Ligands: 50Y
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Crystal Structure Of Janus Kinase 2 In Complex With N,N-Dicyclopropyl-7-[(Dimethyl-1,3-Thiazol-2-Yl)Amino]-10-Ethyl-3-Methyl-3,5,8,10-Tetraazatricyclo[7.3.0.02,6] Dodeca-1(9),2(6),4,7,11-Pentaene-11-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.45 Å Release Date: 2015-08-26 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 50W |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-08-26
Ligands: 50W
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Crystal Structure Of Janus Kinase 2 In Complex With N,N-Dicyclopropyl-10-[(2S)-2,3-Dihydroxypropyl]-3-Methyl-7-(Methylamino)-3,5,8,10-Tetraazatricyclo [7.3.0.02,6]Dodeca-1(9),2(6),4,7,11-Pentaene-11-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2015-08-26 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 50O |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-08-26
Ligands: 50O
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Crystal Structure Of Janus Kinase 2 In Complex With N,N-Dicyclopropyl-10-Ethyl-7-[(3-Methoxypropyl)Amino] -3-Methyl-3,5,8,10-Tetraazatricyclo[7.3.0.0,6] Dodeca-1(9),2(6),4,7,11-Pentaene-11-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2015-08-26 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 50V |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-08-26
Ligands: 50V
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Crystal Structure Of Janus Kinase 2 In Complex With A 9H-Carbazole-1-Carboxamide Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.65 Å Release Date: 2015-06-03 Classification: Transferase/Transferase Inhibitor Ligands: 4OK |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-06-03
Ligands: 4OK
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Crystal Structure Of Coactivator Associated Arginine Methyltransferase 1 (Carm1) In Complex With Sinefungin And Indole Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2011-03-23 Classification: TRANSFERASE Ligands: SFG, 849 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-03-23
Ligands: SFG, 849
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Crystal Structure Of Coactivator Associated Arginine Methyltransferase 1 (Carm1) In Complex With Sinefungin And Indole Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2011-03-23 Classification: TRANSFERASE Ligands: SAH, 845, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-03-23
Ligands: SAH, 845, CL
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Structure Of Janus Kinase 2 With A Pyrrolotriazine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2011-02-16 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: J2I |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-02-16
Ligands: J2I
