Search Count: 12
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Human Wee1 Kinase In Complex With Inhibitor 1-[6-(1-Hydroxy-1-Methyl-Ethyl)-Pyridin-2-Yl]-2-(2-Methoxy-Phenyl)-6-[4-(4-Methyl-Piperazin-1-Yl)-Phenylamino]-1,2-Dihydro-Pyrazolo[3,4-D]Pyrimidin-3-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.53 Å Release Date: 2023-05-31 Classification: TRANSFERASE Ligands: QT9 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-05-31
Ligands: QT9
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Structure Of Human Plk1 In Complex With 2-Allyl-1-[6-(1-Hydroxy-1-Methyl-Ethyl)-Pyridin-2-Yl]-6-[4-(4-Methyl-Piperazin-1-Yl)-Phenylamino]-1,2-Dihydro-Pyrazolo[3,4-D]Pyrimidin-3-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.19 Å Release Date: 2023-04-26 Classification: TRANSFERASE Ligands: ACT, 8X7, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-04-26
Ligands: ACT, 8X7, ZN
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P70 S6K1 In Complex With Msc2317067A-1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.00 Å Release Date: 2022-07-06 Classification: TRANSFERASE/INHIBITOR Ligands: 1RJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-07-06
Ligands: 1RJ
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P70 S6K1 In Complex With Msc2363318A-1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.74 Å Release Date: 2022-07-06 Classification: TRANSFERASE/INHIBITOR Ligands: 1SK |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-07-06
Ligands: 1SK
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Btk1 Soaked With Compound 5, Y551 Is Sequestered
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.84 Å Release Date: 2021-05-19 Classification: TRANSFERASE Ligands: X9J, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-05-19
Ligands: X9J, DMS
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Btk1 Soaked With Compound 5, Y551 Is Sequestered
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.33 Å Release Date: 2021-05-19 Classification: TRANSFERASE Ligands: X9M |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-05-19
Ligands: X9M
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Btk1 Soaked With Compound 26
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.34 Å Release Date: 2021-05-19 Classification: TRANSFERASE Ligands: X9P, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-05-19
Ligands: X9P, DMS
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Btk1 Soaked With Compound 24
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.94 Å Release Date: 2021-05-19 Classification: TRANSFERASE Ligands: X9S, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-05-19
Ligands: X9S, DMS
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Btk1 Soaked With Compound 25
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.83 Å Release Date: 2021-05-19 Classification: TRANSFERASE Ligands: X9V, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-05-19
Ligands: X9V, DMS
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Btk1 Soaked With Compound 30
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.38 Å Release Date: 2021-05-19 Classification: TRANSFERASE Ligands: DMS, X9Y |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-05-19
Ligands: DMS, X9Y
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Structure Of Human Bruton'S Tyrosine Kinase In Complex With Evobrutinib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.41 Å Release Date: 2019-08-14 Classification: Transferase/Transferase Inhibitor Ligands: CL, MZJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-08-14
Ligands: CL, MZJ
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Discovery Of Affinity-Based Probes For Btk Occupancy Assay
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.23 Å Release Date: 2019-02-06 Classification: IMMUNE SYSTEM Ligands: KHD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-02-06
Ligands: KHD
